Synthesis and reactions of 6(4)-(P-benzylphenyl)-4(6)-phenylpyrimidine-2(1H) thione

被引：0
|
作者：
Wasfy, AAF
Amine, MS
Eissa, AMF
机构：
来源：
HETEROCYCLIC COMMUNICATIONS | 1996年 / 2卷 / 04期
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暂无
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
1,3-Diaryl-2-Propen-1-one reacted with thiourea in the presence of sodium ethoxide to furnish 4,6-diarylpyrimidine-2(1H) thione (2) under bar. The behaviour of (2) under bar towards nitrogen nucleophiles, and carbon electrophiles under Michael reaction conditions have been investigated. The oxidation of the thione (2) under bar gave the corresponding disulphide derivative <(12)under bar>. Acylation of (2) under bar yielded the corresponding S-acetyl-<(13)under bar> and N-benzoyl-<(14)under bar> derivatives, respectively.
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页码：375 / 381
页数：7
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