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- [1] GNE-064: A Potent, Selective, and Orally Bioavailable Chemical Probe for the Bromodomains of SMARCA2 and SMARCA4 and the Fifth Bromodomain of PBRM1JOURNAL OF MEDICINAL CHEMISTRY, 2022, 65 (16) : 11177 - 11186Taylor, Alexander M.论文数: 0 引用数: 0 h-index: 0机构: Constellation, Cambridge, MA 02142 USA Constellation, Cambridge, MA 02142 USABailey, Chris论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Constellation, Cambridge, MA 02142 USABelmont, Lisa D.论文数: 0 引用数: 0 h-index: 0机构: Constellation, Cambridge, MA 02142 USA Constellation, Cambridge, MA 02142 USACampbell, Robert论文数: 0 引用数: 0 h-index: 0机构: Constellation, Cambridge, MA 02142 USA Constellation, Cambridge, MA 02142 USACantone, Nico论文数: 0 引用数: 0 h-index: 0机构: Constellation, Cambridge, MA 02142 USA Constellation, Cambridge, MA 02142 USACote, Alexandre论文数: 0 引用数: 0 h-index: 0机构: Constellation, Cambridge, MA 02142 USA Constellation, Cambridge, MA 02142 USACrawford, Terry D.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Constellation, Cambridge, MA 02142 USACummings, Richard论文数: 0 引用数: 0 h-index: 0机构: Constellation, Cambridge, MA 02142 USA Constellation, Cambridge, MA 02142 USADeMent, Kevin论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Constellation, Cambridge, MA 02142 USADuplessis, Martin论文数: 0 引用数: 0 h-index: 0机构: Constellation, Cambridge, MA 02142 USA Constellation, Cambridge, MA 02142 USAFlynn, Megan论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Constellation, Cambridge, MA 02142 USAGood, Andrew C.论文数: 0 引用数: 0 h-index: 0机构: Constellation, Cambridge, MA 02142 USA Constellation, Cambridge, MA 02142 USAHuang, Hon-Ren论文数: 0 引用数: 0 h-index: 0机构: Constellation, Cambridge, MA 02142 USA Constellation, Cambridge, MA 02142 USAJoshi, Shivangi论文数: 0 引用数: 0 h-index: 0机构: Constellation, Cambridge, MA 02142 USA Constellation, Cambridge, MA 02142 USALeblanc, Yves论文数: 0 引用数: 0 h-index: 0机构: Constellation, Cambridge, MA 02142 USA Constellation, Cambridge, MA 02142 USAMurray, Jeremy论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Constellation, Cambridge, MA 02142 USANasveschuk, Christopher G.论文数: 0 引用数: 0 h-index: 0机构: Constellation, Cambridge, MA 02142 USA Constellation, Cambridge, MA 02142 USANeiss, Adrianne论文数: 0 引用数: 0 h-index: 0机构: Constellation, Cambridge, MA 02142 USA Constellation, Cambridge, MA 02142 USAPoy, Florence论文数: 0 引用数: 0 h-index: 0机构: Constellation, Cambridge, MA 02142 USA Constellation, Cambridge, MA 02142 USARomero, F. Anthony论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Constellation, Cambridge, MA 02142 USASandy, Peter论文数: 0 引用数: 0 h-index: 0机构: Constellation, Cambridge, MA 02142 USA Constellation, Cambridge, MA 02142 USATang, Yong论文数: 0 引用数: 0 h-index: 0机构: Constellation, Cambridge, MA 02142 USA Constellation, Cambridge, MA 02142 USATsui, Vickie论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Constellation, Cambridge, MA 02142 USAZawadzke, Laura论文数: 0 引用数: 0 h-index: 0机构: Constellation, Cambridge, MA 02142 USA Constellation, Cambridge, MA 02142 USASims, Robert J., III论文数: 0 引用数: 0 h-index: 0机构: Constellation, Cambridge, MA 02142 USA Constellation, Cambridge, MA 02142 USAAudia, James E.论文数: 0 引用数: 0 h-index: 0机构: Constellation, Cambridge, MA 02142 USA Flare Therapeut, 215 First St,Suite 150, Cambridge, MA 02142 USA Constellation, Cambridge, MA 02142 USABellon, Steven F.论文数: 0 引用数: 0 h-index: 0机构: Constellation, Cambridge, MA 02142 USA Constellation, Cambridge, MA 02142 USAMagnuson, Steven R.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Constellation, Cambridge, MA 02142 USAAlbrecht, Brian K.论文数: 0 引用数: 0 h-index: 0机构: Constellation, Cambridge, MA 02142 USA Constellation, Cambridge, MA 02142 USACochran, Andrea G.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Constellation, Cambridge, MA 02142 USA
