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- [1] AP26113 is a dual ALK/EGFR inhibitor: Characterization against EGFR T790M in cell and mouse models of NSCLCCANCER RESEARCH, 2012, 72Rivera, Victor M.论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Cambridge, MA USA ARIAD Pharmaceut Inc, Cambridge, MA USAWang, Frank论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Cambridge, MA USA ARIAD Pharmaceut Inc, Cambridge, MA USAAnjum, Rana论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Cambridge, MA USA ARIAD Pharmaceut Inc, Cambridge, MA USAZhang, Sen论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Cambridge, MA USA ARIAD Pharmaceut Inc, Cambridge, MA USASquillace, Rachel论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Cambridge, MA USA ARIAD Pharmaceut Inc, Cambridge, MA USAKeats, Jeffrey论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Cambridge, MA USA ARIAD Pharmaceut Inc, Cambridge, MA USAMiller, David论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Cambridge, MA USA ARIAD Pharmaceut Inc, Cambridge, MA USANing, Yaoyu论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Cambridge, MA USA ARIAD Pharmaceut Inc, Cambridge, MA USAWardwell, Scott D.论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Cambridge, MA USA ARIAD Pharmaceut Inc, Cambridge, MA USAMoran, Lauren论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Cambridge, MA USA ARIAD Pharmaceut Inc, Cambridge, MA USAMiret, Juan论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Cambridge, MA USA ARIAD Pharmaceut Inc, Cambridge, MA USANarasimhan, Narayana论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Cambridge, MA USA ARIAD Pharmaceut Inc, Cambridge, MA USADalgarno, David论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Cambridge, MA USA ARIAD Pharmaceut Inc, Cambridge, MA USAClackson, Tim论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Cambridge, MA USA ARIAD Pharmaceut Inc, Cambridge, MA USAShakepeare, William C.论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Cambridge, MA USA ARIAD Pharmaceut Inc, Cambridge, MA USA
- [2] Discovery of a potent dual ALK and EGFR T790M inhibitorEUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 136 : 497 - 510Jang, Jaebong论文数: 0 引用数: 0 h-index: 0机构: Harvard Med Sch, Dept Biol Chem & Mol Pharmacol, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02215 USA Harvard Med Sch, Dept Biol Chem & Mol Pharmacol, Boston, MA 02115 USASon, Jung Beom论文数: 0 引用数: 0 h-index: 0机构: Daegu Gyeongbuk Med Innovat Fdn, New Drug Dev Ctr, Daegu 41061, South Korea Harvard Med Sch, Dept Biol Chem & Mol Pharmacol, Boston, MA 02115 USATo, Ciric论文数: 0 引用数: 0 h-index: 0机构: Harvard Med Sch, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USA Harvard Med Sch, Dept Biol Chem & Mol Pharmacol, Boston, MA 02115 USABahcall, Magda论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Lowe Ctr Thorac Oncol, Boston, MA 02215 USA Harvard Med Sch, Dept Biol Chem & Mol Pharmacol, Boston, MA 02115 USAKim, So Young论文数: 0 引用数: 0 h-index: 0机构: Daegu Gyeongbuk Med Innovat Fdn, New Drug Dev Ctr, Daegu 41061, South Korea Harvard Med Sch, Dept Biol Chem & Mol Pharmacol, Boston, MA 02115 USAKang, Seock Yong论文数: 0 引用数: 0 h-index: 0机构: Daegu Gyeongbuk Med Innovat Fdn, New Drug Dev Ctr, Daegu 41061, South Korea Harvard Med Sch, Dept Biol Chem & Mol Pharmacol, Boston, MA 02115 USAMushajiang, Mierzhati论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Lowe Ctr Thorac Oncol, Boston, MA 02215 USA Harvard Med Sch, Dept Biol Chem & Mol Pharmacol, Boston, MA 02115 USALee, Younho论文数: 0 引用数: 0 h-index: 0机构: Daegu Gyeongbuk Med Innovat Fdn, New Drug Dev Ctr, Daegu 41061, South Korea Harvard Med Sch, Dept Biol Chem & Mol Pharmacol, Boston, MA 02115 USAJanne, Pasi A.