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- [1] Structure and Function Studies of the mGlu5 Receptor in the Design of Novel Negative Allosteric ModulatorsCURRENT NEUROPHARMACOLOGY, 2014, 12 : 3 - 4Bennett, Kirstie A.论文数: 0 引用数: 0 h-index: 0机构: Heptares Therapeut Ltd, Welwyn Garden City AL7 3AX, Herts, England Heptares Therapeut Ltd, Welwyn Garden City AL7 3AX, Herts, EnglandDore, Andrew S.论文数: 0 引用数: 0 h-index: 0机构: Heptares Therapeut Ltd, Welwyn Garden City AL7 3AX, Herts, England Heptares Therapeut Ltd, Welwyn Garden City AL7 3AX, Herts, EnglandOkrasa, Krzysztof论文数: 0 引用数: 0 h-index: 0机构: Heptares Therapeut Ltd, Welwyn Garden City AL7 3AX, Herts, England Heptares Therapeut Ltd, Welwyn Garden City AL7 3AX, Herts, EnglandPatel, Jayesh C.论文数: 0 引用数: 0 h-index: 0机构: Heptares Therapeut Ltd, Welwyn Garden City AL7 3AX, Herts, England Heptares Therapeut Ltd, Welwyn Garden City AL7 3AX, Herts, EnglandSerrano-Vega, Maria论文数: 0 引用数: 0 h-index: 0机构: Heptares Therapeut Ltd, Welwyn Garden City AL7 3AX, Herts, England Heptares Therapeut Ltd, Welwyn Garden City AL7 3AX, Herts, EnglandCooke, Robert M.论文数: 0 引用数: 0 h-index: 0机构: Heptares Therapeut Ltd, Welwyn Garden City AL7 3AX, Herts, England Heptares Therapeut Ltd, Welwyn Garden City AL7 3AX, Herts, EnglandErrey, James C.论文数: 0 引用数: 0 h-index: 0机构: Heptares Therapeut Ltd, Welwyn Garden City AL7 3AX, Herts, England Heptares Therapeut Ltd, Welwyn Garden City AL7 3AX, Herts, EnglandJazayeri, Ali论文数: 0 引用数: 0 h-index: 0机构: Heptares Therapeut Ltd, Welwyn Garden City AL7 3AX, Herts, England Heptares Therapeut Ltd, Welwyn Garden City AL7 3AX, Herts, EnglandTehan, Ben论文数: 0 引用数: 0 h-index: 0机构: Heptares Therapeut Ltd, Welwyn Garden City AL7 3AX, Herts, England Heptares Therapeut Ltd, Welwyn Garden City AL7 3AX, Herts, EnglandWiggin, Giselle R.论文数: 0 引用数: 0 h-index: 0机构: Heptares Therapeut Ltd, Welwyn Garden City AL7 3AX, Herts, England Heptares Therapeut Ltd, Welwyn Garden City AL7 3AX, Herts, EnglandChristopher, John A.论文数: 0 引用数: 0 h-index: 0机构: Heptares Therapeut Ltd, Welwyn Garden City AL7 3AX, Herts, England Heptares Therapeut Ltd, Welwyn Garden City AL7 3AX, Herts, EnglandMarshall, Fiona H.论文数: 0 引用数: 0 h-index: 0机构: Heptares Therapeut Ltd, Welwyn Garden City AL7 3AX, Herts, England Heptares Therapeut Ltd, Welwyn Garden City AL7 3AX, Herts, England
- [2] Discovery and structure-activity relationship of 1,3-cyclohexyl amide derivatives as novel mGluR5 negative allosteric modulatorsBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2013, 23 (05) : 1398 - 1406Zhou, Hao论文数: 0 引用数: 0 h-index: 0机构: Lundbeck Res USA, Discovery Chem, Paramus, NJ 07652 USA Lundbeck Res USA, DMPK, Paramus, NJ 07652 USA Lundbeck Res USA, Discovery Chem, Paramus, NJ 07652 USATopiol, Sidney W.