- [2] Frequent co-inactivation of the SWI/SNF subunits SMARCB1, SMARCA2 and PBRM1 in malignant rhabdoid tumoursHISTOPATHOLOGY, 2015, 67 (01) : 121 - 129Rao, Qiu论文数: 0 引用数: 0 h-index: 0机构: Nanjing Univ, Sch Med, Dept Pathol, Nanjing Jinling Hosp, Nanjing 210002, Jiangsu, Peoples R China Nanjing Univ, Sch Med, Dept Pathol, Nanjing Jinling Hosp, Nanjing 210002, Jiangsu, Peoples R ChinaXia, Qiu-yuan论文数: 0 引用数: 0 h-index: 0机构: Nanjing Univ, Sch Med, Dept Pathol, Nanjing Jinling Hosp, Nanjing 210002, Jiangsu, Peoples R China Nanjing Univ, Sch Med, Dept Pathol, Nanjing Jinling Hosp, Nanjing 210002, Jiangsu, Peoples R ChinaWang, Zi-yu论文数: 0 引用数: 0 h-index: 0机构: Nanjing Univ Tradit Chinese Med, Sch Basic Med Sci, Nanjing, Jiangsu, Peoples R China Nanjing Univ, Sch Med, Dept Pathol, Nanjing Jinling Hosp, Nanjing 210002, Jiangsu, Peoples R ChinaLi, Li论文数: 0 引用数: 0 h-index: 0机构: Nanjing Univ, Sch Med, Dept Pathol, Nanjing Jinling Hosp, Nanjing 210002, Jiangsu, Peoples R China Nanjing Univ, Sch Med, Dept Pathol, Nanjing Jinling Hosp, Nanjing 210002, Jiangsu, Peoples R ChinaShen, Qin论文数: 0 引用数: 0 h-index: 0机构: Nanjing Univ, Sch Med, Dept Pathol, Nanjing Jinling Hosp, Nanjing 210002, Jiangsu, Peoples R China Nanjing Univ, Sch Med, Dept Pathol, Nanjing Jinling Hosp, Nanjing 210002, Jiangsu, Peoples R ChinaShi, Shan-shan论文数: 0 引用数: 0 h-index: 0机构: Nanjing Univ, Sch Med, Dept Pathol, Nanjing Jinling Hosp, Nanjing 210002, Jiangsu, Peoples R China Nanjing Univ, Sch Med, Dept Pathol, Nanjing Jinling Hosp, Nanjing 210002, Jiangsu, Peoples R ChinaWang, Xuan论文数: 0 引用数: 0 h-index: 0机构: Nanjing Univ, Sch Med, Dept Pathol, Nanjing Jinling Hosp, Nanjing 210002, Jiangsu, Peoples R China Nanjing Univ, Sch Med, Dept Pathol, Nanjing Jinling Hosp, Nanjing 210002, Jiangsu, Peoples R ChinaLiu, Biao论文数: 0 引用数: 0 h-index: 0机构: Nanjing Univ, Sch Med, Dept Pathol, Nanjing Jinling Hosp, Nanjing 210002, Jiangsu, Peoples R China Nanjing Univ, Sch Med, Dept Pathol, Nanjing Jinling Hosp, Nanjing 210002, Jiangsu, Peoples R ChinaWang, Yan-fen论文数: 0 引用数: 0 h-index: 0机构: Nanjing Univ, Sch Med, Dept Pathol, Nanjing Jinling Hosp, Nanjing 210002, Jiangsu, Peoples R China Nanjing Univ, Sch Med, Dept Pathol, Nanjing Jinling Hosp, Nanjing 210002, Jiangsu, Peoples R ChinaShi, Qun-li论文数: 0 引用数: 0 h-index: 0机构: Nanjing Univ, Sch Med, Dept Pathol, Nanjing Jinling Hosp, Nanjing 210002, Jiangsu, Peoples R China Nanjing Univ, Sch Med, Dept Pathol, Nanjing Jinling Hosp, Nanjing 210002, Jiangsu, Peoples R ChinaMa, Heng-hui论文数: 0 引用数: 0 h-index: 0机构: Nanjing Univ, Sch Med, Dept Pathol, Nanjing Jinling Hosp, Nanjing 210002, Jiangsu, Peoples R China Nanjing Univ, Sch Med, Dept Pathol, Nanjing Jinling Hosp, Nanjing 210002, Jiangsu, Peoples R ChinaLu, Zhen-feng论文数: 0 引用数: 0 h-index: 0机构: Nanjing Univ, Sch Med, Dept Pathol, Nanjing Jinling Hosp, Nanjing 210002, Jiangsu, Peoples R China Nanjing Univ, Sch Med, Dept Pathol, Nanjing Jinling Hosp, Nanjing 210002, Jiangsu, Peoples R ChinaHe, Yan论文数: 0 引用数: 0 h-index: 0机构: Nanjing Univ, Sch Med, Dept Pathol, Nanjing Jinling Hosp, Nanjing 210002, Jiangsu, Peoples R China Nanjing Univ, Sch Med, Dept Pathol, Nanjing Jinling Hosp, Nanjing 210002, Jiangsu, Peoples R ChinaZhang, Ru-song论文数: 0 引用数: 0 h-index: 0机构: Nanjing Univ, Sch Med, Dept Pathol, Nanjing Jinling Hosp, Nanjing 210002, Jiangsu, Peoples R China Nanjing Univ, Sch Med, Dept Pathol, Nanjing Jinling Hosp, Nanjing 210002, Jiangsu, Peoples R ChinaYu, Bo论文数: 0 引用数: 0 h-index: 0机构: Nanjing Univ, Sch Med, Dept Pathol, Nanjing Jinling Hosp, Nanjing 210002, Jiangsu, Peoples R China Nanjing Univ, Sch Med, Dept Pathol, Nanjing Jinling Hosp, Nanjing 210002, Jiangsu, Peoples R ChinaZhou, Xiao-jun论文数: 0 引用数: 0 h-index: 0机构: Nanjing Univ, Sch Med, Dept Pathol, Nanjing Jinling Hosp, Nanjing 210002, Jiangsu, Peoples R China Nanjing Univ, Sch Med, Dept Pathol, Nanjing Jinling Hosp, Nanjing 210002, Jiangsu, Peoples R China