论文数: 0 引用数: 0 h-index: 0机构: Harvard Med Sch, Boston, MA 02115 USA Dana Farber Canc Inst, Lowe Ctr Thorac Oncol, Boston, MA 02215 USA Dana Farber Canc Inst, Belfer Ctr Appl Canc Sci, Boston, MA 02215 USA Brigham & Womens Hosp, Dept Med, 75 Francis St, Boston, MA 02115 USA Harvard Med Sch, Dept Biol Chem & Mol Pharmacol, Boston, MA 02115 USAChoi, Hwan Geun论文数: 0 引用数: 0 h-index: 0机构: Daegu Gyeongbuk Med Innovat Fdn, New Drug Dev Ctr, Daegu 41061, South Korea Harvard Med Sch, Dept Biol Chem & Mol Pharmacol, Boston, MA 02115 USAGray, Nathanael S.论文数: 0 引用数: 0 h-index: 0机构: Harvard Med Sch, Dept Biol Chem & Mol Pharmacol, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02215 USA Harvard Med Sch, Dept Biol Chem & Mol Pharmacol, Boston, MA 02115 USA
- [3] The Dual ALK/EGFR Inhibitor AP26113 Also Potently Inhibits Activated and Gatekeeper Mutant Forms of ROS1EUROPEAN JOURNAL OF CANCER, 2012, 48 : 50 - 50Anjum, R.论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Biol, Cambridge, MA 02139 USA ARIAD Pharmaceut Inc, Biol, Cambridge, MA 02139 USAZhang, S.论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Biol, Cambridge, MA 02139 USA ARIAD Pharmaceut Inc, Biol, Cambridge, MA 02139 USASquillace, R.论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Biol, Cambridge, MA 02139 USA ARIAD Pharmaceut Inc, Biol, Cambridge, MA 02139 USAClackson, T.论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Biol, Cambridge, MA 02139 USA ARIAD Pharmaceut Inc, Biol, Cambridge, MA 02139 USAGarner, A. P.论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Biol, Cambridge, MA 02139 USA ARIAD Pharmaceut Inc, Biol, Cambridge, MA 02139 USARivera, V. M.论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Biol, Cambridge, MA 02139 USA ARIAD Pharmaceut Inc, Biol, Cambridge, MA 02139 USA
- [4] The Potent ALK Inhibitor Brigatinib (AP26113) Overcomes Mechanisms of Resistance to First- and Second-Generation ALK Inhibitors in Preclinical ModelsCLINICAL CANCER RESEARCH, 2016, 22 (22) : 5527 - 5538Zhang, Sen论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Cambridge, MA USA ARIAD Pharmaceut Inc, Cambridge, MA USAAnjum, Rana论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Cambridge, MA USA ARIAD Pharmaceut Inc, Cambridge, MA USASquillace, Rachel论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Cambridge, MA USA ARIAD Pharmaceut Inc, Cambridge, MA USANadworny, Sara论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Cambridge, MA USA ARIAD Pharmaceut Inc, Cambridge, MA USAZhou, Tianjun论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Cambridge, MA USA ARIAD Pharmaceut Inc, Cambridge, MA USAKeats, Jeff论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Cambridge, MA USA ARIAD Pharmaceut Inc, Cambridge, MA USANing, Yaoyu论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Cambridge, MA USA ARIAD Pharmaceut Inc, Cambridge, MA USAWardwell, Scott D.论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Cambridge, MA USA ARIAD Pharmaceut Inc, Cambridge, MA USAMiller, David论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Cambridge, MA USA ARIAD Pharmaceut Inc, Cambridge, MA USASong, Youngchul论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Cambridge, MA USA ARIAD Pharmaceut Inc, Cambridge, MA USAEichinger, Lindsey论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Cambridge, MA USA ARIAD Pharmaceut Inc, Cambridge, MA USAMoran, Lauren论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Cambridge, MA USA ARIAD Pharmaceut Inc, Cambridge, MA