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- [1] Design, Synthesis, and Activity of a Novel Series of Pyridazine-Based ALK5 InhibitorsACS MEDICINAL CHEMISTRY LETTERS, 2024, 15 (11): : 1925 - 1932Pala, Daniele论文数: 0 引用数: 0 h-index: 0机构: Chiesi Farmaceut SpA, Ctr Ric, I-43122 Parma, Italy Chiesi Farmaceut SpA, Ctr Ric, I-43122 Parma, ItalyRonchi, Paolo论文数: 0 引用数: 0 h-index: 0机构: Chiesi Farmaceut SpA, Ctr Ric, I-43122 Parma, Italy Chiesi Farmaceut SpA, Ctr Ric, I-43122 Parma, ItalyRescigno, Donatella论文数: 0 引用数: 0 h-index: 0机构: Evotec Co, Aptuit, I-37135 Verona, Italy Chiesi Farmaceut SpA, Ctr Ric, I-43122 Parma, ItalyBertani, Barbara论文数: 0 引用数: 0 h-index: 0机构: Evotec Co, Aptuit, I-37135 Verona, Italy Chiesi Farmaceut SpA, Ctr Ric, I-43122 Parma, ItalyCapelli, Anna Maria论文数: 0 引用数: 0 h-index: 0机构: Chiesi Farmaceut SpA, Ctr Ric, I-43122 Parma, Italy Chiesi Farmaceut SpA, Ctr Ric, I-43122 Parma, ItalyGuariento, Sara论文数: 0 引用数: 0 h-index: 0机构: Chiesi Farmaceut SpA, Ctr Ric, I-43122 Parma, Italy Chiesi Farmaceut SpA, Ctr Ric, I-43122 Parma, ItalyMarchini, Gessica论文数: 0 引用数: 0 h-index: 0机构: Chiesi Farmaceut SpA, Ctr Ric, I-43122 Parma, Italy Chiesi Farmaceut SpA, Ctr Ric, I-43122 Parma, ItalyMilioli, Marco论文数: 0 引用数: 0 h-index: 0机构: Chiesi Farmaceut SpA, Ctr Ric, I-43122 Parma, Italy Chiesi Farmaceut SpA, Ctr Ric, I-43122 Parma, ItalyCesari, Nicola论文数: 0 引用数: 0 h-index: 0机构: Chiesi Farmaceut SpA, Ctr Ric, I-43122 Parma, Italy Chiesi Farmaceut SpA, Ctr Ric, I-43122 Parma, ItalyFederico, Giuseppina论文数: 0 引用数: 0 h-index: 0机构: Chiesi Farmaceut SpA, Ctr Ric, I-43122 Parma, Italy Chiesi Farmaceut SpA, Ctr Ric, I-43122 Parma, ItalyGrandi, Andrea论文数: 0 引用数: 0 h-index: 0机构: Chiesi Farmaceut SpA, Ctr Ric, I-43122 Parma, Italy Chiesi Farmaceut SpA, Ctr Ric, I-43122 Parma, ItalyStellari, Franco F.论文数: 0 引用数: 0 h-index: 0机构: Chiesi Farmaceut SpA, Ctr Ric, I-43122 Parma, Italy Chiesi Farmaceut SpA, Ctr Ric, I-43122 Parma, ItalyFernandez, Sergio Xanxo论文数: 0 引用数: 0 h-index: 0机构: Chiesi Farmaceut SpA, Ctr Ric, I-43122 Parma, Italy Chiesi Farmaceut SpA, Ctr Ric, I-43122 Parma, ItalyPappani, Alice论文数: 0 引用数: 0 h-index: 0机构: Chiesi Farmaceut SpA, Ctr Ric, I-43122 Parma, Italy Chiesi Farmaceut SpA, Ctr Ric, I-43122 Parma, ItalyVenturi, Luca论文数: 0 引用数: 0 h-index: 0机构: Chiesi Farmaceut SpA, Ctr Ric, I-43122 Parma, Italy Chiesi Farmaceut SpA, Ctr Ric, I-43122 Parma, ItalyBiagetti, Matteo论文数: 0 引用数: 0 h-index: 0机构: Chiesi Farmaceut SpA, Ctr Ric, I-43122 Parma, Italy Chiesi Farmaceut SpA, Ctr Ric, I-43122 Parma, ItalyCivelli, Maurizio论文数: 0 引用数: 0 h-index: 0机构: Chiesi Farmaceut SpA, Ctr Ric, I-43122 Parma, Italy Chiesi Farmaceut SpA, Ctr Ric, I-43122 Parma, ItalySemeraro, Teresa论文数: 0 引用数: 0 h-index: 0机构: Evotec Co, Aptuit, I-37135 Verona, Italy Chiesi Farmaceut SpA, Ctr Ric, I-43122 Parma, ItalyBianchi, Federica论文数: 0 引用数: 0 h-index: 0机构: Evotec Co, Aptuit, I-37135 Verona, Italy Chiesi Farmaceut SpA, Ctr Ric, I-43122 Parma, ItalyTrist, Iuni M. L.