- [3] The impact of PBRM1 mutations on overall survival in greater than 2,100 patients treated with immune checkpoint blockade (ICB).JOURNAL OF CLINICAL ONCOLOGY, 2019, 37 (07)Hakimi, A. Ari论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USA Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAGed, Yasser论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USA Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAFlynn, Jessica论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USA Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAHoen, Douglas R.论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USA Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USADi Natale, Renzo G.论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USA Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USABlum, Kyle A.论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USA Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAMakarov, Vladimir论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USA Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAKuo, Fengshen论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USA Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USACarlo, Maria Isabel论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USA Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USALee, Chung-Han论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USA Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAVoss, Martin Henner论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USA Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAOstrovnaya, Irina论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USA Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAChan, Timothy An-thy论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USA Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAMotzer, Robert J.论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USA Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USA
- [4] Aberrant promoter hypermethylation of PBRM1, BAP1, SETD2, KDM6A and other chromatin-modifying genes is absent or rare in clear cell RCCEPIGENETICS, 2013, 8 (05) : 486 - 493Ibragimova, Ilsiya论文数: 0 引用数: 0 h-index: 0机构: Fox Chase Canc Ctr, Canc Epigenet Program, Philadelphia, PA 19111 USA Fox Chase Canc Ctr, Kidney Keystone Program, Philadelphia, PA 19111 USA Fox Chase Canc Ctr, Canc Epigenet Program, Philadelphia, PA 19111 USAMaradeo, Marie E.论文数: 0 引用数: 0 h-index: 0机构: Fox Chase Canc Ctr, Canc Epigenet Program, Philadelphia, PA 19111 USA Fox Chase Canc Ctr, Kidney Keystone Program, Philadelphia, PA 19111 USA Fox Chase Canc Ctr, Canc Epigenet Program, Philadelphia, PA 19111 USADulaimi, Essel论文数: 0 引用数: 0 h-index: 0机构: Fox Chase Canc Ctr, Kidney Keystone Program, Philadelphia, PA 19111 USA Fox Chase Canc Ctr, Dept Pathol, Philadelphia, PA 19111 USA Fox Chase Canc Ctr, Canc Epigenet Program, Philadelphia, PA 19111 USACairns, Paul论文数: 0 引用数: 0 h-index: 0机构: Fox Chase Canc Ctr, Canc Epigenet Program, Philadelphia, PA 19111 USA Fox Chase Canc Ctr, Kidney Keystone Program, Philadelphia, PA 19111 USA Fox Chase Canc Ctr, Canc Epigenet Program, Philadelphia, PA 19111 USA