共 50 条
- [1] Inhibitors of LSD1 as a potential therapy for acute myeloid leukemiaEXPERT OPINION ON INVESTIGATIONAL DRUGS, 2016, 25 (07) : 771 - 780Przespolewski, Amanda论文数: 0 引用数: 0 h-index: 0机构: Roswell Pk Canc Inst, Dept Med, Elm & Carlton St, Buffalo, NY 14263 USA Roswell Pk Canc Inst, Dept Med, Elm & Carlton St, Buffalo, NY 14263 USAWang, Eunice S.论文数: 0 引用数: 0 h-index: 0机构: Roswell Pk Canc Inst, Dept Med, Elm & Carlton St, Buffalo, NY 14263 USA Roswell Pk Canc Inst, Dept Med, Elm & Carlton St, Buffalo, NY 14263 USA
- [2] Discovery of reversible LSD1 inhibitorsABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2017, 254Kanouni, Toufike论文数: 0 引用数: 0 h-index: 0机构: Celgene, Chem, San Diego, CA USA Celgene, Chem, San Diego, CA USA
- [3] A comprehensive comparative study on LSD1 in different cancers and tumor specific LSD1 inhibitorsEUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2022, 240Dong, Jianshu论文数: 0 引用数: 0 h-index: 0机构: Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Key Lab Adv Drug Preparat Technol, Minist Educ, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Key Lab Henan Prov Drug Qual Control & Evaluat, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Inst Drug Discovery & Dev, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R China论文数: 引用数: h-index:机构:Tayyab, Bilal论文数: 0 引用数: 0 h-index: 0机构: Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Key Lab Adv Drug Preparat Technol, Minist Educ, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Key Lab Henan Prov Drug Qual Control & Evaluat, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Inst Drug Discovery & Dev, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R ChinaLi, Die论文数: 0 引用数: 0 h-index: 0机构: Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Key Lab Adv Drug Preparat Technol, Minist Educ, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Key Lab Henan Prov Drug Qual Control & Evaluat, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Inst Drug Discovery & Dev, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R ChinaKang, Lei论文数: 0 引用数: 0 h-index: 0机构: Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Key Lab Adv Drug Preparat Technol, Minist Educ, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Key Lab Henan Prov Drug Qual Control & Evaluat, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Inst Drug Discovery & Dev, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R ChinaZhang, Huimin论文数: 0 引用数: 0 h-index: 0机构: Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Key Lab Adv Drug Preparat Technol, Minist Educ, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Key Lab Henan Prov Drug Qual Control & Evaluat, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Collaborat Innovat Ctr New Drug Res & Safety Evalu, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Inst Drug Discovery & Dev, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R ChinaGong, Huimin论文数: 0 引用数: 0 h-index: 0机构: Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Key Lab Adv Drug Preparat Technol, Minist Educ, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Key Lab Henan Prov Drug Qual Control & Evaluat, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Inst Drug Discovery & Dev, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R ChinaMa, Xinli论文数: 0 引用数: 0 h-index: 0机构: China US Henan Hormel Canc Inst, 127,Dongming Rd,Jinshui Dist, Zhengzhou 450008, Henan, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R ChinaLi, Jian论文数: 0 引用数: 0 h-index: 0机构: China US Henan Hormel Canc Inst, 127,Dongming Rd,Jinshui Dist, Zhengzhou 450008, Henan, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R ChinaAgboyibor, Clement论文数: 0 引用数: 