论文数: 0 引用数: 0 h-index: 0机构: Evotec Co, Aptuit, I-37135 Verona, Italy Chiesi Farmaceut SpA, Ctr Ric, I-43122 Parma, ItalyRemelli, Rosaria论文数: 0 引用数: 0 h-index: 0机构: Evotec Co, Aptuit, I-37135 Verona, Italy Chiesi Farmaceut SpA, Ctr Ric, I-43122 Parma, ItalyArmani, Elisabetta论文数: 0 引用数: 0 h-index: 0机构: Chiesi Farmaceut SpA, Ctr Ric, I-43122 Parma, Italy Chiesi Farmaceut SpA, Ctr Ric, I-43122 Parma, ItalyPizzirani, Daniela论文数: 0 引用数: 0 h-index: 0机构: Chiesi Farmaceut SpA, Ctr Ric, I-43122 Parma, Italy Chiesi Farmaceut SpA, Ctr Ric, I-43122 Parma, Italy
- [2] A novel series of cysteine-dependent, allosteric inverse agonists of the nuclear receptor RORγtBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2020, 30 (06)Jiang, Xin论文数: 0 引用数: 0 h-index: 0机构: Reata Pharmaceut Inc, 2801 Gateway Dr,Suite 150, Irving, TX 75063 USA Reata Pharmaceut Inc, 2801 Gateway Dr,Suite 150, Irving, TX 75063 USADulubova, Irina论文数: 0 引用数: 0 h-index: 0机构: Reata Pharmaceut Inc, 2801 Gateway Dr,Suite 150, Irving, TX 75063 USA Reata Pharmaceut Inc, 2801 Gateway Dr,Suite 150, Irving, TX 75063 USAReisman, Scott A.论文数: 0 引用数: 0 h-index: 0机构: Reata Pharmaceut Inc, 2801 Gateway Dr,Suite 150, Irving, TX 75063 USA Reata Pharmaceut Inc, 2801 Gateway Dr,Suite 150, Irving, TX 75063 USAHotema, Martha论文数: 0 引用数: 0 h-index: 0机构: Reata Pharmaceut Inc, 2801 Gateway Dr,Suite 150, Irving, TX 75063 USA Reata Pharmaceut Inc, 2801 Gateway Dr,Suite 150, Irving, TX 75063 USALee, Chun-Yue, I论文数: 0 引用数: 0 h-index: 0机构: Reata Pharmaceut Inc, 2801 Gateway Dr,Suite 150, Irving, TX 75063 USA Reata Pharmaceut Inc, 2801 Gateway Dr,Suite 150, Irving, TX 75063 USALiu, Liping论文数: 0 引用数: 0 h-index: 0机构: Reata Pharmaceut Inc, 2801 Gateway Dr,Suite 150, Irving, TX 75063 USA Reata Pharmaceut Inc, 2801 Gateway Dr,Suite 150, Irving, TX 75063 USAMcCauley, Lyndsey论文数: 0 引用数: 0 h-index: 0机构: Reata Pharmaceut Inc, 2801 Gateway Dr,Suite 150, Irving, TX 75063 USA Reata Pharmaceut Inc, 2801 Gateway Dr,Suite 150, Irving, TX 75063 USATrevino, Isaac论文数: 0 引用数: 0 h-index: 0机构: Reata Pharmaceut Inc, 2801 Gateway Dr,Suite 150, Irving, TX 75063 USA Reata Pharmaceut Inc, 2801 Gateway Dr,Suite 150, Irving, TX 75063 USAFerguson, Deborah A.论文数: 0 引用数: 0 h-index: 0机构: Reata Pharmaceut Inc, 2801 Gateway Dr,Suite 150, Irving, TX 75063 USA Reata Pharmaceut Inc, 2801 Gateway Dr,Suite 150, Irving, TX 75063 USAEken, Yigitcan论文数: 0 引用数: 0 h-index: 0机构: Michigan State Univ, Dept Chem, 578 South Shaw Lane, E Lansing, MI 48824 USA Reata Pharmaceut Inc, 2801 Gateway Dr,Suite 150, Irving, TX 75063 USAWilson, Angela K.