Stereo selective synthesis of 2-amino-1-hydroxy-3-phenylpropylphosphonic acid

被引：26
|
作者：
Zygmunt, J
Gancarz, R
Lejczak, B
Wieczorek, P
Kafarski, P
机构：
[1] WROCLAW TECH UNIV,INST ORGAN CHEM BIOCHEM & BIOTECHNOL,PL-50370 WROCLAW,POLAND
[2] UNIV OPOLE,INST CHEM,PL-45052 OPOLE,POLAND
来源：
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS | 1996年 / 6卷 / 24期
关键词：
D O I：
10.1016/S0960-894X(96)00545-8
中图分类号：
R914 [药物化学];
学科分类号：
100701 ;
摘要：
A highly stereoselective synthesis of 2-amino-1-hydroxy-3-phenylpropyl-phosphonic acid was achieved by simple addition of diethyl phosphite to enantiomeric N-blocked phenylalaninals. These compouds exhibit significant herbicidal activity. Copyright (C) 1996 Elsevier Science Ltd
引用
收藏
页码：2989 / 2992
页数：4
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