Synthesis of substituted maleimide derivatives using the Baylis-Hillman adducts

被引：0
|
作者：
Basavaiah, Deevi [1 ]
Lenin, Dandamudi V. [1 ]
Veeraraghavaiah, Gorre [1 ]
机构：
[1] Univ Hyderabad, Sch Chem, Hyderabad 500046, Andhra Pradesh, India
来源：
CURRENT SCIENCE | 2011年 / 101卷 / 07期
关键词：
Baylis-Hillman adducts; cyclization; Friedel Crafts reaction; pyrrole-2,5-diones; alpha-keto esters; ALPHA-KETO ESTERS; ONE-POT SYNTHESIS; BIOLOGICAL EVALUATION; FRAMEWORKS;
D O I：
暂无
中图分类号：
O [数理科学和化学]; P [天文学、地球科学]; Q [生物科学]; N [自然科学总论];
学科分类号：
07 ; 0710 ; 09 ;
摘要：
The Baylis-Hillman alcohols, 3-ethoxycarbonyl-3-hydroxy-3-aryl(alkyl)-2-methylenepropanenitriles, derived from alpha-keto esters and acrylonitrile, have been conveniently transformed into 3,4-disubstituted 1H-pyrrole-2,5-dione (maleimide) derivatives on treatment with FeCl3/RCO2H in a one-pot operation.
引用
收藏
页码：888 / 893
页数：6
相关论文
共 50 条
  • [1] Synthesis of substituted uracil derivatives from the acetates of the Baylis-Hillman adducts
    Lee, CG
    Gowrisankar, S
    Kim, JN
    BULLETIN OF THE KOREAN CHEMICAL SOCIETY, 2005, 26 (03) : 481 - 484
  • [2] The first successful intermolecular Heck reaction of Baylis-Hillman adducts:: synthesis of β-aryl substituted Baylis-Hillman adducts
    Kim, Jeong Mi
    Kim, Ko Hoon
    Kim, Taek Hyeon
    Kim, Jae Nyoung
    TETRAHEDRON LETTERS, 2008, 49 (20) : 3248 - 3251
  • [3] An expedient synthesis of β-phenyl substituted Baylis-Hillman and Aza-Baylis-Hillman adducts
    Kim, Seong Jin
    Lee, Hyun Seung
    Kim, Jeong Mi
    Kim, Jae Nyoung
    BULLETIN OF THE KOREAN CHEMICAL SOCIETY, 2008, 29 (01): : 265 - 268
  • [4] Diastereoselective peroxidation of derivatives of Baylis-Hillman adducts
    Zuckerman, Dylan S.
    Woerpel, K. A.
    TETRAHEDRON, 2019, 75 (31) : 4118 - 4129
  • [5] Baylis-Hillman reaction and chemical transformations of Baylis-Hillman adducts
    Lee, KY
    Gowrisankar, S
    Kim, JN
    BULLETIN OF THE KOREAN CHEMICAL SOCIETY, 2005, 26 (10): : 1481 - 1490
  • [6] An efficient synthesis of Baylis-Hillman adducts of acrylamide: Pd-catalyzed hydration of Baylis-Hillman adducts of acrylonitrile
    Kim, Eun Sun
    Lee, Hyun Seung
    Kim, Jae Nyoung
    TETRAHEDRON LETTERS, 2009, 50 (46) : 6286 - 6289
  • [7] Baylis-Hillman adducts as an important synthon for the synthesis of α-carbolinone and α-carboline derivatives
    Lenin, Dandamudi V.
    Malvi, Payal
    JOURNAL OF HETEROCYCLIC CHEMISTRY, 2023, 60 (06) : 957 - 965
  • [8] Synthesis of iodoenol lactone derivatives from the Baylis-Hillman adducts using lodolactonization protocol
    GowriSankar, S
    Lee, MJ
    Lee, S
    Kim, JN
    BULLETIN OF THE KOREAN CHEMICAL SOCIETY, 2004, 25 (12) : 1963 - 1965
  • [9] Deracemization of Baylis-Hillman adducts
    Trost, Barry M.
    Tsui, Hon-Chung
    Toste, F. Dean
    1600, ACS, Washington, DC, USA (122):
  • [10] Arylation of the Baylis-Hillman adducts
    Basavaiah, D
    Muthukumaran, K
    TETRAHEDRON, 1998, 54 (19) : 4943 - 4948
12345