论文数: 0 引用数: 0 h-index: 0机构: Michigan State Univ, Dept Chem, 578 South Shaw Lane, E Lansing, MI 48824 USA Reata Pharmaceut Inc, 2801 Gateway Dr,Suite 150, Irving, TX 75063 USAWigley, W. Christian论文数: 0 引用数: 0 h-index: 0机构: Reata Pharmaceut Inc, 2801 Gateway Dr,Suite 150, Irving, TX 75063 USA Reata Pharmaceut Inc, 2801 Gateway Dr,Suite 150, Irving, TX 75063 USAVisnick, Melean论文数: 0 引用数: 0 h-index: 0机构: Reata Pharmaceut Inc, 2801 Gateway Dr,Suite 150, Irving, TX 75063 USA Reata Pharmaceut Inc, 2801 Gateway Dr,Suite 150, Irving, TX 75063 USA
- [3] Discovery of carbazole carboxamides as novel RORγt inverse agonistsEUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 148 : 465 - 476Huang, Yafei论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Sch Pharm, Dept Med Chem, 826 Zhangheng Rd, Shanghai 201203, Peoples R China Fudan Univ, Sch Pharm, Dept Med Chem, 826 Zhangheng Rd, Shanghai 201203, Peoples R ChinaYu, Mingcheng论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Sch Pharm, Dept Med Chem, 826 Zhangheng Rd, Shanghai 201203, Peoples R China Fudan Univ, Sch Pharm, Dept Med Chem, 826 Zhangheng Rd, Shanghai 201203, Peoples R ChinaSun, Nannan论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Sch Pharm, Dept Med Chem, 826 Zhangheng Rd, Shanghai 201203, Peoples R China Fudan Univ, Sch Pharm, Dept Med Chem, 826 Zhangheng Rd, Shanghai 201203, Peoples R ChinaTang, Ting论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Sch Pharm, Dept Med Chem, 826 Zhangheng Rd, Shanghai 201203, Peoples R China Fudan Univ, Sch Pharm, Dept Med Chem, 826 Zhangheng Rd, Shanghai 201203, Peoples R ChinaYu, Fazhi论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Sch Pharm, Dept Med Chem, 826 Zhangheng Rd, Shanghai 201203, Peoples R China Fudan Univ, Sch Pharm, Dept Med Chem, 826 Zhangheng Rd, Shanghai 201203, Peoples R ChinaSong, Xiaoxia论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Sch Pharm, Dept Med Chem, 826 Zhangheng Rd, Shanghai 201203, Peoples R China Fudan Univ, Sch Pharm, Dept Med Chem, 826 Zhangheng Rd, Shanghai 201203, Peoples R ChinaXie, Qiong论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Sch Pharm, Dept Med Chem, 826 Zhangheng Rd, Shanghai 201203, Peoples R China Fudan Univ, Sch Pharm, Dept Med Chem, 826 Zhangheng Rd, Shanghai 201203, Peoples R ChinaFu, Wei论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Sch Pharm, Dept Med Chem, 826 Zhangheng Rd, Shanghai 201203, Peoples R China Fudan Univ, Sch Pharm, Dept Med Chem, 826 Zhangheng Rd, Shanghai 201203, Peoples R ChinaShao, Liming论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Sch Pharm, Dept Med Chem, 826 Zhangheng Rd, Shanghai 201203, Peoples R China Fudan Univ, Sch Pharm, Dept Med Chem, 826 Zhangheng Rd, Shanghai 201203, Peoples R ChinaWang, Yonghui论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Sch Pharm, Dept Med Chem, 826 Zhangheng Rd, Shanghai 201203, Peoples R China Fudan Univ, Sch Pharm, Dept Med Chem, 826 Zhangheng Rd, Shanghai 201203, Peoples R China