论文数: 0 引用数: 0 h-index: 0机构: Lundbeck Res USA, Discovery Chem, Paramus, NJ 07652 USA Lundbeck Res USA, DMPK, Paramus, NJ 07652 USA Lundbeck Res USA, Discovery Chem, Paramus, NJ 07652 USAGrenon, Michel论文数: 0 引用数: 0 h-index: 0机构: Lundbeck Res USA, Discovery Chem, Paramus, NJ 07652 USA Lundbeck Res USA, DMPK, Paramus, NJ 07652 USA Lundbeck Res USA, Discovery Chem, Paramus, NJ 07652 USAJimenez, Hermogenes N.论文数: 0 引用数: 0 h-index: 0机构: Lundbeck Res USA, Discovery Chem, Paramus, NJ 07652 USA Lundbeck Res USA, DMPK, Paramus, NJ 07652 USA Lundbeck Res USA, Discovery Chem, Paramus, NJ 07652 USAUberti, Michelle A.论文数: 0 引用数: 0 h-index: 0机构: Lundbeck Res USA, Mol Pharmacol, Paramus, NJ 07652 USA Lundbeck Res USA, SAR, Paramus, NJ 07652 USA Lundbeck Res USA, Discovery Chem, Paramus, NJ 07652 USASmith, Daniel G.论文数: 0 引用数: 0 h-index: 0机构: Lundbeck Res USA, Mol Pharmacol, Paramus, NJ 07652 USA Lundbeck Res USA, SAR, Paramus, NJ 07652 USA Lundbeck Res USA, Discovery Chem, Paramus, NJ 07652 USABrodbeck, Robbin M.论文数: 0 引用数: 0 h-index: 0机构: Lundbeck Res USA, Mol Pharmacol, Paramus, NJ 07652 USA Lundbeck Res USA, SAR, Paramus, NJ 07652 USA Lundbeck Res USA, Discovery Chem, Paramus, NJ 07652 USAChandrasena, Gamini论文数: 0 引用数: 0 h-index: 0机构: Lundbeck Res USA, Bioanal & Physiol, Paramus, NJ 07652 USA Lundbeck Res USA, Discovery Chem, Paramus, NJ 07652 USAPedersen, Henrik论文数: 0 引用数: 0 h-index: 0机构: H Lundbeck & Co AS, Discovery Chem, DK-2500 Valby, Denmark H Lundbeck & Co AS, DMPK, DK-2500 Valby, Denmark Lundbeck Res USA, Discovery Chem, Paramus, NJ 07652 USAMadsen, Jens Christian论文数: 0 引用数: 0 h-index: 0机构: H Lundbeck & Co AS, Discovery Chem, DK-2500 Valby, Denmark H Lundbeck & Co AS, DMPK, DK-2500 Valby, Denmark Lundbeck Res USA, Discovery Chem, Paramus, NJ 07652 USADoller, Dario论文数: 0 引用数: 0 h-index: 0机构: Lundbeck Res USA, Discovery Chem, Paramus, NJ 07652 USA Lundbeck Res USA, DMPK, Paramus, NJ 07652 USA Lundbeck Res USA, Discovery Chem, Paramus, NJ 07652 USALi, Guiying论文数: 0 引用数: 0 h-index: 0机构: Lundbeck Res USA, Discovery Chem, Paramus, NJ 07652 USA Lundbeck Res USA, DMPK, Paramus, NJ 07652 USA Lundbeck Res USA, Discovery Chem, Paramus, NJ 07652 USA
- [3] Heteroarylcyclohexylamides as mGlu5 Receptor Negative Allosteric ModulatorsCURRENT NEUROPHARMACOLOGY, 2011, 9 : 35 - 36Li, G.论文数: 0 引用数: 0 h-index: 0机构: Lundbeck Res USA, Chem & Pharmacokinet Sci Dept, Paramus, NJ 07652 USA Lundbeck Res USA, Chem & Pharmacokinet Sci Dept, Paramus, NJ 07652 USAApril, M.论文数: 0 引用数: 0 h-index: 0机构: Lundbeck Res USA, Chem & Pharmacokinet Sci Dept, Paramus, NJ 07652 USA Lundbeck Res USA, Chem & Pharmacokinet Sci Dept, Paramus, NJ 07652 USAZhou, H.论文数: 0 引用数: 0 h-index: 0机构: Lundbeck Res USA, Chem & Pharmacokinet Sci Dept, Paramus, NJ 07652 USA Lundbeck Res USA, Chem & Pharmacokinet Sci Dept, Paramus, NJ 07652 USAPu, X.论文数: 0 引用数: 0 h-index: 0机构: Lundbeck Res USA, Chem & Pharmacokinet Sci Dept, Paramus, NJ 07652 USA Lundbeck Res USA, Chem & Pharmacokinet Sci Dept, Paramus, NJ 07652 USAUberti, M. A.