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- [1] MEDI 316-Ureas substituted with partially reduced heteroaromatics as novel transient receptor potential vanilloid 1 (TRPV1) antagonists for the treatment of painABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2006, 232Gomtsyan, Arthur论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Neurosci Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Neurosci Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USABayburt, Erol K.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Neurosci Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Neurosci Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USASchmidt, Robert G.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Neurosci Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Neurosci Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USADaanen, Jerome F.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Neurosci Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Neurosci Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAKoenig, John R.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Neurosci Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Neurosci Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USALatshaw, Steven P.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Neurosci Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Neurosci Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAJinkerson, Tammie K.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Neurosci Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Neurosci Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USABrown, Brian S.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Neurosci Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Neurosci Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAMcdonald, Heath A.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Neurosci Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Neurosci Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USABianchi, Bruce论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Neurosci Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Neurosci Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAPuttfarcken, Pamela论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Neurosci Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Neurosci Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAMoreland, Robert论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Neurosci Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Neurosci Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USACui, Minglei论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Neurosci Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Neurosci Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAHonore, Prisca论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Neurosci Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Neurosci Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USASt George, Karen论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Neurosci Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USADarbyshire, John F.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Neurosci Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAMarsh, Kennan C.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Neurosci Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAFaltynek, Connie R.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Neurosci Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Neurosci Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USALee, Chih-Hung论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Neurosci Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Neurosci Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA
- [2] Discovery of novel pyrrolopyridazine scaffolds as transient receptor potential vanilloid (TRPV1) antagonistsBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2012, 22 (22) : 6888 - 6895Dorange, Ismet论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca R&D, CNSP iMed Sci, Med Chem, Innovat Med, SE-15185 Sodertalje, Sweden AstraZeneca R&D, CNSP iMed Sci, Med Chem, Innovat Med, SE-15185 Sodertalje, SwedenForsblom, Rickard论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca R&D, CNSP iMed Sci, Med Chem, Innovat Med, SE-15185 Sodertalje, Sweden AstraZeneca R&D, CNSP iMed Sci, Med Chem, Innovat Med, SE-15185 Sodertalje, SwedenMacsari, Istvan论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca R&D, CNSP iMed Sci, Med Chem, Innovat Med, SE-15185 Sodertalje, Sweden AstraZeneca R&D, CNSP iMed Sci, Med Chem, Innovat Med, SE-15185 Sodertalje, SwedenSvensson, Mats论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca R&D, CNSP iMed Sci, Med Chem, Innovat Med, SE-15185 Sodertalje, Sweden AstraZeneca R&D, CNSP iMed Sci, Med Chem, Innovat Med, SE-15185 Sodertalje, SwedenBylund, Johan论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca R&D, CNSP iMed Sci, DMPK, Innovat Med, SE-15185 Sodertalje, Sweden AstraZeneca R&D, CNSP iMed Sci, Med Chem, Innovat Med, SE-15185 Sodertalje, SwedenBesidski, Yevgeni论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca R&D, CNSP iMed Sci, Med Chem, Innovat Med, SE-15185 Sodertalje, Sweden AstraZeneca R&D, CNSP iMed Sci, Med Chem, Innovat Med, SE-15185 Sodertalje, SwedenBlid, Jan论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca R&D, CNSP iMed Sci, Med Chem, Innovat Med, SE-15185 Sodertalje, Sweden AstraZeneca R&D, CNSP iMed Sci, Med Chem, Innovat Med, SE-15185 Sodertalje, SwedenSohn, Daniel论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca R&D, CNSP iMed Sci, Med Chem, Innovat Med, SE-15185 Sodertalje, Sweden AstraZeneca R&D, CNSP iMed Sci, Med Chem, Innovat Med, SE-15185 Sodertalje, SwedenGravenfors, Ylva论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca R&D, CNSP iMed Sci, Med Chem, Innovat Med, SE-15185 Sodertalje, Sweden AstraZeneca R&D, CNSP iMed Sci, Med Chem, Innovat Med, SE-15185 Sodertalje, Sweden
- [3] Chroman and tetrahydroquinoline ureas as potent TRPV1 antagonistsBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2011, 21 (05) : 1338 - 1341Schmidt, Robert G.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USABayburt, Erol K.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USALatshaw, Steven P.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAKoenig, John R.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USADaanen, Jerome F.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAMcDonald, Heath A.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USABianchi, Bruce R.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAZhong, Chengmin论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAJoshi, Shailen论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAHonore, Prisca论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAMarsh, Kennan C.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USALee, Chih-Hung论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAFaltynek, Connie R.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAGomtsyan, Arthur论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA
- [4] Tetrahydropyridine-4-carboxamides as novel, potent transient receptor potential vanilloid 1 (TRPV1) antagonistsBIOORGANIC & MEDICINAL CHEMISTRY, 2008, 16 (18) : 8516 - 8525Brown, Brian S.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Neurosci Res, Global Pharmaceut Res & Dev, Dept R4PM, Abbott Pk, IL 60064 USA Abbott Labs, Neurosci Res, Global Pharmaceut Res & Dev, Dept R4PM, Abbott Pk, IL 60064 USAKeddy, Ryan论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Neurosci Res, Global Pharmaceut Res & Dev, Dept R4PM, Abbott Pk, IL 60064 USA Abbott Labs, Neurosci Res, Global Pharmaceut Res & Dev, Dept R4PM, Abbott Pk, IL 60064 USAZheng, Guo Zhu论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Neurosci Res, Global Pharmaceut Res & Dev, Dept R4PM, Abbott Pk, IL 60064 USA Abbott Labs, Neurosci Res, Global Pharmaceut Res & Dev, Dept R4PM, Abbott Pk, IL 60064 USASchmidt, Robert G.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Neurosci Res, Global Pharmaceut Res & Dev, Dept R4PM, Abbott Pk, IL 60064 USA Abbott Labs, Neurosci Res, Global Pharmaceut Res & Dev, Dept R4PM, Abbott Pk, IL 60064 USAKoenig, John R.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Neurosci Res, Global Pharmaceut Res & Dev, Dept R4PM, Abbott Pk, IL 60064 USA Abbott Labs, Neurosci Res, Global Pharmaceut Res & Dev, Dept R4PM, Abbott Pk, IL 60064 USAMcDonald, Heath A.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Neurosci Res, Global Pharmaceut Res & Dev, Dept R4PM, Abbott Pk, IL 60064 USA Abbott Labs, Neurosci Res, Global Pharmaceut Res & Dev, Dept R4PM, Abbott Pk, IL 60064 USABianchi, Bruce R.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Neurosci Res, Global Pharmaceut Res & Dev, Dept R4PM, Abbott Pk, IL 60064 USA Abbott Labs, Neurosci Res, Global Pharmaceut Res & Dev, Dept R4PM, Abbott Pk, IL 60064 USAHonore, Prisca论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Neurosci Res, Global Pharmaceut Res & Dev, Dept R4PM, Abbott Pk, IL 60064 USA Abbott Labs, Neurosci Res, Global Pharmaceut Res & Dev, Dept R4PM, Abbott Pk, IL 60064 USAJarvis, Michael F.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Neurosci Res, Global Pharmaceut Res & Dev, Dept R4PM, Abbott Pk, IL 60064 USA Abbott Labs, Neurosci Res, Global Pharmaceut Res & Dev, Dept R4PM, Abbott Pk, IL 60064 USASurowy, Carol S.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Neurosci Res, Global Pharmaceut Res & Dev, Dept R4PM, Abbott Pk, IL 60064 USA Abbott Labs, Neurosci Res, Global Pharmaceut Res & Dev, Dept R4PM, Abbott Pk, IL 60064 USAPolakowski, James S.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Neurosci Res, Global Pharmaceut Res & Dev, Dept R4PM, Abbott Pk, IL 60064 USA Abbott Labs, Neurosci Res, Global Pharmaceut Res & Dev, Dept R4PM, Abbott Pk, IL 60064 USAMarsh, Kennan C.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Neurosci Res, Global Pharmaceut Res & Dev, Dept R4PM, Abbott Pk, IL 60064 USA Abbott Labs, Neurosci Res, Global Pharmaceut Res & Dev, Dept R4PM, Abbott Pk, IL 60064 USAFaltynek, Connie R.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Neurosci Res, Global Pharmaceut Res & Dev, Dept R4PM, Abbott Pk, IL 60064 USA Abbott Labs, Neurosci Res, Global Pharmaceut Res & Dev, Dept R4PM, Abbott Pk, IL 60064 USALee, Chih-Hung论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Neurosci Res, Global Pharmaceut Res & Dev, Dept R4PM, Abbott Pk, IL 60064 USA Abbott Labs, Neurosci Res, Global Pharmaceut Res & Dev, Dept R4PM, Abbott Pk, IL 60064 USA