- [4] Computer-Aided Discovery of Novel Human RORγ Inverse AgonistsFASEB JOURNAL, 2020, 34Huang, Mian论文数: 0 引用数: 0 h-index: 0机构: Kansas State Univ, Manhattan, KS 66506 USA Kansas State Univ, Manhattan, KS 66506 USABolin, Shelby论文数: 0 引用数: 0 h-index: 0机构: Kansas State Univ, Manhattan, KS 66506 USA Kansas State Univ, Manhattan, KS 66506 USAMiller, Hannah论文数: 0 引用数: 0 h-index: 0机构: Kansas State Univ, Manhattan, KS 66506 USA Kansas State Univ, Manhattan, KS 66506 USADykeman, Anna论文数: 0 引用数: 0 h-index: 0机构: Kansas State Univ, Manhattan, KS 66506 USA Kansas State Univ, Manhattan, KS 66506 USANg, Ho论文数: 0 引用数: 0 h-index: 0机构: Kansas State Univ, Manhattan, KS 66506 USA Kansas State Univ, Manhattan, KS 66506 USA
- [5] Discovery of novel pyrazole-containing benzamides as potent RORγ inverse agonistsBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2015, 25 (15) : 2985 - 2990Wang, Tao论文数: 0 引用数: 0 h-index: 0机构: Biogen, Cambridge Ctr 12, Chem & Mol Therapeut, Cambridge, MA 02142 USA Biogen, Cambridge Ctr 12, Chem & Mol Therapeut, Cambridge, MA 02142 USABanerjee, Daliya论文数: 0 引用数: 0 h-index: 0机构: Biogen, Immunol Discovery, Cambridge, MA 02142 USA Biogen, Cambridge Ctr 12, Chem & Mol Therapeut, Cambridge, MA 02142 USABohnert, Tonika论文数: 0 引用数: 0 h-index: 0机构: Biogen, Cambridge Ctr 12, Chem & Mol Therapeut, Cambridge, MA 02142 USA Biogen, Cambridge Ctr 12, Chem & Mol Therapeut, Cambridge, MA 02142 USAChao, Jianhua论文数: 0 引用数: 0 h-index: 0机构: Biogen, Cambridge Ctr 12, Chem & Mol Therapeut, Cambridge, MA 02142 USA Biogen, Cambridge Ctr 12, Chem & Mol Therapeut, Cambridge, MA 02142 USAEnyedy, Istvan论文数: 0 引用数: 0 h-index: 0机构: Biogen, Cambridge Ctr 12, Chem & Mol Therapeut, Cambridge, MA 02142 USA Biogen, Cambridge Ctr 12, Chem & Mol Therapeut, Cambridge, MA 02142 USAFontenot, Jason论文数: 0 引用数: 0 h-index: 0机构: Biogen, Immunol Discovery, Cambridge, MA 02142 USA Biogen, Cambridge Ctr 12, Chem & Mol Therapeut, Cambridge, MA 02142 USAGuertin, Kevin论文数: 0 引用数: 0 h-index: 0机构: Biogen, Cambridge Ctr 12, Chem & Mol Therapeut, Cambridge, MA 02142 USA Biogen, Cambridge Ctr 12, Chem & Mol Therapeut, Cambridge, MA 02142 USAJones, Howard论文数: 0 引用数: 0 h-index: 0机构: Biogen, Cambridge Ctr 12, Chem & Mol Therapeut, Cambridge, MA 02142 USA Biogen, Cambridge Ctr 12, Chem & Mol Therapeut, Cambridge, MA 02142 USALin, Edward Y.