5-HT6 MEDICINAL CHEMISTRY

被引:64
|
作者
Liu, Kevin G. [1 ]
Robichaud, Albert J. [1 ]
机构
[1] Lundbeck Res USA, Paramus, NJ 07652 USA
来源
关键词
ATYPICAL ANTIPSYCHOTIC AGENTS; SEROTONIN RECEPTOR-BINDING; BRAIN PENETRANT; ANTISENSE OLIGONUCLEOTIDES; BIOLOGICAL EVALUATION; ALZHEIMERS-DISEASE; H5-HT6; RECEPTORS; HIGH-AFFINITY; RO; 04-6790; ANTAGONISTS;
D O I
10.1016/B978-0-12-384976-2.00001-0
中图分类号
Q189 [神经科学];
学科分类号
071006 ;
摘要
引用
收藏
页码:1 / 34
页数:34
相关论文
共 50 条
  • [1] The Medicinal Chemistry of 5-HT6 Receptor Ligands with a Focus on Arylsulfonyltryptamine Analogs
    Glennon, Richard A.
    Siripurapu, Uma
    Roth, Bryan L.
    Kolanos, Renata
    Bondarev, Mikhail L.
    Sikazwe, Donald
    Lee, Mase
    Dukat, Malgorzata
    CURRENT TOPICS IN MEDICINAL CHEMISTRY, 2010, 10 (05) : 579 - 595
  • [2] Medicinal chemistry approaches toward novel, selective 5-HT6 receptor ligands
    Holenz, J.
    Pauwels, P. J.
    Diaz, J. L.
    Merce, R.
    Codony, X.
    Buschmann, H.
    JOURNAL OF PHARMACOLOGICAL SCIENCES, 2006, 101 : 51 - 51
  • [3] Medicinal chemistry driven approaches toward novel and selective serotonin 5-HT6 receptor ligands
    Holenz, J
    Mercè, R
    Díaz, JL
    Guitart, X
    Codony, X
    Dordal, A
    Romero, G
    Torrens, A
    Mas, J
    Andaluz, B
    Hernández, S
    Monroy, X
    Sánchez, E
    Hernández, E
    Pérez, R
    Cubí, R
    Sanfeliu, O
    Buschmann, H
    JOURNAL OF MEDICINAL CHEMISTRY, 2005, 48 (06) : 1781 - 1795
  • [4] Medicinal chemistry strategies to 5-HT6 receptor ligands as potential cognitive enhancers and antiobesity agents
    Holenz, J
    Pauwels, PJ
    Díaz, JL
    Mercè, R
    Codony, X
    Buschmann, H
    DRUG DISCOVERY TODAY, 2006, 11 (7-8) : 283 - 299
  • [5] 5-ht6 Receptors
    Woolley, Marie L.
    Marsden, Charles A.
    Fone, Kevin C. F.
    CNS & NEUROLOGICAL DISORDERS-DRUG TARGETS, 2004, 3 (01) : 59 - 79
  • [6] ELECTROPHYSIOLOGY OF 5-HT6 RECEPTORS
    Tassone, Annalisa
    Madeo, Graziella
    Sciamanna, Giuseppe
    Pisani, Antonio
    Bonsi, Paola
    PHARMACOLOGY OF 5-HT6 RECEPTORS, PT 1, 2010, 94 : 111 - 128
  • [7] 5-HT5与5-HT6受体
    曹文辉
    国外医学(分子生物学分册), 1995, (02) : 86 - 88
  • [8] 5-HT6 pharmacology inconsistencies
    Borsini, Franco
    Bordi, Fabio
    Riccioni, Teresa
    PHARMACOLOGY BIOCHEMISTRY AND BEHAVIOR, 2011, 98 (02) : 169 - 172
  • [9] 5-HT6 receptor antagonist
    Lloyd, AW
    DRUG DISCOVERY TODAY, 1999, 4 (05) : 238 - 238
  • [10] 5-HT6 receptor and cognition
    Codony, Xabier
    Miguel Vela, Jose
    Javier Ramirez, Maria
    CURRENT OPINION IN PHARMACOLOGY, 2011, 11 (01) : 94 - 100