0 h-index: 0机构: Zhengzhou Univ, Key Lab Henan Prov Drug Qual Control & Evaluat, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Collaborat Innovat Ctr New Drug Res & Safety Evalu, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Inst Drug Discovery & Dev, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R ChinaBi, Yuefeng论文数: 0 引用数: 0 h-index: 0机构: Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Key Lab Adv Drug Preparat Technol, Minist Educ, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Key Lab Henan Prov Drug Qual Control & Evaluat, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Collaborat Innovat Ctr New Drug Res & Safety Evalu, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Inst Drug Discovery & Dev, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci, 100 Kexue Dadao,Gaoxin Dist, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R ChinaLiu, Hongmin论文数: 0 引用数: 0 h-index: 0机构: Zhengzhou Univ, Key Lab Henan Prov Drug Qual Control & Evaluat, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Inst Drug Discovery & Dev, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci, 100 Kexue Dadao,Gaoxin Dist, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R China
- [4] Reversible Lysine Specific Demethylase 1 (LSD1) Inhibitors: A Promising Wrench to Impair LSD1JOURNAL OF MEDICINAL CHEMISTRY, 2021, 64 (05) : 2466 - 2488Dai, Xing-Jie论文数: 0 引用数: 0 h-index: 0机构: Zhengzhou Univ, Sch Pharmaceut Sci,Inst Drug Discovery & Dev, Key Lab Adv Drug Preparat Technol,Key Lab Henan P, Minist Educ China,State Key Lab Esophageal Canc P, Zhengzhou 450001, Henan, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci,Inst Drug Discovery & Dev, Key Lab Adv Drug Preparat Technol,Key Lab Henan P, Minist Educ China,State Key Lab Esophageal Canc P, Zhengzhou 450001, Henan, Peoples R ChinaLiu, Ying论文数: 0 引用数: 0 h-index: 0机构: Zhengzhou Univ, Sch Pharmaceut Sci,Inst Drug Discovery & Dev, Key Lab Adv Drug Preparat Technol,Key Lab Henan P, Minist Educ China,State Key Lab Esophageal Canc P, Zhengzhou 450001, Henan, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci,Inst Drug Discovery & Dev, Key Lab Adv Drug Preparat Technol,Key Lab Henan P, Minist Educ China,State Key Lab Esophageal Canc P, Zhengzhou 450001, Henan, Peoples R ChinaXue, Lei-Peng论文数: 0 引用数: 0 h-index: 0机构: Zhengzhou Univ, Sch Pharmaceut Sci,Inst Drug Discovery & Dev, Key Lab Adv Drug Preparat Technol,Key Lab Henan P, Minist Educ China,State Key Lab Esophageal Canc P, Zhengzhou 450001, Henan, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci,Inst Drug Discovery & Dev, Key Lab Adv Drug Preparat Technol,Key Lab Henan P, Minist Educ China,State Key Lab Esophageal Canc P, Zhengzhou 450001, Henan, Peoples R ChinaXiong, Xiao-Peng论文数: 0 引用数: 0 h-index: 0机构: Zhengzhou Univ, Sch Pharmaceut Sci,Inst Drug Discovery & Dev, Key Lab Adv Drug Preparat Technol,Key Lab Henan P, Minist Educ China,State Key Lab Esophageal Canc P, Zhengzhou 450001, Henan, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci,Inst Drug Discovery & Dev, Key Lab Adv Drug Preparat Technol,Key Lab Henan P, Minist Educ China,State Key Lab Esophageal Canc P, Zhengzhou 450001, Henan, Peoples R ChinaZhou, Ying论文数: 0 引用数: 0 h-index: 0机构: Zhengzhou Univ, Sch Pharmaceut Sci,Inst Drug Discovery & Dev, Key Lab Adv Drug Preparat Technol,Key Lab Henan P, Minist Educ China,State Key Lab Esophageal Canc P, Zhengzhou 450001, Henan, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci,Inst Drug Discovery & Dev, Key Lab Adv Drug Preparat Technol,Key Lab Henan P, Minist Educ China,State Key Lab Esophageal Canc P, Zhengzhou 450001, Henan, Peoples R ChinaZheng, Yi-Chao论文数: 0 引用数: 0 h-index: 0机构: Zhengzhou