论文数: 0 引用数: 0 h-index: 0机构: Lundbeck Res USA, Chem & Pharmacokinet Sci Dept, Paramus, NJ 07652 USA Lundbeck Res USA, Chem & Pharmacokinet Sci Dept, Paramus, NJ 07652 USABrodbeck, R. M.论文数: 0 引用数: 0 h-index: 0机构: Lundbeck Res USA, Chem & Pharmacokinet Sci Dept, Paramus, NJ 07652 USA Lundbeck Res USA, Chem & Pharmacokinet Sci Dept, Paramus, NJ 07652 USACajina, M.论文数: 0 引用数: 0 h-index: 0机构: Lundbeck Res USA, Chem & Pharmacokinet Sci Dept, Paramus, NJ 07652 USA Lundbeck Res USA, Chem & Pharmacokinet Sci Dept, Paramus, NJ 07652 USAChandrasena, G.论文数: 0 引用数: 0 h-index: 0机构: Lundbeck Res USA, Chem & Pharmacokinet Sci Dept, Paramus, NJ 07652 USA Lundbeck Res USA, Chem & Pharmacokinet Sci Dept, Paramus, NJ 07652 USADoller, D.论文数: 0 引用数: 0 h-index: 0机构: Lundbeck Res USA, Chem & Pharmacokinet Sci Dept, Paramus, NJ 07652 USA Lundbeck Res USA, Chem & Pharmacokinet Sci Dept, Paramus, NJ 07652 USA
- [4] Discovery of novel positive allosteric modulators of the metabotropic glutamate receptor 5 (mGlu5)BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2011, 21 (05) : 1402 - 1406Varnes, Jeffrey G.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, CNS Discovery Res, Wilmington, DE 19850 USA AstraZeneca, CNS Discovery Res, Wilmington, DE 19850 USAMarcus, Andrew P.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, CNS Discovery Res, Wilmington, DE 19850 USA AstraZeneca, CNS Discovery Res, Wilmington, DE 19850 USAMauger, Russell C.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, CNS Discovery Res, Wilmington, DE 19850 USA AstraZeneca, CNS Discovery Res, Wilmington, DE 19850 USAThroner, Scott R.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, CNS Discovery Res, Wilmington, DE 19850 USA AstraZeneca, CNS Discovery Res, Wilmington, DE 19850 USAHoesch, Valerie论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, CNS Discovery Res, Wilmington, DE 19850 USA AstraZeneca, CNS Discovery Res, Wilmington, DE 19850 USAKing, Megan M.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, CNS Discovery Res, Wilmington, DE 19850 USA AstraZeneca, CNS Discovery Res, Wilmington, DE 19850 USAWang, Xia论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, CNS Discovery Res, Wilmington, DE 19850 USA AstraZeneca, CNS Discovery Res, Wilmington, DE 19850 USASygowski, Linda A.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, CNS Discovery Res, Wilmington, DE 19850 USA AstraZeneca, CNS Discovery Res, Wilmington, DE 19850 USASpear, Nathan论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, CNS Discovery Res, Wilmington, DE 19850 USA AstraZeneca, CNS Discovery Res, Wilmington, DE 19850 USAGadient, Reto论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, CNS Discovery Res, Wilmington, DE 19850 USA AstraZeneca, CNS Discovery Res, Wilmington, DE 19850 USABrown, Dean G.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, CNS Discovery Res, Wilmington, DE 19850 USA AstraZeneca, CNS Discovery Res, Wilmington, DE 19850 USACampbell, James B.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, CNS Discovery Res, Wilmington, DE 19850 USA AstraZeneca, CNS Discovery Res, Wilmington, DE 19850 USA