- [5] Novel piperazine urea derivatives as highly potent transient receptor potential vanilloid 1 (TRPV1) antagonistsBIOORGANIC CHEMISTRY, 2021, 115Hu, Jing论文数: 0 引用数: 0 h-index: 0机构: Henan Univ, Inst Innovat Drug Design & Evaluat, Sch Pharm, N Jinming Ave, Kaifeng 475004, Henan, Peoples R China Henan Univ, Inst Innovat Drug Design & Evaluat, Sch Pharm, N Jinming Ave, Kaifeng 475004, Henan, Peoples R ChinaGao, Mengkang论文数: 0 引用数: 0 h-index: 0机构: Henan Univ, Inst Innovat Drug Design & Evaluat, Sch Pharm, N Jinming Ave, Kaifeng 475004, Henan, Peoples R China Henan Univ, Inst Innovat Drug Design & Evaluat, Sch Pharm, N Jinming Ave, Kaifeng 475004, Henan, Peoples R ChinaZhang, Yang论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Ctr Drug Discovery, State Key Lab Nat Med, 24 Tongjiaxiang, Nanjing 210009, Jiangsu, Peoples R China Henan Univ, Inst Innovat Drug Design & Evaluat, Sch Pharm, N Jinming Ave, Kaifeng 475004, Henan, Peoples R ChinaWang, Yusui论文数: 0 引用数: 0 h-index: 0机构: Henan Univ, Inst Innovat Drug Design & Evaluat, Sch Pharm, N Jinming Ave, Kaifeng 475004, Henan, Peoples R China Henan Univ, Inst Innovat Drug Design & Evaluat, Sch Pharm, N Jinming Ave, Kaifeng 475004, Henan, Peoples R ChinaQiao, Zhenrui论文数: 0 引用数: 0 h-index: 0机构: Henan Univ, Inst Innovat Drug Design & Evaluat, Sch Pharm, N Jinming Ave, Kaifeng 475004, Henan, Peoples R China Henan Univ, Inst Innovat Drug Design & Evaluat, Sch Pharm, N Jinming Ave, Kaifeng 475004, Henan, Peoples R ChinaZhang, Weiya论文数: 0 引用数: 0 h-index: 0机构: Henan Univ, Inst Innovat Drug Design & Evaluat, Sch Pharm, N Jinming Ave, Kaifeng 475004, Henan, Peoples R China Henan Univ, Inst Innovat Drug Design & Evaluat, Sch Pharm, N Jinming Ave, Kaifeng 475004, Henan, Peoples R ChinaWang, Qiang论文数: 0 引用数: 0 h-index: 0机构: South Cent Univ Nationalities, Sch Pharmaceut Sci, 182 Minyuan Rd, Wuhan 430074, Hubei, Peoples R China Henan Univ, Inst Innovat Drug Design & Evaluat, Sch Pharm, N Jinming Ave, Kaifeng 475004, Henan, Peoples R ChinaYan, Lin论文数: 0 引用数: 0 h-index: 0机构: Henan Univ, Inst Innovat Drug Design & Evaluat, Sch Pharm, N Jinming Ave, Kaifeng 475004, Henan, Peoples R China Zhengzhou Univ, Key Lab Adv Drug Preparat Technol, Minist Educ, Zhengzhou 450001, Henan, Peoples R China Henan Univ, Inst Innovat Drug Design & Evaluat, Sch Pharm, N Jinming Ave, Kaifeng 475004, Henan, Peoples R ChinaQian, Hai论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Ctr Drug Discovery, State Key Lab Nat Med, 24 Tongjiaxiang, Nanjing 210009, Jiangsu, Peoples R China Henan Univ, Inst Innovat Drug Design & Evaluat, Sch Pharm, N Jinming Ave, Kaifeng 475004, Henan, Peoples R China
- [6] Trisubstituted pyrimidines as transient receptor potential vanilloid 1 (TRPV1) antagonists with improved solubilityBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2007, 17 (23) : 6539 - 6545Wang, Xianghong论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Chem Res & Discovery, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Chem Res & Discovery, Thousand Oaks, CA 91320 USAChakrabarti, Partha P.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Chem Res & Discovery, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Chem Res & Discovery, Thousand Oaks, CA 91320 USAOgnyanov, Vassil I.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Chem Res & Discovery, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Chem Res & Discovery, Thousand Oaks, CA 91320 USAPettus, Liping H.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Chem Res & Discovery, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Chem Res & Discovery, Thousand Oaks, CA 91320 USATamir, Rami论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Neurosci, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Chem Res & Discovery, Thousand Oaks, CA 91320 USATan, Helming论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Chem Res & Discovery, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Chem Res & Discovery, Thousand Oaks, CA 91320 USATang, Phi论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Chem Res & Discovery, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Chem Res & Discovery, Thousand Oaks, CA 91320 USATreanor, James J. S.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Neurosci, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Chem Res & Discovery, Thousand Oaks, CA 91320 USAGavva, Narender R.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Neurosci, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Chem Res & Discovery, Thousand Oaks, CA 91320 USANorman, Mark H.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Chem Res & Discovery, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Chem Res & Discovery, Thousand Oaks, CA 91320 USA
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