USAHuang, Wei-Sheng论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Cambridge, MA USA ARIAD Pharmaceut Inc, Cambridge, MA USALiu, Shuangying论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Cambridge, MA USA ARIAD Pharmaceut Inc, Cambridge, MA USAZou, Dong论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Cambridge, MA USA ARIAD Pharmaceut Inc, Cambridge, MA USAWang, Yihan论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Cambridge, MA USA ARIAD Pharmaceut Inc, Cambridge, MA USAMohemmad, Qurish论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Cambridge, MA USA ARIAD Pharmaceut Inc, Cambridge, MA USAJang, Hyun Gyung论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Cambridge, MA USA ARIAD Pharmaceut Inc, Cambridge, MA USAYe, Emily论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Cambridge, MA USA ARIAD Pharmaceut Inc, Cambridge, MA USANarasimhan, Narayana论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Cambridge, MA USA ARIAD Pharmaceut Inc, Cambridge, MA USAWang, Frank论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Cambridge, MA USA ARIAD Pharmaceut Inc, Cambridge, MA USAMiret, Juan论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Cambridge, MA USA ARIAD Pharmaceut Inc, Cambridge, MA USAZhu, Xiaotian论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Cambridge, MA USA ARIAD Pharmaceut Inc, Cambridge, MA USAClackson, Tim论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Cambridge, MA USA ARIAD Pharmaceut Inc, Cambridge, MA USADalgarno, David论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Cambridge, MA USA ARIAD Pharmaceut Inc, Cambridge, MA USAShakespeare, William C.论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Cambridge, MA USA ARIAD Pharmaceut Inc, Cambridge, MA USARivera, Victor M.论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Cambridge, MA USA ARIAD Pharmaceut Inc, Cambridge, MA USA
- [5] TAS-2913 is a Mutant Selective EGFR Inhibitor for NSCLC: Characterization Against EGFR T790M in Cell and Xenograft ModelsEUROPEAN JOURNAL OF CANCER, 2012, 48 : 44 - 44Miyadera, K.论文数: 0 引用数: 0 h-index: 0机构: Taiho Pharmaceut Co Ltd, Tsukuba Res Ctr, Tsukuba, Ibaraki, Japan Taiho Pharmaceut Co Ltd, Tsukuba Res Ctr, Tsukuba, Ibaraki, JapanKato, M.论文数: 0 引用数: 0 h-index: 0机构: Taiho Pharmaceut Co Ltd, Tsukuba Res Ctr, Tsukuba, Ibaraki, Japan Taiho Pharmaceut Co Ltd, Tsukuba Res Ctr, Tsukuba, Ibaraki, JapanTakahashi, I.论文数: 0 引用数: 0 h-index: 0机构: Taiho Pharmaceut Co Ltd, Tsukuba Res Ctr, Tsukuba, Ibaraki, Japan Taiho Pharmaceut Co Ltd, Tsukuba Res Ctr, Tsukuba, Ibaraki, JapanIto, K.论文数: 0 引用数: 0 h-index: 0机构: Taiho Pharmaceut Co Ltd, Tsukuba Res Ctr, Tsukuba, Ibaraki, Japan Taiho Pharmaceut Co Ltd, Tsukuba Res Ctr, Tsukuba, Ibaraki, JapanAoyagi, Y.论文数: 0 引用数: 0 h-index: 0机构: Taiho Pharmaceut Co Ltd, Tsukuba Res Ctr, Tsukuba, Ibaraki, Japan Taiho Pharmaceut Co Ltd, Tsukuba Res Ctr, Tsukuba, Ibaraki, JapanFukasawa, K.论文数: 0 引用数: 0 h-index: 0机构: Taiho Pharmaceut Co Ltd, Tsukuba Res Ctr, Tsukuba, Ibaraki, Japan Taiho Pharmaceut Co Ltd, Tsukuba Res Ctr, Tsukuba, Ibaraki, JapanSagara, T.论文数: 0 引用数: 0 h-index: 0机构: Taiho Pharmaceut Co Ltd, Tsukuba Res Ctr, Tsukuba, Ibaraki, Japan Taiho Pharmaceut Co Ltd, Tsukuba Res Ctr, Tsukuba, Ibaraki, JapanYonekura, K.论文数: 0 引用数: 0 h-index: 0机构: Taiho Pharmaceut Co Ltd, Tsukuba Res Ctr, Tsukuba, Ibaraki, Japan Taiho Pharmaceut Co Ltd, Tsukuba Res Ctr, Tsukuba, Ibaraki, JapanIwasawa, Y.论文数: 0 引用数: 0 h-index: 0机构: Taiho Pharmaceut Co Ltd, Tsukuba Res Ctr, Tsukuba, Ibaraki, Japan Taiho Pharmaceut Co Ltd, Tsukuba Res Ctr, Tsukuba, Ibaraki, JapanUtsugi, T.论文数: 0 引用数: 0 h-index: 0机构: Taiho Pharmaceut Co Ltd, Tsukuba Res Ctr, Tsukuba, Ibaraki, Japan Taiho Pharmaceut Co Ltd, Tsukuba Res Ctr, Tsukuba, Ibaraki, Japan
