Rational design of inhibitors of human ecto-5′-nucleotidase

被引:0
|
作者
Pippel, J. [1 ]
Yates, K. [1 ]
Zebisch, M. [1 ]
Mueller, C. E. [2 ]
Straeter, N. [1 ]
机构
[1] Ctr Biotechnol & Biomed, Inst Bioanalyt Chem, D-04103 Leipzig, Germany
[2] Inst Pharmazeut, D-53121 Bonn, Germany
关键词
D O I
暂无
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:163 / 163
页数:1
相关论文
共 50 条
  • [1] Rational design of inhibitors for ecto-5′-nucleotidase (CD73)
    Pippel, Jan
    Knapp, Karen
    Zebisch, Matthias
    El-Tayeb, Ali
    Mueller, Christa E.
    Straeter, Norbert
    PURINERGIC SIGNALLING, 2014, 10 (04) : 767 - 767
  • [2] Be Aware of Aggregators in the Search for Potential Human ecto-5′-Nucleotidase Inhibitors
    Viviani, Lucas G.
    Piccirillo, Erika
    Cheffer, Arquimedes
    de Rezende, Leandro
    Ulrich, Henning
    Carmona-Ribeiro, Ana Maria
    T-do Amaral, Antonia
    MOLECULES, 2018, 23 (08)
  • [3] Isonicotinohydrazones as inhibitors of alkaline phosphatase and ecto-5′-nucleotidase
    Channar, Pervaiz Ali
    Shah, Syed Jawad Ali
    Hassan, Sidra
    Nisa, Zaib un
    Lecka, Joanna
    Sevigny, Jean
    Bajorath, Juergen
    Saeed, Aamer
    Iqbal, Jamshed
    CHEMICAL BIOLOGY & DRUG DESIGN, 2017, 89 (03) : 365 - 370
  • [4] CHARACTERIZATION OF THE HUMAN ECTO-5'-NUCLEOTIDASE PROMOTER
    HANSEN, KR
    RESTA, R
    WEBB, CF
    THOMPSON, LF
    FASEB JOURNAL, 1995, 9 (06): : A1461 - A1461
  • [5] ECTO-5'NUCLEOTIDASE ACTIVITY IN HUMAN MONOCLONAL GAMMOPATHIES
    MASSAIA, M
    BOCCADORO, M
    DIANZANI, U
    PIOPPO, P
    PILERI, A
    EXPERIMENTAL HEMATOLOGY, 1984, 12 (06) : 393 - 393
  • [6] REGULATION OF HUMAN LYMPHOBLAST ECTO-5'-NUCLEOTIDASE BY ZINC
    PILZ, RB
    WILLIS, RC
    WANLASS, S
    SEEGMILLER, JE
    ADVANCES IN EXPERIMENTAL MEDICINE AND BIOLOGY, 1984, 165 : 147 - 152
  • [7] Identification of sulfonic acids as efficient ecto-5′-nucleotidase inhibitors
    Iqbal, Jamshed
    Saeed, Aamer
    Raza, Rabia
    Matin, Abdul
    Hameed, Abdul
    Furtmann, Norbert
    Lecka, Joanna
    Sevigny, Jean
    Bajorath, Juergen
    EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2013, 70 : 685 - 691
  • [8] INDUCTION OF ECTO-5'-NUCLEOTIDASE ACTIVITY IN HUMAN THYMOCYTES
    COHEN, A
    DOSCH, HM
    GELFAND, EW
    CLINICAL IMMUNOLOGY AND IMMUNOPATHOLOGY, 1981, 18 (02): : 287 - 290
  • [9] ECTO-5'-NUCLEOTIDASE ACTIVITY IN THE HIPPOCAMPUS
    SEBASTIAO, AM
    CUNHA, RA
    RIBEIRO, JA
    JOURNAL OF NEUROCHEMISTRY, 1993, 61 : S181 - S181
  • [10] FUNCTIONAL-CHARACTERIZATION OF ECTO-5'-NUCLEOTIDASE-POSITIVE AND ECTO-5'-NUCLEOTIDASE-NEGATIVE HUMAN LYMPHOCYTE-T
    THOMPSON, LF
    RUEDI, JM
    JOURNAL OF IMMUNOLOGY, 1989, 142 (05): : 1518 - 1522