A facile synthesis of 1-alkyl-5-arylalkoxy-6-methoxy-3,4-dihydroisoquinolines

被引：1

作者：

Yim, Heong-Seup

Kim, Ho-Kyun

Kim, Jeum-Jong

Kweon, Deok-Heon

Lee, Sang-Gyeong ^{[1
]}

Kim, Jung-Ho

Yoon, Yong-Jin

机构：

[1] Gyeongsang Natl Univ, Grad Sch Mol Mat & Nanochem, Environm Biotechnol Natl Core Res Ctr, Res Inst Nat Sci,Dept Chem, Jinju 660701, South Korea

[2] Gyeongsang Natl Univ, Grad Sch Mol Mat & Nanochem, Res Inst Life Sci, Dept Chem, Jinju 660701, South Korea

[3] Hanwha Chem R&D Ctr, Taejon 305345, South Korea

来源：

JOURNAL OF HETEROCYCLIC CHEMISTRY | 2007年 / 44卷 / 04期

关键词：

D O I：

10.1002/jhet.5570440426

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

1-Alkyl-5-arylalkoxy-6-methoxy-3,4-dihydroisoquinolines were synthesized by the alkylation of 1-alkyl-5-hydroxy-6-methoxy-3,4-dihydroisoquinolines with arylalkyl halide in the presence of potassium carbonate. 1-Alkyl-5-hydroxy-6-methoxy-3,4-dihydroisoquinolines as key precursor prepared from o-vaniline via 6 steps.

引用

页码：909 / 914

页数：6

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