Microwave-assisted synthesis of 5-carboxymethoxy-N-acetyltryptamine derivatives

被引：29
|
作者：
Fînaru, A
Berthault, A
Besson, T
Guillaumet, G
Berteina-Raboin, S
机构：
[1] Univ Orleans, CNRS, UMR 6005, Inst Chim Organ & Analyt, F-45067 Orleans 2, France
[2] Univ Rochelle, UFR Sci Fondamentales & Sci Ingn, Grp Chim Organ, EA3169,Lab Genie Prot & Cellulaire, F-17042 La Rochelle 1, France
来源：
TETRAHEDRON LETTERS | 2002年 / 43卷 / 05期
关键词：
melatoninergic analogs; microwave irradiation; palladium coupling;
D O I：
10.1016/S0040-4039(01)02273-0
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
The synthesis of the indole core structure was investigated using microwave irradiation. The experimental microwave conditions described allow significant rate enhancements and good yields compared to conventional reaction conditions. (C) 2002 Elsevier Science Ltd. All rights reserved.
引用
收藏
页码：787 / 790
页数：4
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