Synthesis of (1H)-3,4-dihydropyrrolo[2,1-c][1,4]oxazin-1-one derivatives

被引：0
|
作者：
Fu, DC [1 ]
Yu, H [1 ]
Zhang, SF [1 ]
机构：
[1] Shenyang Pharmaceut Univ, Shenyang 110016, Peoples R China
来源：
CHINESE CHEMICAL LETTERS | 2002年 / 13卷 / 11期
关键词：
(1H)-3,4-dihydropyrrolo[2,1-c][1,4]oxazin-1-; synthesis;
D O I：
暂无
中图分类号：
O6 [化学];
学科分类号：
0703 ;
摘要：
In search of new anti-inflammatory and analgesic agents, (1H)-3,4-dihydro- pyrrolo [2,1-c][1,4]oxazin-1-one (3) and its acyl derivatives were designed and prepared. compound 3 was prepared by treatment of methyl 1-(2-bromoethyl) pyrrole-2-carboxy late with silver oxide and its derivatives were obtained by Friedel-Cralles reaction. Nine of 6-acyl derivatives of compound 3 were prepared.
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页码：1051 / 1054
页数：4
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