- [5] Pyrimidine derivatives as mGlu5 receptor negative allosteric modulatorsABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2014, 248Li, Guiying论文数: 0 引用数: 0 h-index: 0机构: Lundbeck Res USA, Discovery Chem & DMPK, Paramus, NJ 07652 USA Lundbeck Res USA, Discovery Chem & DMPK, Paramus, NJ 07652 USAApril, Myriam论文数: 0 引用数: 0 h-index: 0机构: Novartis, Cambridge, MA USA Lundbeck Res USA, Discovery Chem & DMPK, Paramus, NJ 07652 USAPu, Xiaosui论文数: 0 引用数: 0 h-index: 0机构: Lundbeck Res USA, Mol Pharmacol, Paramus, NJ 07652 USA Lundbeck Res USA, Discovery Chem & DMPK, Paramus, NJ 07652 USAUberti, Michelle A.论文数: 0 引用数: 0 h-index: 0机构: ETHOS Hlth Commun, Newtown, PA 18940 USA Lundbeck Res USA, Discovery Chem & DMPK, Paramus, NJ 07652 USABrodbeck, Robbin M.论文数: 0 引用数: 0 h-index: 0机构: Lundbeck Res USA, Mol Pharmacol, Paramus, NJ 07652 USA Lundbeck Res USA, Discovery Chem & DMPK, Paramus, NJ 07652 USABacolod, Maria D.论文数: 0 引用数: 0 h-index: 0机构: Celgene Avil Res, Bedford, MA 01730 USA Lundbeck Res USA, Discovery Chem & DMPK, Paramus, NJ 07652 USAChandrasena, Gamini论文数: 0 引用数: 0 h-index: 0机构: Lundbeck Res USA, Bioanalysis, Paramus, NJ 07652 USA Lundbeck Res USA, Discovery Chem & DMPK, Paramus, NJ 07652 USADoller, Dario论文数: 0 引用数: 0 h-index: 0机构: Lundbeck Res USA, Discovery Chem & DMPK, Paramus, NJ 07652 USA Lundbeck Res USA, Discovery Chem & DMPK, Paramus, NJ 07652 USA
- [6] Discovery of biological evaluation of pyrazole/imidazole amides as mGlu5 receptor negative allosteric modulatorsBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2013, 23 (07) : 2134 - 2139Chae, Eunhee论文数: 0 引用数: 0 h-index: 0机构: SK Biopharmaceut, Drug Dev Ctr, CNS Drug Discovery, Taejon 305712, South Korea SK Biopharmaceut, Drug Dev Ctr, CNS Drug Discovery, Taejon 305712, South KoreaShin, Yong-Je论文数: 0 引用数: 0 h-index: 0机构: SK Biopharmaceut, Drug Dev Ctr, CNS Drug Discovery, Taejon 305712, South Korea SK Biopharmaceut, Drug Dev Ctr, CNS Drug Discovery, Taejon 305712, South KoreaRyu, Eun-Ju论文数: 0 引用数: 0 h-index: 0机构: SK Biopharmaceut, Drug Dev Ctr, CNS Drug Discovery, Taejon 305712, South Korea SK Biopharmaceut, Drug Dev Ctr, CNS Drug Discovery, Taejon 305712, South KoreaJi, Mi Kyung论文数: 0 引用数: 0 h-index: 0机构: SK Biopharmaceut, Drug Dev Ctr, CNS Drug Discovery, Taejon 305712, South Korea SK Biopharmaceut, Drug Dev Ctr, CNS Drug Discovery, Taejon 305712, South KoreaCho, Nahm Ryune论文数: 0 引用数: 0 h-index: 0机构: SK Biopharmaceut, Drug Dev Ctr, CNS Drug Discovery, Taejon 305712, South Korea SK Biopharmaceut, Drug Dev Ctr, CNS Drug Discovery, Taejon 305712, South KoreaLee, Ki-Ho论文数: 0 引用数: 0 h-index: 0机构: SK Biopharmaceut, Drug Dev Ctr, CNS Drug Discovery, Taejon 305712, South Korea SK Biopharmaceut, Drug Dev Ctr, CNS Drug Discovery, Taejon 