论文数: 0 引用数: 0 h-index: 0机构: Biogen, Cambridge Ctr 12, Chem & Mol Therapeut, Cambridge, MA 02142 USA Biogen, Cambridge Ctr 12, Chem & Mol Therapeut, Cambridge, MA 02142 USAMarcotte, Douglas论文数: 0 引用数: 0 h-index: 0机构: Biogen, Cambridge Ctr 12, Chem & Mol Therapeut, Cambridge, MA 02142 USA Biogen, Cambridge Ctr 12, Chem & Mol Therapeut, Cambridge, MA 02142 USATalreja, Tina论文数: 0 引用数: 0 h-index: 0机构: Biogen, Cambridge Ctr 12, Chem & Mol Therapeut, Cambridge, MA 02142 USA Biogen, Cambridge Ctr 12, Chem & Mol Therapeut, Cambridge, MA 02142 USAVan Vloten, Kurt论文数: 0 引用数: 0 h-index: 0机构: Biogen, Cambridge Ctr 12, Chem & Mol Therapeut, Cambridge, MA 02142 USA Biogen, Cambridge Ctr 12, Chem & Mol Therapeut, Cambridge, MA 02142 USA
- [6] Discovery of Novel Pyridazine-Based Cyclooxygenase-2 Inhibitors with a Promising Gastric Safety ProfileMOLECULES, 2020, 25 (09):Khan, Abida论文数: 0 引用数: 0 h-index: 0机构: Apeejay Stya Univ, Sch Pharmaceut Sci, Sohna Palwal Rd, Sohna 2203, India Apeejay Stya Univ, Sch Pharmaceut Sci, Sohna Palwal Rd, Sohna 2203, IndiaDiwan, Anupama论文数: 0 引用数: 0 h-index: 0机构: Apeejay Stya Univ, Sch Pharmaceut Sci, Sohna Palwal Rd, Sohna 2203, India Apeejay Stya Univ, Sch Pharmaceut Sci, Sohna Palwal Rd, Sohna 2203, IndiaThabet, Hamdy Kh论文数: 0 引用数: 0 h-index: 0机构: Northern Border Univ, Fac Arts & Sci, Dept Chem, Rafha 91911, Saudi Arabia Apeejay Stya Univ, Sch Pharmaceut Sci, Sohna Palwal Rd, Sohna 2203, IndiaImran, Mohd论文数: 0 引用数: 0 h-index: 0机构: Northern Border Univ, Fac Pharm, Dept Pharmaceut Chem, Rafha 91911, Saudi Arabia Apeejay Stya Univ, Sch Pharmaceut Sci, Sohna Palwal Rd, Sohna 2203, India论文数: 引用数: h-index:机构:
- [7] Design and synthesis of novel ROR inverse agonists with a dibenzosilole scaffold as a hydrophobic core structureBIOORGANIC & MEDICINAL CHEMISTRY, 2015, 23 (13) : 2982 - 2988Toyama, Hirozumi论文数: 0 引用数: 0 h-index: 0机构: Univ Tokyo, Inst Mol & Cellular Biosci, Bunkyo Ku, Tokyo 1130032, Japan Univ Tokyo, Inst Mol & Cellular Biosci, Bunkyo Ku, Tokyo 1130032, JapanNakamura, Masaharu论文数: 0 引用数: 0 h-index: 0机构: Univ Tokyo, Inst Mol & Cellular Biosci, Bunkyo Ku, Tokyo 1130032, Japan Univ Tokyo, Inst Mol & Cellular Biosci, Bunkyo Ku, Tokyo 1130032, JapanHashimoto, Yuichi论文数: 0 引用数: 0 h-index: 0机构: Univ Tokyo, Inst Mol & Cellular Biosci, Bunkyo Ku, Tokyo 1130032, Japan Univ Tokyo, Inst Mol & Cellular Biosci, Bunkyo Ku, Tokyo 1130032, JapanFujii, Shinya论文数: 0 引用数: 0 h-index: 0机构: Univ Tokyo, Inst Mol & Cellular Biosci, Bunkyo Ku, Tokyo 1130032, Japan Univ Tokyo, Inst Mol & Cellular Biosci, Bunkyo Ku, Tokyo 1130032, Japan
