A simple method for estimation of agonist activity at GPCRs: characterization of responses elicited by M2 and M3 muscarinic receptors

被引：0
|
作者：
Tran, John A. [1 ]
Chang, Alex [1 ]
Matsui, Minoru [2 ]
Ehlert, Frederick J. [1 ]
机构：
[1] Univ Calif Irvine, Irvine, CA USA
[2] Darthmouth Med Sch, Lebanon, NH USA
来源：
FASEB JOURNAL | 2008年 / 22卷
关键词：
D O I：
暂无
中图分类号：
Q5 [生物化学]; Q7 [分子生物学];
学科分类号：
071010 ; 081704 ;
摘要：
引用
收藏
页数：1
相关论文
共 50 条
  • [1] Differential agonist-induced regulation of human M2 and M3 muscarinic receptors
    Stope, MB
    Kunkel, C
    Kories, C
    Schmidt, M
    Michel, MC
    BIOCHEMICAL PHARMACOLOGY, 2003, 66 (11) : 2099 - 2105
  • [2] Interaction of edrophonium with muscarinic acetylcholine M2 and M3 receptors
    Tanito, Y
    Miwa, T
    Endou, M
    Hirose, Y
    Gamoh, M
    Nakaya, H
    Okumura, F
    ANESTHESIOLOGY, 2001, 94 (05) : 804 - 814
  • [3] Neuromuscular relaxants as antagonists for M2 and M3 muscarinic receptors
    Hou, VY
    Hirshman, CA
    Emala, CW
    ANESTHESIOLOGY, 1998, 88 (03) : 744 - 750
  • [4] Cholinergic receptors in the marine coronary circulation: Role of M2 and M3 muscarinic receptors in responses to acetylcholine
    Lamping, KG
    Wess, J
    Nuno, DW
    Faraci, FM
    FASEB JOURNAL, 2003, 17 (04): : A507 - A507
  • [5] Contribution of M2 and M3 Muscarinic Receptors in Small Airway Contraction
    Brown, S. M.
    Sturton, R. G.
    Koarai, A.
    Barnes, P. J.
    Donnelly, L. E.
    AMERICAN JOURNAL OF RESPIRATORY AND CRITICAL CARE MEDICINE, 2009, 179
  • [6] Cystometric findings in mice lacking muscarinic M2 or M3 receptors
    Igawa, Y
    Zhang, XY
    Nishizawa, O
    Umeda, M
    Iwata, A
    Taketo, MM
    Manabe, T
    Matsui, M
    Andersson, KE
    JOURNAL OF UROLOGY, 2004, 172 (06): : 2460 - 2464
  • [7] Muscarinic agonist-mediated heterologous desensitization in isolated ileum requires activation of both muscarinic M2 and M3 receptors
    Griffin, MT
    Matsui, M
    Shehnaz, D
    Ansari, KZ
    Taketo, MM
    Manabe, T
    Ehlert, FJ
    JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS, 2004, 308 (01): : 339 - 349
  • [8] CLOZAPINE IS A POTENT AGONIST AT HUMAN M4 MUSCARINIC RECEPTORS AND AN ANTAGONIST AT M1, M2, M3, AND M5 RECEPTORS
    LISTON, D
    WARD, KM
    JONES, SB
    ZORN, SH
    LIFE SCIENCES, 1995, 56 (11-12) : 1018 - 1018
  • [9] Inverse agonist activity of pirenzepine at M2 muscarinic acetylcholine receptors
    Daeffler, L
    Schmidlin, F
    Gies, JP
    Landry, Y
    BRITISH JOURNAL OF PHARMACOLOGY, 1999, 126 (05) : 1246 - 1252
  • [10] Contractile roles of the M2 and M3 muscarinic receptors in the guinea pig colon
    Sawyer, GW
    Ehlert, FJ
    JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS, 1998, 284 (01): : 269 - 277
12345