Facile synthesis of novel indeno[1,2-b]indol-10-one derivatives by the oxidation with DDQ

被引:17
|
作者
Wang, JB [1 ]
Ji, QG [1 ]
Xu, J [1 ]
Wu, XH [1 ]
Xie, YY [1 ]
机构
[1] Chinese Acad Sci, SIBS, Shanghai Inst Mat Med, State Key Lab Drug Res, Shanghai 201203, Peoples R China
关键词
5,10-dihydroindeno[1,2-b]indole; indeno[1,2-b]indol-10(5H)-one; oxidation; DDQ;
D O I
10.1081/SCC-200049795
中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
The synthesis of indeno[1,2-b]indol-10-one analogues with a wide range of biological activities was described. They are also important intermediates of some selective estrogen receptor modulators (SERMs).
引用
收藏
页码:581 / 588
页数:8
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