- [6] The potent ALK inhibitor AP26113 can overcome mechanisms of resistance to first- and second-generation ALK TKIs in preclinical modelsCANCER RESEARCH, 2015, 75Zhang, Sen论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Cambridge, MA USA ARIAD Pharmaceut Inc, Cambridge, MA USANadworny, Sara论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Cambridge, MA USA ARIAD Pharmaceut Inc, Cambridge, MA USAWardwell, Scott D.论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Cambridge, MA USA ARIAD Pharmaceut Inc, Cambridge, MA USAEichinger, Lindsey论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Cambridge, MA USA ARIAD Pharmaceut Inc, Cambridge, MA USADas, Biplab论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Cambridge, MA USA ARIAD Pharmaceut Inc, Cambridge, MA USAYe, Emily Y.论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Cambridge, MA USA ARIAD Pharmaceut Inc, Cambridge, MA USAHodgson, J. Graeme论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Cambridge, MA USA ARIAD Pharmaceut Inc, Cambridge, MA USARivera, Victor M.论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Cambridge, MA USA ARIAD Pharmaceut Inc, Cambridge, MA USA
- [7] Discovery of AP26113, a potent, orally active inhibitor of anaplastic lymphoma kinase and clinically relevant mutantsCANCER RESEARCH, 2015, 75Huang, Wei-Sheng论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA ARIAD Pharmaceut Inc, Cambridge, MA 02139 USALi, Feng论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA ARIAD Pharmaceut Inc, Cambridge, MA 02139 USACai, Lisi论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA ARIAD Pharmaceut Inc, Cambridge, MA 02139 USAXu, Yongjin论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA ARIAD Pharmaceut Inc, Cambridge, MA 02139 USAZhang, Sen论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA ARIAD Pharmaceut Inc, Cambridge, MA 02139 USAWardwell, Scott D.论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA ARIAD Pharmaceut Inc, Cambridge, MA 02139 USANing, Yaoyu论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA ARIAD Pharmaceut Inc, Cambridge, MA 02139 USAKohlmann, Anna论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA ARIAD Pharmaceut Inc, Cambridge, MA 02139 USAZhou, Tianjun论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA ARIAD Pharmaceut Inc, Cambridge, MA 02139 USAYe, Emily Y.论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA ARIAD Pharmaceut Inc, Cambridge, MA 02139 USAZhu, Xiaotian论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA ARIAD Pharmaceut Inc, Cambridge, MA 02139 USANarasimhan, Narayana I.论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA ARIAD Pharmaceut Inc, Cambridge, MA 02139 USAClackson, Tim论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA ARIAD Pharmaceut Inc, Cambridge, MA 02139 USARivera, Victor M.论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA ARIAD Pharmaceut Inc, Cambridge, MA 02139 USADalgarno, David论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA ARIAD Pharmaceut Inc, Cambridge, MA 02139 USAShakespeare, William C.论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