- [8] Discovery of novel quinoline sulphonamide derivatives as potent, selective and orally active RORγ inverse agonistsBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2019, 29 (14) : 1799 - 1806Amaudrut, Jerome论文数: 0 引用数: 0 h-index: 0机构: Inventiva, 50 Rue Dijon, F-21121 Daix, France Inventiva, 50 Rue Dijon, F-21121 Daix, FranceArgiriadi, Maria A.论文数: 0 引用数: 0 h-index: 0机构: AbbVie, 381 Plantat St, Worcester, MA 01605 USA Inventiva, 50 Rue Dijon, F-21121 Daix, FranceBarth, Martine论文数: 0 引用数: 0 h-index: 0机构: Inventiva, 50 Rue Dijon, F-21121 Daix, France Inventiva, 50 Rue Dijon, F-21121 Daix, FranceBreinlinger, Eric C.论文数: 0 引用数: 0 h-index: 0机构: AbbVie, 381 Plantat St, Worcester, MA 01605 USA Inventiva, 50 Rue Dijon, F-21121 Daix, FranceBressac, Didier论文数: 0 引用数: 0 h-index: 0机构: Inventiva, 50 Rue Dijon, F-21121 Daix, France Inventiva, 50 Rue Dijon, F-21121 Daix, FranceBroqua, Pierre论文数: 0 引用数: 0 h-index: 0机构: Inventiva, 50 Rue Dijon, F-21121 Daix, France Inventiva, 50 Rue Dijon, F-21121 Daix, FranceCalderwood, David J.论文数: 0 引用数: 0 h-index: 0机构: AbbVie, 100 Res Dr, Worcester, MA 01605 USA Inventiva, 50 Rue Dijon, F-21121 Daix, FranceChatar, Mohamed论文数: 0 引用数: 0 h-index: 0机构: Inventiva, 50 Rue Dijon, F-21121 Daix, France Inventiva, 50 Rue Dijon, F-21121 Daix, FranceCusack, Kevin P.论文数: 0 引用数: 0 h-index: 0机构: AbbVie, 381 Plantat St, Worcester, MA 01605 USA Inventiva, 50 Rue Dijon, F-21121 Daix, FranceGauld, Stephen B.论文数: 0 引用数: 0 h-index: 0机构: AbbVie, 1 North Waukegan Rd, N Chicago, IL 60064 USA Inventiva, 50 Rue Dijon, F-21121 Daix, FranceJacquet, Sebastien论文数: 0 引用数: 0 h-index: 0机构: Inventiva, 50 Rue Dijon, F-21121 Daix, France Inventiva, 50 Rue Dijon, F-21121 Daix, FranceKamath, Rajesh, V论文数: 0 引用数: 0 h-index: 0机构: AbbVie, 100 Res Dr, Worcester, MA 01605 USA Inventiva, 50 Rue Dijon, F-21121 Daix, FranceKort, Michael E.论文数: 0 引用数: 0 h-index: 0机构: AbbVie, 1 North Waukegan Rd, N Chicago, IL 60064 USA Inventiva, 50 Rue Dijon, F-21121 Daix, FranceLepais, Valerie论文数: 0 引用数: 0 h-index: 0机构: Inventiva, 50 Rue Dijon, F-21121 Daix, France Inventiva, 50 Rue Dijon, F-21121 Daix, FranceLuccarini, Jean-Michel论文数: 0 引用数: 0 h-index: 0机构: Inventiva, 50 Rue Dijon, F-21121 Daix, France Inventiva, 50 Rue Dijon, F-21121 Daix, FranceMasson, Philippe论文数: 0 引用数: 0 h-index: 0机构: Inventiva, 50 Rue Dijon, F-21121 Daix, France Inventiva, 50 Rue Dijon, F-21121 Daix, FranceMontalbetti, Christian论文数: 0 引用数: 0 h-index: 0机构: Inventiva, 50 Rue Dijon, F-21121 Daix, France Inventiva, 50 Rue Dijon, F-21121 Daix, FranceMounier, Laurent论文数: 0 引用数: 0 h-index: 0机构: Inventiva, 50 Rue Dijon, F-21121 Daix, France Inventiva, 50 Rue Dijon, F-21121 Daix, FrancePotin, Dominique论文数: 0 引用数: 0 h-index: 0机构: Inventiva, 50 Rue Dijon, F-21121 Daix, France Inventiva, 50 Rue Dijon, F-21121 Daix, FrancePoupardin, Olivia论文数: 0 引用数: 0 h-index: 0机构: Inventiva, 50 Rue Dijon, F-21121 Daix, France Inventiva, 50 Rue Dijon, F-21121 Daix, FranceRouaud, Sylvie论文数: 0 引用数: 0 h-index: 0机构: Inventiva, 50 Rue Dijon, F-21121 Daix, France Inventiva, 50 Rue Dijon, F-21121 Daix, FranceSpitzer, Luc论文数: 0 引用数: 0 h-index: 0机构: Inventiva, 50 Rue Dijon, F-21121 Daix, France Inventiva, 50 Rue Dijon, F-21121 Daix, FranceWallace, Craig D.论文数: 0 引用数: 0 h-index: 0机构: AbbVie, 100 Res Dr, Worcester, MA 01605 USA Inventiva, 50 Rue Dijon, F-21121 Daix, France