Univ, Sch Pharmaceut Sci,Inst Drug Discovery & Dev, Key Lab Adv Drug Preparat Technol,Key Lab Henan P, Minist Educ China,State Key Lab Esophageal Canc P, Zhengzhou 450001, Henan, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci,Inst Drug Discovery & Dev, Key Lab Adv Drug Preparat Technol,Key Lab Henan P, Minist Educ China,State Key Lab Esophageal Canc P, Zhengzhou 450001, Henan, Peoples R ChinaLiu, Hong-Min论文数: 0 引用数: 0 h-index: 0机构: Zhengzhou Univ, Sch Pharmaceut Sci,Inst Drug Discovery & Dev, Key Lab Adv Drug Preparat Technol,Key Lab Henan P, Minist Educ China,State Key Lab Esophageal Canc P, Zhengzhou 450001, Henan, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci,Inst Drug Discovery & Dev, Key Lab Adv Drug Preparat Technol,Key Lab Henan P, Minist Educ China,State Key Lab Esophageal Canc P, Zhengzhou 450001, Henan, Peoples R China
- [5] Design, synthesis and in vitro evaluation of stilbene derivatives as novel LSD1 inhibitors for AML therapyBIOORGANIC & MEDICINAL CHEMISTRY, 2018, 26 (23-24) : 6000 - 6014Duan, Yingchao论文数: 0 引用数: 0 h-index: 0机构: Xinxiang Med Univ, Sch Pharm, Xinxiang 453003, Henan, Peoples R China Xinxiang Med Univ, Sch Pharm, Xinxiang 453003, Henan, Peoples R ChinaQin, Wenping论文数: 0 引用数: 0 h-index: 0机构: Xinxiang Med Univ, Sch Pharm, Xinxiang 453003, Henan, Peoples R China Xinxiang Med Univ, Sch Pharm, Xinxiang 453003, Henan, Peoples R ChinaSuo, Fengzhi论文数: 0 引用数: 0 h-index: 0机构: Zhengzhou Univ, Key Lab Adv Pharmaceut Technol, Coinnovat Ctr Henan Prov New Drug R&D & Preclin S, Inst Drug Discovery & Dev,Sch Pharmaceut Sci, 100 Kexue Ave, Zhengzhou 450001, Henan, Peoples R China Xinxiang Med Univ, Sch Pharm, Xinxiang 453003, Henan, Peoples R ChinaZhai, Xiaoyu论文数: 0 引用数: 0 h-index: 0机构: Xinxiang Med Univ, Sch Pharm, Xinxiang 453003, Henan, Peoples R China Xinxiang Med Univ, Sch Pharm, Xinxiang 453003, Henan, Peoples R ChinaGuan, Yuanyuan论文数: 0 引用数: 0 h-index: 0机构: Xinxiang Med Univ, Sch Pharm, Xinxiang 453003, Henan, Peoples R China Xinxiang Med Univ, Sch Pharm, Xinxiang 453003, Henan, Peoples R ChinaWang, Xiaojuan论文数: 0 引用数: 0 h-index: 0机构: Shangqiu Normal Univ, Coll Chem & Chem Engn, Shangqiu 476000, Henan, Peoples R China Xinxiang Med Univ, Sch Pharm, Xinxiang 453003, Henan, Peoples R ChinaZheng, Yichao论文数: 0 引用数: 0 h-index: 0机构: Zhengzhou Univ, Key Lab Adv Pharmaceut Technol, Coinnovat Ctr Henan Prov New Drug R&D & Preclin S, Inst Drug Discovery & Dev,Sch Pharmaceut Sci, 100 Kexue Ave, Zhengzhou 450001, Henan, Peoples R China Xinxiang Med Univ, Sch Pharm, Xinxiang 453003, Henan, Peoples R ChinaLiu, Hongmin论文数: 0 引用数: 0 h-index: 0机构: Zhengzhou Univ, Key Lab Adv Pharmaceut Technol, Coinnovat Ctr Henan Prov New Drug R&D & Preclin S, Inst Drug Discovery & Dev,Sch Pharmaceut Sci, 100 Kexue Ave, Zhengzhou 450001, Henan, Peoples R China Xinxiang Med Univ, Sch Pharm, Xinxiang 453003, Henan, Peoples R China
- [6] Antitumor activity of novel reversible LSD1 inhibitors in preclinical models of AML and SCLC.CANCER RESEARCH, 2021, 81 (13)Byun, Joo-Yun论文数: 0 引用数: 0 h-index: 0机构: Hanmi Res Ctr, Hwaseong Si, South Korea Hanmi Res Ctr, Hwaseong Si, South KoreaLee, Won Jong论文数: 0 引用数: 0 h-index: 0机构: Hanmi Res Ctr, Hwaseong Si, South Korea Hanmi Res Ctr, Hwaseong Si, South KoreaKim, Won jung论文数: 0 引用数: 0 h-index: 0机构: Hanmi Res Ctr, Hwaseong Si, South Korea Hanmi Res Ctr, Hwaseong Si, South KoreaKim, Minjeong论文数: 0 引用数: 0 h-index: 0机构: Hanmi Res Ctr, Hwaseong Si, South Korea Hanmi Res Ctr, Hwaseong Si, South KoreaBae, Inhwan论文数: 0 引用数: 0 h-index: 0机构: Hanmi Res Ctr, Hwaseong Si, South Korea Hanmi Res Ctr, Hwaseong Si, South KoreaHong, Seokhyun论文数: 0 引用数: 0 h-index: 0机构: Hanmi Res Ctr, Hwaseong Si, South Korea Hanmi Res