Targeting Bromodomains in Myeloma

被引:0
|
作者
Bradner, James E. [1 ]
机构
[1] Harvard Univ, Sch Med, Dana Farber Canc Inst, Boston, MA 02115 USA
关键词
D O I
暂无
中图分类号
R5 [内科学];
学科分类号
1002 ; 100201 ;
摘要
6
引用
收藏
页数:1
相关论文
共 50 条
  • [1] Targeting BET bromodomains for cancer treatment
    Jung, Marie
    Gelato, Kathy A.
    Fernandez-Montalvan, Amaury
    Siegel, Stephan
    Haendler, Bernard
    EPIGENOMICS, 2015, 7 (03) : 487 - 501
  • [2] Dihydropyridine Lactam Analogs Targeting BET Bromodomains
    Jiang, Jiewei
    Sigua, Logan H.
    Chan, Alice
    Kalra, Prakriti
    Pomerantz, William C. K.
    Schonbrunn, Ernst
    Qi, Jun
    Georg, Gunda, I
    CHEMMEDCHEM, 2022, 17 (01)
  • [3] Targeting bromodomains: epigenetic readers of lysine acetylation
    Filippakopoulos, Panagis
    Knapp, Stefan
    NATURE REVIEWS DRUG DISCOVERY, 2014, 13 (05) : 339 - 358
  • [4] Targeting bromodomains: epigenetic readers of lysine acetylation
    Panagis Filippakopoulos
    Stefan Knapp
    Nature Reviews Drug Discovery, 2014, 13 : 337 - 356
  • [5] Selective Targeting of Different Bromodomains by Small Molecules
    Qi, Jun
    Shi, Yang
    CANCER CELL, 2020, 37 (06) : 764 - 766
  • [6] Interactome Rewiring Following Pharmacological Targeting of BET Bromodomains
    Lambert, Jean-Philippe
    Picaud, Sarah
    Fujisawa, Takao
    Hou, Huayun
    Savitsky, Pavel
    Uuskula-Reimand, Liis
    Gupta, Gagan D.
    Abdouni, Hala
    Lin, Zhen-Yuan
    Tucholska, Monika
    Knight, James D. R.
    Gonzalez-Badillo, Beatriz
    St-Denis, Nicole
    Newman, Joseph A.
    Stucki, Manuel
    Pelletier, Laurence
    Bandeira, Nuno
    Wilson, Michael D.
    Filippakopoulos, Panagis
    Gingras, Anne-Claude
    MOLECULAR CELL, 2019, 73 (03) : 621 - +
  • [7] Targeting MYC dependence in cancer by inhibiting BET bromodomains
    Mertz, Jennifer A.
    Conery, Andrew R.
    Bryant, Barbara M.
    Sandy, Peter
    Balasubramanian, Srividya
    Mele, Deanna A.
    Bergeron, Louise
    Sims, Robert J., III
    PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2011, 108 (40) : 16669 - 16674
  • [8] Annual Review of Cancer Biology Targeting BET Bromodomains in Cancer
    Trojer, Patrick
    ANNUAL REVIEW OF CANCER BIOLOGY, 2022, 6 : 313 - 336
  • [9] Benzodiazepines and benzotriazepines as protein interaction inhibitors targeting bromodomains of the BET family
    Filippakopoulos, Panagis
    Picaud, Sarah
    Fedorov, Oleg
    Keller, Marco
    Wrobel, Matthias
    Morgenstern, Olaf
    Bracher, Franz
    Knapp, Stefan
    BIOORGANIC & MEDICINAL CHEMISTRY, 2012, 20 (06) : 1878 - 1886
  • [10] Targeting BET Bromodomains in Pre-Clinical Models of Burkitt Lymphoma
    Ippolito, Thomas
    Gu, Juan J.
    Tang, Gregory
    Mavis, Cory
    Miles, Rodney R.
    Hernandez-Ilizaliturri, Francisco J.
    Barth, Matthew J.
    BLOOD, 2016, 128 (22)