305712, South KoreaJeong, Hyun Ji论文数: 0 引用数: 0 h-index: 0机构: SK Biopharmaceut, Drug Dev Ctr, CNS Drug Discovery, Taejon 305712, South Korea SK Biopharmaceut, Drug Dev Ctr, CNS Drug Discovery, Taejon 305712, South KoreaKim, Soo-Jin论文数: 0 引用数: 0 h-index: 0机构: SK Biopharmaceut, Drug Dev Ctr, CNS Drug Discovery, Taejon 305712, South Korea SK Biopharmaceut, Drug Dev Ctr, CNS Drug Discovery, Taejon 305712, South KoreaChoi, Yeonjung论文数: 0 引用数: 0 h-index: 0机构: SK Biopharmaceut, Drug Dev Ctr, CNS Drug Discovery, Taejon 305712, South Korea SK Biopharmaceut, Drug Dev Ctr, CNS Drug Discovery, Taejon 305712, South KoreaOh, Kyung Seok论文数: 0 引用数: 0 h-index: 0机构: SK Biopharmaceut, Drug Dev Ctr, CNS Drug Discovery, Taejon 305712, South Korea SK Biopharmaceut, Drug Dev Ctr, CNS Drug Discovery, Taejon 305712, South KoreaPark, Chun-Eung论文数: 0 引用数: 0 h-index: 0机构: SK Biopharmaceut, Drug Dev Ctr, CNS Drug Discovery, Taejon 305712, South Korea SK Biopharmaceut, Drug Dev Ctr, CNS Drug Discovery, Taejon 305712, South KoreaYoon, Young Soo论文数: 0 引用数: 0 h-index: 0机构: SK Biopharmaceut, Drug Dev Ctr, CNS Drug Discovery, Taejon 305712, South Korea SK Biopharmaceut, Drug Dev Ctr, CNS Drug Discovery, Taejon 305712, South Korea
- [7] Recent Advances in the Design and Development of Novel Negative Allosteric Modulators of mGlu5ACS CHEMICAL NEUROSCIENCE, 2011, 2 (08): : 411 - 432Emmitte, Kyle A.论文数: 0 引用数: 0 h-index: 0机构: Vanderbilt Univ, Med Ctr, Dept Pharmacol, Vanderbilt Ctr Neurosci Drug Discovery, Nashville, TN 37232 USA Vanderbilt Univ, Med Ctr, Dept Chem, Nashville, TN 37232 USA Vanderbilt Univ, Med Ctr, Dept Pharmacol, Vanderbilt Ctr Neurosci Drug Discovery, Nashville, TN 37232 USA
- [8] 6-Aryl-3-pyrrolidinylpyridines as mGlu5 receptor negative allosteric modulatorsBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2011, 21 (16) : 4891 - 4899Weiss, Jesse M.论文数: 0 引用数: 0 h-index: 0机构: Lundbeck Res USA, Chem & Pharmacokinet Sci, Paramus, NJ 07652 USA Lundbeck Res USA, Chem & Pharmacokinet Sci, Paramus, NJ 07652 USAJimenez, Hermogenes N.论文数: 0 引用数: 0 h-index: 0机构: Lundbeck Res USA, Chem & Pharmacokinet Sci, Paramus, NJ 07652 USA Lundbeck Res USA, Chem & Pharmacokinet Sci, Paramus, NJ 07652 USALi, Guiying论文数: 0 引用数: 0 h-index: 0机构: Lundbeck Res USA, Chem & Pharmacokinet Sci, Paramus, NJ 07652 USA Lundbeck Res USA, Chem & Pharmacokinet Sci, Paramus, NJ 07652 USAApril, Myriam论文数: 0 引用数: 0 h-index: 0机构: Lundbeck Res USA, Chem & Pharmacokinet Sci, Paramus, NJ 07652 USA Lundbeck Res USA, Chem & Pharmacokinet Sci, Paramus, NJ 07652 USAUberti, Michelle A.论文数: 0 引用数: 0 h-index: 0机构: Lundbeck Res USA, Synapt Transmiss Dis Biol Unit, Paramus, NJ 07652 USA Lundbeck Res USA, Chem & Pharmacokinet Sci, Paramus, NJ 07652 USABacolod, Maria D.论文数: 0 引用数: 0 h-index: 0机构: Lundbeck Res USA, Chem & Pharmacokinet Sci, Paramus, NJ 07652 USA Lundbeck Res USA, Chem & Pharmacokinet Sci, Paramus, NJ 07652 USABrodbeck, Robb M.论文数: 0 引用数: 0 h-index: 0机构: Lundbeck Res USA, Synapt Transmiss Dis Biol Unit, Paramus, NJ 07652 USA Lundbeck Res USA, Chem & Pharmacokinet Sci, Paramus, NJ 07652 USADoller, Dario论文数: 0 引用数: 0 h-index: 0机构: Lundbeck Res USA, Chem & Pharmacokinet Sci, Paramus, NJ 07652 USA Lundbeck Res USA, Chem & Pharmacokinet Sci, Paramus, NJ 07652 USA
