Novel Inhibitors of Microtubule Affinity-Regulating Kinase 4 for Vascular Cognitive Impairment

被引:0
|
作者
Vohra, Manu [1 ]
Cohn, Whitaker [1 ]
Campagna, Jesus [1 ]
John, Varghese [1 ]
Hinman, Jason D. [1 ]
机构
[1] Univ Calif Los Angeles, Los Angeles, CA USA
关键词
D O I
暂无
中图分类号
R74 [神经病学与精神病学];
学科分类号
摘要
M144
引用
收藏
页码:S75 / S75
页数:1
相关论文
共 50 条
  • [1] Microtubule Affinity-Regulating Kinase 4: Structure, Function, and Regulation
    Naz, Farha
    Anjum, Farah
    Islam, Asimul
    Ahmad, Faizan
    Hassan, Md. Imtaiyaz
    CELL BIOCHEMISTRY AND BIOPHYSICS, 2013, 67 (02) : 485 - 499
  • [2] Microtubule Affinity-Regulating Kinase 4: Structure, Function, and Regulation
    Farha Naz
    Farah Anjum
    Asimul Islam
    Faizan Ahmad
    Md. Imtaiyaz Hassan
    Cell Biochemistry and Biophysics, 2013, 67 : 485 - 499
  • [3] Atypical PKC phosphorylates microtubule affinity-regulating kinase 4 in vitro
    Naz, Farha
    Islam, Asimul
    Ahmad, Faizan
    Hassan, Md. Imtaiyaz
    MOLECULAR AND CELLULAR BIOCHEMISTRY, 2015, 410 (1-2) : 223 - 228
  • [4] Human microtubule affinity-regulating kinase 4 is stable at extremes of pH
    Naz, Farha
    Singh, Parvesh
    Islam, Asimul
    Ahmad, Faizan
    Hassan, Md. Imtaiyaz
    JOURNAL OF BIOMOLECULAR STRUCTURE & DYNAMICS, 2016, 34 (06): : 1241 - 1251
  • [5] Atypical PKC phosphorylates microtubule affinity-regulating kinase 4 in vitro
    Farha Naz
    Asimul Islam
    Faizan Ahmad
    Md. Imtaiyaz Hassan
    Molecular and Cellular Biochemistry, 2015, 410 : 223 - 228
  • [6] Research Progress of Microtubule Affinity-regulating Kinase 4 as Drug Target
    Zhou Jian
    Ye He-Yang
    Yin Xiu-Shan
    Li Jian
    PROGRESS IN BIOCHEMISTRY AND BIOPHYSICS, 2022, 49 (08) : 1422 - 1430
  • [7] Evaluation of human microtubule affinity-regulating kinase 4 inhibitors: fluorescence binding studies, enzyme, and cell assays
    Naz, Farha
    Sami, Neha
    Naqvi, Abu Turab
    Islam, Asimul
    Ahmad, Faizan
    Hassan, Md. Imtaiyaz
    JOURNAL OF BIOMOLECULAR STRUCTURE & DYNAMICS, 2017, 35 (14): : 3194 - 3203
  • [8] Therapeutic targeting of microtubule affinity-regulating kinase 4 in cancer and neurodegenerative diseases
    Alam, Manzar
    Ahmed, Sarfraz
    Abid, Mohammad
    Hasan, Gulam Mustafa
    Islam, Asimul
    Hassan, Md. Imtaiyaz
    JOURNAL OF CELLULAR BIOCHEMISTRY, 2023, 124 (09) : 1223 - 1240
  • [9] PKR-inhibitor binds efficiently with human microtubule affinity-regulating kinase 4
    Naz, Farha
    Shahbaaz, Mohd.
    Khan, Shama
    Bisetty, Krishna
    Islam, Asimul
    Ahmad, Faizan
    Hassan, Md. Imtaiyaz
    JOURNAL OF MOLECULAR GRAPHICS & MODELLING, 2015, 62 : 245 - 252
  • [10] Synthesis, Structural Modification, and Bioactivity Evaluation of Substituted Acridones as Potent Microtubule Affinity-Regulating Kinase 4 Inhibitors
    Voura, Maria
    Anwar, Saleha
    Sigala, Ioanna
    Parasidou, Eleftheria
    Fragoulidou, Souzanna
    Hassan, Md. Imtaiyaz
    Sarli, Vasiliki
    ACS PHARMACOLOGY & TRANSLATIONAL SCIENCE, 2023, 6 (07) : 1052 - 1074