nBu4NI-catalyzed C3-formylation of indoles with N-methylaniline

被引：98
|
作者：
Li, Lan-Tao [1 ,2 ]
Huang, Juan [1 ,2 ]
Li, Hong-Ying [1 ,2 ]
Wen, Li-Juan [1 ,2 ]
Wang, Peng [1 ,2 ]
Wang, Bin [1 ,2 ]
机构：
[1] Nankai Univ, Coll Pharm, State Key Lab Med Chem Biol, Tianjin 300071, Peoples R China
[2] Nankai Univ, Tianjin Key Lab Mol Drug Res, Tianjin 300071, Peoples R China
来源：
CHEMICAL COMMUNICATIONS | 2012年 / 48卷 / 42期
基金：
中国国家自然科学基金;
关键词：
STUDIEN ZUM ABLAUF; BETA-KETO-ESTERS; MOLECULAR-OXYGEN; OXIDATION; DIBENZOYLPEROXYD; SUBSTITUTION; ACTIVATION; CATALYSIS; IODINE; CORE;
D O I：
10.1039/c2cc31578e
中图分类号：
O6 [化学];
学科分类号：
0703 ;
摘要：
nBu(4)NI-catalyzed C3-selective formylation of N-H and N-substituted indoles by using N-methylaniline as a formylating reagent was first successfully demonstrated.
引用
收藏
页码：5187 / 5189
页数：3
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