Synthesis of 2-dienylindole, SB 242784, by a three-component palladium-catalyzed coupling reaction

被引：46
|
作者：
Yu, MS [1 ]
de Leon, LL [1 ]
McGuire, MA [1 ]
Botha, G [1 ]
机构：
[1] SmithKline Beecham Pharmaceut, King Of Prussia, PA 19403 USA
来源：
TETRAHEDRON LETTERS | 1998年 / 39卷 / 51期
关键词：
D O I：
10.1016/S0040-4039(98)02161-3
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
The synthesis of SE 242784 using a novel one-pot Castro-Stephens-Suzuki reaction as the key reaction is described. (C) 1998 Elsevier Science Ltd. All rights reserved.
引用
收藏
页码：9347 / 9350
页数：4
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