Ctr, Hwaseong Si, South KoreaKim, Yu-Yon论文数: 0 引用数: 0 h-index: 0机构: Hanmi Res Ctr, Hwaseong Si, South Korea Hanmi Res Ctr, Hwaseong Si, South KoreaPark, Hyunjin论文数: 0 引用数: 0 h-index: 0机构: Hanmi Res Ctr, Hwaseong Si, South Korea Hanmi Res Ctr, Hwaseong Si, South KoreaKim, Eunyoung论文数: 0 引用数: 0 h-index: 0机构: Hanmi Res Ctr, Hwaseong Si, South Korea Hanmi Res Ctr, Hwaseong Si, South KoreaKim, Young Hoon论文数: 0 引用数: 0 h-index: 0机构: Hanmi Res Ctr, Hwaseong Si, South Korea Hanmi Res Ctr, Hwaseong Si, South KoreaAhn, Young Gil论文数: 0 引用数: 0 h-index: 0机构: Hanmi Res Ctr, Hwaseong Si, South Korea Hanmi Res Ctr, Hwaseong Si, South KoreaSuh, Kwee Hyun论文数: 0 引用数: 0 h-index: 0机构: Hanmi Res Ctr, Hwaseong Si, South Korea Hanmi Res Ctr, Hwaseong Si, South Korea
- [7] Design and Synthesis of Styrenylcyclopropylamine LSD1 InhibitorsACS MEDICINAL CHEMISTRY LETTERS, 2020, 11 (06): : 1213 - 1220Gehling, Victor S.论文数: 0 引用数: 0 h-index: 0机构: Constellat Pharmaceut, Cambridge, MA 02142 USA Constellat Pharmaceut, Cambridge, MA 02142 USAMcgrath, John P.论文数: 0 引用数: 0 h-index: 0机构: Constellat Pharmaceut, Cambridge, MA 02142 USA Constellat Pharmaceut, Cambridge, MA 02142 USADuplessis, Martin论文数: 0 引用数: 0 h-index: 0机构: Constellat Pharmaceut, Cambridge, MA 02142 USA Constellat Pharmaceut, Cambridge, MA 02142 USAKhanna, Avinash论文数: 0 引用数: 0 h-index: 0机构: Constellat Pharmaceut, Cambridge, MA 02142 USA Constellat Pharmaceut, Cambridge, MA 02142 USABrucelle, Francois论文数: 0 引用数: 0 h-index: 0机构: Constellat Pharmaceut, Cambridge, MA 02142 USA Constellat Pharmaceut, Cambridge, MA 02142 USAVaswani, Rishi G.论文数: 0 引用数: 0 h-index: 0机构: Constellat Pharmaceut, Cambridge, MA 02142 USA Constellat Pharmaceut, Cambridge, MA 02142 USACote, Alexandre论文数: 0 引用数: 0 h-index: 0机构: Constellat Pharmaceut, Cambridge, MA 02142 USA Constellat Pharmaceut, Cambridge, MA 02142 USAStuckey, Jacob论文数: 0 引用数: 0 h-index: 0机构: Constellat Pharmaceut, Cambridge, MA 02142 USA Constellat Pharmaceut, Cambridge, MA 02142 USAWatson, Venita论文数: 0 引用数: 0 h-index: 0机构: Constellat Pharmaceut, Cambridge, MA 02142 USA Constellat Pharmaceut, Cambridge, MA 02142 USACummings, Richard T.论文数: 0 引用数: 0 h-index: 0机构: Constellat Pharmaceut, Cambridge, MA 02142 USA Constellat Pharmaceut, Cambridge, MA 02142 USABalasubramanian, Srividya论文数: 0 引用数: 0 h-index: 0机构: Constellat Pharmaceut, Cambridge, MA 02142 USA Constellat Pharmaceut, Cambridge, MA 02142 USAIyer, Priya论文数: 0 引用数: 0 h-index: 0机构: Constellat Pharmaceut, Cambridge, MA 02142 USA Constellat Pharmaceut, Cambridge, MA 02142 USASawant, Priyanka论文数: 0 引用数: 0 h-index: 0机构: Constellat Pharmaceut, Cambridge, MA 02142 USA Constellat Pharmaceut, Cambridge, MA 02142 USAGood, Andrew C.论文数: 0 引用数: 0 h-index: 0机构: Constellat Pharmaceut, Cambridge, MA 02142 USA Constellat Pharmaceut, Cambridge, MA 02142 USAAlbrecht, Brian K.论文数: 0 引用数: 0 h-index: 0机构: Constellat Pharmaceut, Cambridge, MA 02142 USA Constellat Pharmaceut, Cambridge, MA 02142 USAHarmange, Jean-Christophe论文数: 0 引用数: 0 h-index: 0机构: Constellat Pharmaceut, Cambridge, MA 02142 USA Constellat Pharmaceut, Cambridge, MA 02142 USAAudia, James E.论文数: 0 引用数: 0 h-index: 0机构: Constellat Pharmaceut, Cambridge, MA 02142 USA Constellat Pharmaceut, Cambridge, MA 02142 USABellon, Steven F.论文数: 0 引用数: 0 h-index: 0机构: Constellat Pharmaceut, Cambridge, MA 02142 USA Constellat Pharmaceut, Cambridge, MA 02142 USATrojer, Patrick论文数: 0 引用数: 0 h-index: 0机构: Constellat Pharmaceut, Cambridge, MA 02142 USA Constellat Pharmaceut, Cambridge, MA 02142 USALevell, Julian R.论文数: 0 引用数: 0 h-index: 0机构: Constellat Pharmaceut, Cambridge, MA 02142 USA Constellat Pharmaceut, Cambridge, MA 02142 USA
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