- [9] Discovery and SAR of novel series of imidazopyrimidinones and dihydroimidazopyrimidinones as positive allosteric modulators of the metabotropic glutamate receptor 5 (mGlu5)BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2015, 25 (06) : 1310 - 1317Luz Martin-Martin, Maria论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev, Neurosci Med Chem, Toledo 45007, Spain Janssen Res & Dev, Neurosci Med Chem, Toledo 45007, SpainManuel Bartolome-Nebreda, Jose论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev, Neurosci Med Chem, Toledo 45007, Spain Janssen Res & Dev, Neurosci Med Chem, Toledo 45007, SpainConde-Ceide, Susana论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev, Neurosci Med Chem, Toledo 45007, Spain Janssen Res & Dev, Neurosci Med Chem, Toledo 45007, SpainAlonso de Diego, Sergio A.论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev, Neurosci Med Chem, Toledo 45007, Spain Janssen Res & Dev, Neurosci Med Chem, Toledo 45007, SpainLopez, Silvia论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev, Neurosci Med Chem, Toledo 45007, Spain Janssen Res & Dev, Neurosci Med Chem, Toledo 45007, SpainMartinez-Viturro, Carlos M.论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev, Neurosci Med Chem, Toledo 45007, Spain Janssen Res & Dev, Neurosci Med Chem, Toledo 45007, SpainHan Min Tong论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev, Neurosci Med Chem, Toledo 45007, Spain Janssen Res & Dev, Neurosci Med Chem, Toledo 45007, SpainLavreysen, Hilde论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev, Neurosci, B-2340 Beerse, Belgium Janssen Res & Dev, Neurosci Med Chem, Toledo 45007, SpainMacdonald, Gregor J.论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev, Neurosci, B-2340 Beerse, Belgium Janssen Res & Dev, Neurosci Med Chem, Toledo 45007, SpainSteckler, Thomas论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev, Neurosci, B-2340 Beerse, Belgium Janssen Res & Dev, Neurosci Med Chem, Toledo 45007, SpainMackie, Claire论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev, Discovery Sci ADME Tox, B-2340 Beerse, Belgium Janssen Res & Dev, Neurosci Med Chem, Toledo 45007, SpainBridges, Thomas M.论文数: 0 引用数: 0 h-index: 0机构: Vanderbilt Univ, Med Ctr, Dept Pharmacol, Nashville, TN 37232 USA Vanderbilt Univ, Med Ctr, Vanderbilt Ctr Neurosci Drug Discovery, Nashville, TN 37232 USA Vanderbilt Specialized Chem Ctr Probe Dev MLPCN, Nashville, TN 37232 USA Janssen Res & Dev, Neurosci Med Chem, Toledo 45007, SpainDaniels, J. Scott论文数: 0 引用数: 0 h-index: 0机构: Vanderbilt Univ, Med Ctr, Dept Pharmacol, Nashville, TN 37232 USA Vanderbilt Univ, Med Ctr, Vanderbilt Ctr Neurosci Drug Discovery, Nashville, TN 37232 USA Vanderbilt Specialized Chem Ctr Probe Dev MLPCN, Nashville, TN 37232 USA Janssen Res & Dev, Neurosci Med Chem, Toledo 45007, SpainNiswender, Colleen M.