Synthesis and evaluation of new triazolobenzothiazole derivatives as potential anti-tubercular agents

被引：0
|
作者：
Paranjape, SD [1 ]
Bobade, AS [1 ]
Khadse, BG [1 ]
机构：
[1] Haffkine Inst, Dept Chemotherapy, Bombay 400012, Maharashtra, India
来源：
ARZNEIMITTEL-FORSCHUNG-DRUG RESEARCH | 2001年 / 51卷 / 11期
关键词：
Mycobacterium tuberculosis; sulfonamides; triazolobenzothiazoles; antitubercular activity; S-benzyl derivatives;
D O I：
暂无
中图分类号：
R914 [药物化学];
学科分类号：
100701 ;
摘要：
A series of sulfonamides and S-benzyl derivatives of substituted/unsubstituted S-triazolo-(3,4,-b)-benzothiazole-3-thiones were synthesized. These triazolobenzothiazole derivatives were evaluated for antitubercular activity against H(37)Rv strain of Mycobacterium tuberculosis. A number of promising compounds have been obtained.
引用
收藏
页码：916 / 919
页数：4
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