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- [1] Design and Synthesis of Novel Lactate Dehydrogenase A Inhibitors by Fragment-Based Lead GenerationJOURNAL OF MEDICINAL CHEMISTRY, 2012, 55 (07) : 3285 - 3306Ward, Richard A.Brassington, ClaireBreeze, Alexander L.Caputo, AlessandroCritchlow, SusanDavies, GarethGoodwin, LouiseHassall, GilesGreenwood, RyanHoldgate, Geoffrey A.Mrosek, MichaelNorman, Richard A.Pearson, StuartTart, JonathanTucker, Julie A.Vogtherr, MartinWhittaker, DavidWingfield, JonathanWinter, JonHudson, Kevin
- [2] Identification of novel non-nucleoside reverse transcriptase inhibitors using fragment-based lead generationMEDICINAL CHEMISTRY RESEARCH, 2005, 14 (8-9) : 475 - 487Ramajayam, R.Giridhar, RajaniYadav, M. R.De Clercq, ErickPannecouque, ChristophePrajapati, Dhaval G.
- [3] Identification of novel p38α MAP kinase inhibitors using fragment-based lead generationJOURNAL OF MEDICINAL CHEMISTRY, 2005, 48 (02) : 414 - 426Gill, ALFrederickson, MCleasby, AWoodhead, SJCarr, MGWoodhead, AJWalker, MTCongreve, MSDevine, LATisi, DO'Reilly, MSeavers, LCADavis, DJCurry, JAnthony, RPadova, AMurray, CWCarr, RAEJhoti, H
- [4] Identification of Novel Non-nucleoside Reverse Transcriptase Inhibitors Using Fragment-based Lead GenerationMedicinal Chemistry Research, 2005, 14 : 475 - 487R. RamajayamRajani GiridharM. R. YadavErick De ClercqChristophe PannecouqueDhaval G. Prajapati
- [5] Identification of inhibitors of protein kinase B using fragment-based lead discoveryJOURNAL OF MEDICINAL CHEMISTRY, 2007, 50 (10) : 2293 - 2296Saxty, GordonWoodhead, Steven J.Berdini, ValerioDavies, Thomas G.Verdonk, Marcel L.Wyatt, Paul G.Boyle, Robert G.Barford, DavidDownham, RobertGarrett, Michelle D.Carr, Robin A.
- [6] Fragment-Based Lead Identification of Selective Inhibitors of a Key Metabolic EnzymeFASEB JOURNAL, 2011, 25Arachea, Buenafe T.Gao, GengPavlovsky, Alexander G.Viola, Ronald E.
- [7] Fragment-based identification of phosphatase inhibitorsABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2009, 238Rawls, KatherineSoellner, MatthewTakeuchi, JunImamura, ShinichiBaguley, TylerGrundner, ChristophAlber, TomEllman, Jonathan A.
- [8] Fragment-based lead generation: identification of seed fragments by a highly efficient fragment screening technologyJOURNAL OF COMPUTER-AIDED MOLECULAR DESIGN, 2009, 23 (08) : 501 - 511Neumann, LarsRitscher, AllegraMueller, GerhardHafenbradl, Doris
- [9] Fragment-based lead generation: identification of seed fragments by a highly efficient fragment screening technologyJournal of Computer-Aided Molecular Design, 2009, 23 : 501 - 511Lars NeumannAllegra RitscherGerhard MüllerDoris Hafenbradl
- [10] Fragment-Based Identification of Influenza Endonuclease InhibitorsJOURNAL OF MEDICINAL CHEMISTRY, 2016, 59 (13) : 6444 - 6454Credille, Cy V.Chen, YaoCohen, Seth M.