论文数: 0 引用数: 0 h-index: 0机构: Vanderbilt Univ, Med Ctr, Dept Pharmacol, Nashville, TN 37232 USA Vanderbilt Univ, Med Ctr, Vanderbilt Ctr Neurosci Drug Discovery, Nashville, TN 37232 USA Vanderbilt Specialized Chem Ctr Probe Dev MLPCN, Nashville, TN 37232 USA Janssen Res & Dev, Neurosci Med Chem, Toledo 45007, SpainNoetzel, Meredith J.论文数: 0 引用数: 0 h-index: 0机构: Vanderbilt Univ, Med Ctr, Dept Pharmacol, Nashville, TN 37232 USA Vanderbilt Univ, Med Ctr, Vanderbilt Ctr Neurosci Drug Discovery, Nashville, TN 37232 USA Vanderbilt Specialized Chem Ctr Probe Dev MLPCN, Nashville, TN 37232 USA Janssen Res & Dev, Neurosci Med Chem, Toledo 45007, SpainJones, Carrie K.论文数: 0 引用数: 0 h-index: 0机构: Vanderbilt Univ, Med Ctr, Dept Pharmacol, Nashville, TN 37232 USA Vanderbilt Univ, Med Ctr, Vanderbilt Ctr Neurosci Drug Discovery, Nashville, TN 37232 USA Vanderbilt Specialized Chem Ctr Probe Dev MLPCN, Nashville, TN 37232 USA Janssen Res & Dev, Neurosci Med Chem, Toledo 45007, SpainConn, P. Jeffrey论文数: 0 引用数: 0 h-index: 0机构: Vanderbilt Univ, Med Ctr, Dept Pharmacol, Nashville, TN 37232 USA Vanderbilt Univ, Med Ctr, Vanderbilt Ctr Neurosci Drug Discovery, Nashville, TN 37232 USA Vanderbilt Specialized Chem Ctr Probe Dev MLPCN, Nashville, TN 37232 USA Janssen Res & Dev, Neurosci Med Chem, Toledo 45007, SpainLindsley, Craig W.论文数: 0 引用数: 0 h-index: 0机构: Vanderbilt Univ, Med Ctr, Dept Pharmacol, Nashville, TN 37232 USA Vanderbilt Univ, Med Ctr, Vanderbilt Ctr Neurosci Drug Discovery, Nashville, TN 37232 USA Vanderbilt Specialized Chem Ctr Probe Dev MLPCN, Nashville, TN 37232 USA Vanderbilt Univ, Dept Chem, Nashville, TN 37232 USA Janssen Res & Dev, Neurosci Med Chem, Toledo 45007, SpainStauffer, Shaun R.论文数: 0 引用数: 0 h-index: 0机构: Vanderbilt Univ, Med Ctr, Dept Pharmacol, Nashville, TN 37232 USA Vanderbilt Univ, Med Ctr, Vanderbilt Ctr Neurosci Drug Discovery, Nashville, TN 37232 USA Vanderbilt Specialized Chem Ctr Probe Dev MLPCN, Nashville, TN 37232 USA Vanderbilt Univ, Dept Chem, Nashville, TN 37232 USA Janssen Res & Dev, Neurosci Med Chem, Toledo 45007, Spain
- [10] SAR Studies on mGlu5 Receptor Positive Allosteric Modulators (2003-2013)CURRENT TOPICS IN MEDICINAL CHEMISTRY, 2014, 14 (15) : 1789 - 1841Hao, Junliang论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Lilly Corp Ctr, Discovery Chem Res & Technol, Indianapolis, IN 46285 USA Eli Lilly & Co, Lilly Corp Ctr, Discovery Chem Res & Technol, Indianapolis, IN 46285 USAXiong, Hui论文数: 0 引用数: 0 h-index: 0机构: Avid Radiopharmaceut, Philadelphia, PA 19104 USA Eli Lilly & Co, Lilly Corp Ctr, Discovery Chem Res & Technol, Indianapolis, IN 46285 USA