An alternative synthesis of a potent GPIIb/IIIa receptor antagonist

被引：0
|
作者：
Hayes, JF [1 ]
机构：
[1] SmithKline Beecham Pharmaceut, Tonbridge TN11 9AN, Kent, England
来源：
SYNLETT | 1999年
关键词：
benzodiazepine; cyclization; quinone; hydroquinone; oxidation;
D O I：
暂无
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
A key intermediate to SE-214857 was prepared via an oxidative cyclization of a hydroquinone with a flanking aspartate side chain using Fremy's salt.
引用
收藏
页码：865 / 866
页数：2
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