Efficient synthesis of C-11 functionalized steroids

被引：6

作者：

Bazzini, Patrick

Ibrahim-Ouali, Malika

Pellissier, Helene

Santelli, Maurice

机构：

[1] CNRS, UMR 6180, F-13397 Marseille 20, France

[2] Univ Aix Marseille 3, CNRS, Fac Sci & Tech St Jerome, Lab Synthese Organ Associe, Marseille 20, France

来源：

STEROIDS | 2006年 / 71卷 / 06期

关键词：

non-natural steroids; functionalization; C-11 substituted steroids;

D O I：

10.1016/j.steroids.2006.01.003

中图分类号：

Q5 [生物化学]; Q7 [分子生物学];

学科分类号：

071010 ; 081704 ;

摘要：

An efficient synthesis from readily available materials of numerous steroids functionalized at C-11 position, interesting from a biological point of view, is described using our general approach. The characteristic H-1 and C-13 NMR spectroscopic features of the synthesized steroids are reported. (c) 2006 Elsevier Inc. All rights reserved.

引用

页码：459 / 468

页数：10

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