- [8] A FIRST-IN-HUMAN DOSE-FINDING STUDY OF THE ALK/EGFR INHIBITOR AP26113 IN PATIENTS WITH ADVANCED MALIGNANCIESANNALS OF ONCOLOGY, 2012, 23 : 152 - 152Gettinger, S.论文数: 0 引用数: 0 h-index: 0机构: Yale Univ, Sch Med, Sect Med Oncol, New Haven, CT USA Yale Univ, Sch Med, Sect Med Oncol, New Haven, CT USAWeiss, G. J.论文数: 0 引用数: 0 h-index: 0机构: Scottsdale Healthcare, Virginia G Piper Canc Ctr Clin Trials, Scottsdale, AZ USA Yale Univ, Sch Med, Sect Med Oncol, New Haven, CT USASalgia, R.论文数: 0 引用数: 0 h-index: 0机构: Univ Chicago, Dept Med, Hematol Oncol Sect, Chicago, IL 60637 USA Yale Univ, Sch Med, Sect Med Oncol, New Haven, CT USABazhenova, L.论文数: 0 引用数: 0 h-index: 0机构: Univ Calif San Diego, Moores Canc Ctr, Div Hematol Oncol, La Jolla, CA 92093 USA Yale Univ, Sch Med, Sect Med Oncol, New Haven, CT USANarasimhan, N. I.论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, DMPK, Cambridge, MA USA Yale Univ, Sch Med, Sect Med Oncol, New Haven, CT USADorer, J.论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Biostat, Cambridge, MA USA Yale Univ, Sch Med, Sect Med Oncol, New Haven, CT USARivera, V. M.论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Biol, Cambridge, MA USA Yale Univ, Sch Med, Sect Med Oncol, New Haven, CT USAZhang, J.论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Clin Res, Cambridge, MA USA Yale Univ, Sch Med, Sect Med Oncol, New Haven, CT USAClackson, T.论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Res & Dev, Cambridge, MA USA Yale Univ, Sch Med, Sect Med Oncol, New Haven, CT USAHaluska, F.论文数: 0 引用数: 0 h-index: 0机构: ARIAD Pharmaceut Inc, Clin Res, Cambridge, MA USA Yale Univ, Sch Med, Sect Med Oncol, New Haven, CT USAShaw, A. T.论文数: 0 引用数: 0 h-index: 0机构: Massachusetts Gen Hosp, Boston, MA 02114 USA Yale Univ, Sch Med, Sect Med Oncol, New Haven, CT USACamidge, D. R.论文数: 0 引用数: 0 h-index: 0机构: Univ Colorado, Ctr Canc, Aurora, CO USA Yale Univ, Sch Med, Sect Med Oncol, New Haven, CT USA
- [9] Molecular dynamics and pharmacophore modelling studies of different subtype (ALK and EGFR (T790M)) inhibitors in NSCLCSAR AND QSAR IN ENVIRONMENTAL RESEARCH, 2017, 28 (03) : 221 - 233Singh, P. K.论文数: 0 引用数: 0 h-index: 0机构: Punjabi Univ, Dept Pharmaceut Sci & Drug Res, MML, Patiala, Punjab, India Punjabi Univ, Dept Pharmaceut Sci & Drug Res, MML, Patiala, Punjab, IndiaSilakari, O.论文数: 0 引用数: 0 h-index: 0机构: Punjabi Univ, Dept Pharmaceut Sci & Drug Res, MML, Patiala, Punjab, India Punjabi Univ, Dept Pharmaceut Sci & Drug Res, MML, Patiala, Punjab, India
- [10] Amplification of EGFR T790M causes resistance to an irreversible EGFR inhibitorOncogene, 2010, 29 : 2346 - 2356D Ercan论文数: 0 引用数: 0 h-index: 0机构: Lowe Center for Thoracic Oncology,Department of Medical OncologyK Zejnullahu论文数: 0 引用数: 0 h-index: 0机构: Lowe Center for Thoracic Oncology,Department of Medical OncologyK Yonesaka论文数: 0 引用数: 0 h-index: 0机构: Lowe Center for Thoracic Oncology,Department of Medical OncologyY Xiao论文数: 0 引用数: 0 h-index: 0机构: Lowe Center for Thoracic Oncology,Department of Medical OncologyM Capelletti论文数: 0 引用数: 0 h-index: 0机构: Lowe Center for Thoracic Oncology,Department of Medical OncologyA Rogers论文数: 0 引用数: 0 h-index: 0机构: Lowe Center for Thoracic Oncology,Department of Medical OncologyE Lifshits论文数: 0 引用数: 0 h-index: 0机构: Lowe Center for Thoracic Oncology,Department of Medical OncologyA Brown论文数: 0 引用数: 0 h-index: 0机构: Lowe Center for Thoracic Oncology,Department of Medical OncologyC Lee论文数: 0 引用数: 0 h-index: 0机构: Lowe Center for Thoracic Oncology,Department of Medical OncologyJ G Christensen论文数: 0 引用数: 0 h-index: 0机构: Lowe Center for Thoracic Oncology,Department of Medical OncologyD J Kwiatkowski论文数: 0 引用数: 0 h-index: 0机构: Lowe Center for Thoracic Oncology,Department of Medical OncologyJ A Engelman论文数: 0 引用数: 0 h-index: 0机构: Lowe Center for Thoracic Oncology,Department of Medical OncologyP A Jänne论文数: 0 引用数: 0 h-index: 0机构: Lowe Center for Thoracic Oncology,Department of Medical Oncology