Potent and orally bioavailable stearoyl-CoA desaturase (SCD) inhibitors based on the pyrrolo[1,2-f][1,2,4]triazin-4(3H)-one scaffold

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|
作者：
Parkhill, Eric Q. [1 ]
Koltun, Dmitry [1 ]
Brunn, Sandra A. [2 ]
Mollova, Nevena [3 ]
Leung, Kwan [3 ]
Chisholm, Jeffrey W. [2 ]
Zablocki, Jeff [1 ]
机构：
[1] CV Therapeut, Dept Bioorgan Chem, Palo Alto, CA 94304 USA
[2] CV Therapeut, Dept Pharmacol Sci, Palo Alto, CA 94304 USA
[3] CV Therapeut, Dept Preclin Dev, Palo Alto, CA 94304 USA
来源：
ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY | 2009年 / 238卷
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中图分类号：
O6 [化学];
学科分类号：
0703 ;
摘要：
147-MEDI
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页数：1
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