- [9] Discovery of novel quinoline sulfonamide derivatives as potent, selective and orally active RORγ inverse agonistsABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2018, 256Potin, Dominique论文数: 0 引用数: 0 h-index: 0机构: Inventiva, Daix, France Inventiva, Daix, FranceAmaudrut, Jerome论文数: 0 引用数: 0 h-index: 0机构: Inventiva, Daix, France Inventiva, Daix, FranceArgiriadi, Maria论文数: 0 引用数: 0 h-index: 0机构: AbbVie, Worcester, MA USA Inventiva, Daix, FranceBarth, Martine论文数: 0 引用数: 0 h-index: 0机构: Inventiva, Daix, France Inventiva, Daix, FranceBreinlinger, Eric论文数: 0 引用数: 0 h-index: 0机构: AbbVie, Worcester, MA USA Inventiva, Daix, FranceBressac, Didier论文数: 0 引用数: 0 h-index: 0机构: Inventiva, Daix, France Inventiva, Daix, FranceBroqua, Pierre论文数: 0 引用数: 0 h-index: 0机构: Inventiva, Daix, France Inventiva, Daix, FranceCalderwood, David论文数: 0 引用数: 0 h-index: 0机构: AbbVie, Worcester, MA USA Inventiva, Daix, FranceChatar, Mohamed论文数: 0 引用数: 0 h-index: 0机构: Inventiva, Daix, France Inventiva, Daix, FranceCusack, Kevin论文数: 0 引用数: 0 h-index: 0机构: AbbVie, Worcester, MA USA Inventiva, Daix, FranceGauld, Stephen论文数: 0 引用数: 0 h-index: 0机构: AbbVie, N Chicago, IL USA Inventiva, Daix, FranceJacquet, Sebastien论文数: 0 引用数: 0 h-index: 0机构: Inventiva, Daix, France Inventiva, Daix, FranceKamath, Rajesh论文数: 0 引用数: 0 h-index: 0机构: AbbVie, Worcester, MA USA Inventiva, Daix, FranceLepais, Valerie论文数: 0 引用数: 0 h-index: 0机构: Inventiva, Daix, France Inventiva, Daix, FranceLuccarini, Jean Michel论文数: 0 引用数: 0 h-index: 0机构: Inventiva, Daix, France Inventiva, Daix, FranceMasson, Philippe论文数: 0 引用数: 0 h-index: 0机构: Inventiva, Daix, France Inventiva, Daix, FranceMontalbetti, Christian论文数: 0 引用数: 0 h-index: 0机构: Inventiva, Daix, France Inventiva, Daix, FranceMounier, Laurent论文数: 0 引用数: 0 h-index: 0机构: Inventiva, Daix, France Inventiva, Daix, FrancePoupardin, Olivia论文数: 0 引用数: 0 h-index: 0机构: Inventiva, Daix, France Inventiva, Daix, FranceRouaud, Sylvie论文数: 0 引用数: 0 h-index: 0机构: Inventiva, Daix, France Inventiva, Daix, FranceWallace, Craig论文数: 0 引用数: 0 h-index: 0机构: AbbVie, Worcester, MA USA Inventiva, Daix, France
