Discovery of triazolopyrimidine-based PDE8 inhibitors: Exceptionally ligand-efficient and lipophilic ligand-efficient compounds

被引：0
|
作者：
DeNinno, Michael P. [1 ]
Wright, Stephen W. [1 ]
Etienne, John B. [1 ]
Olson, Thanh V. [1 ]
Rocke, Benjamin N. [1 ]
Millham, Michele L. [1 ]
Boyer, David D. [1 ]
Doran, Shawn D. [1 ]
Houseknecht, Karen [1 ]
机构：
[1] Pfizer Global Res & Dev, Cardiovasc & Metab Dis, Groton, CT 06340 USA
来源：
ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY | 2012年 / 243卷
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中图分类号：
O6 [化学];
学科分类号：
0703 ;
摘要：
262-MEDI
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页数：1
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