- [10] Structure-based design of novel RORgamma inverse agonistsABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2016, 252Zheng, Yajun论文数: 0 引用数: 0 h-index: 0机构: Vitae Pharmaceut, Ft Washington, PA USA Vitae Pharmaceut, Ft Washington, PA USAJia, Lanqi论文数: 0 引用数: 0 h-index: 0机构: Vitae Pharmaceut, Ft Washington, PA USA Vitae Pharmaceut, Ft Washington, PA USAYuan, Jing论文数: 0 引用数: 0 h-index: 0机构: Vitae Pharmaceut, Ft Washington, PA USA Vitae Pharmaceut, Ft Washington, PA USADillard, Lawrence论文数: 0 引用数: 0 h-index: 0机构: Vitae Pharmaceut, Ft Washington, PA USA Vitae Pharmaceut, Ft Washington, PA USAZhuang, Linghang论文数: 0 引用数: 0 h-index: 0机构: Vitae Pharmaceut, Ft Washington, PA USA Vitae Pharmaceut, Ft Washington, PA USAFan, Kristi论文数: 0 引用数: 0 h-index: 0机构: Vitae Pharmaceut, Ft Washington, PA USA Vitae Pharmaceut, Ft Washington, PA USATice, Colin论文数: 0 引用数: 0 h-index: 0机构: Vitae Pharmaceut, Ft Washington, PA USA Vitae Pharmaceut, Ft Washington, PA USADong, Chengguo论文数: 0 引用数: 0 h-index: 0机构: Vitae Pharmaceut, Ft Washington, PA USA Vitae Pharmaceut, Ft Washington, PA USAMarcus, Andrew论文数: 0 引用数: 0 h-index: 0机构: Vitae Pharmaceut, Ft Washington, PA USA Vitae Pharmaceut, Ft Washington, PA USALotesta, Steve论文数: 0 引用数: 0 h-index: 0机构: Vitae Pharmaceut, Ft Washington, PA USA Vitae Pharmaceut, Ft Washington, PA USANoto, Paul论文数: 0 引用数: 0 h-index: 0机构: Vitae Pharmaceut, Ft Washington, PA USA Vitae Pharmaceut, Ft Washington, PA USAMeng, Shi论文数: 0 引用数: 0 h-index: 0机构: Vitae Pharmaceut, Ft Washington, PA USA Vitae Pharmaceut, Ft Washington, PA USALipinski, Kerri论文数: 0 引用数: 0 h-index: 0机构: Vitae Pharmaceut, Ft Washington, PA USA Vitae Pharmaceut, Ft Washington, PA USAKandpal, Geeta论文数: 0 引用数: 0 h-index: 0机构: Vitae Pharmaceut, Ft Washington, PA USA Vitae Pharmaceut, Ft Washington, PA USABukhtiyarov, Yuri论文数: 0 引用数: 0 h-index: 0机构: Vitae Pharmaceut, Ft Washington, PA USA Vitae Pharmaceut, Ft Washington, PA USAZhao, Yi论文数: 0 引用数: 0 h-index: 0机构: Vitae Pharmaceut, Ft Washington, PA USA Vitae Pharmaceut, Ft Washington, PA USALala, Deepak论文数: 0 引用数: 0 h-index: 0机构: Vitae Pharmaceut, Ft Washington, PA USA Vitae Pharmaceut, Ft Washington, PA USAZhou, Jing论文数: 0 引用数: 0 h-index: 0机构: Vitae Pharmaceut, Ft Washington, PA USA Vitae Pharmaceut, Ft Washington, PA USAvan Order, Rebecca论文数: 0 引用数: 0 h-index: 0机构: Vitae Pharmaceut, Ft Washington, PA USA Vitae Pharmaceut, Ft Washington, PA USAChen, Guozhou论文数: 0 引用数: 0 h-index: 0机构: Vitae Pharmaceut, Ft Washington, PA USA Vitae Pharmaceut, Ft Washington, PA USAMckeever, Brian论文数: 0 引用数: 0 h-index: 0机构: Vitae Pharmaceut, Ft Washington, PA USA Vitae Pharmaceut, Ft Washington, PA USAMcGeehan, Gerald论文数: 0 引用数: 0 h-index: 0机构: Vitae Pharmaceut, Ft Washington, PA USA Vitae Pharmaceut, Ft Washington, PA USAClaremon, David论文数: 0 引用数: 0 h-index: 0机构: Vitae Pharmaceut, Ft Washington, PA USA Vitae Pharmaceut, Ft Washington, PA USASingh, Suresh论文数: 0 引用数: 0 h-index: 0机构: Vitae Pharmaceut, Ft Washington, PA USA Vitae Pharmaceut, Ft Washington, PA USA