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- [1] Advances in structure-based drug design of novel bacterial topoisomerase inhibitorsFUTURE MEDICINAL CHEMISTRY, 2010, 2 (11) : 1619 - 1622Widdowson, Katherine论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Antibacterial Discovery Performance Unit, Infect Dis CEDD, Collegeville, PA 19426 USA GlaxoSmithKline, Antibacterial Discovery Performance Unit, Infect Dis CEDD, Collegeville, PA 19426 USAHennessy, Alan论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Antibacterial Discovery Performance Unit, Infect Dis CEDD, Stevenage SG1 2NY, Herts, England GlaxoSmithKline, Antibacterial Discovery Performance Unit, Infect Dis CEDD, Collegeville, PA 19426 USA
- [2] Novel DNA Topoisomerase IIα Inhibitors from Combined Ligand- and Structure-Based Virtual ScreeningPLOS ONE, 2014, 9 (12):Drwal, Malgorzata N.论文数: 0 引用数: 0 h-index: 0机构: UNSW Australia, Sch Med Sci, Dept Pharmacol, Sydney, NSW, Australia UNSW Australia, Sch Med Sci, Dept Pharmacol, Sydney, NSW, AustraliaMarinello, Jessica论文数: 0 引用数: 0 h-index: 0机构: Univ Bologna, Dept Pharm & Biotechnol, Bologna, Italy UNSW Australia, Sch Med Sci, Dept Pharmacol, Sydney, NSW, Australia论文数: 引用数: h-index:机构:Wakelin, Laurence P. G.论文数: 0 引用数: 0 h-index: 0机构: UNSW Australia, Sch Med Sci, Dept Pharmacol, Sydney, NSW, Australia UNSW Australia, Sch Med Sci, Dept Pharmacol, Sydney, NSW, AustraliaCapranico, Giovanni论文数: 0 引用数: 0 h-index: 0机构: Univ Bologna, Dept Pharm & Biotechnol, Bologna, Italy UNSW Australia, Sch Med Sci, Dept Pharmacol, Sydney, NSW, AustraliaGriffith, Renate论文数: 0 引用数: 0 h-index: 0机构: UNSW Australia, Sch Med Sci, Dept Pharmacol, Sydney, NSW, Australia UNSW Australia, Sch Med Sci, Dept Pharmacol, Sydney, NSW, Australia
- [3] Discovery and structure-activity relationships of a novel isothiazolone class of bacterial type II topoisomerase inhibitorsBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2016, 26 (17) : 4179 - 4183Cooper, Ian R.论文数: 0 引用数: 0 h-index: 0机构: Redx Pharma, Alderley Pk, Macclesfield SK10 4TG, Cheshire, England Redx Pharma, Alderley Pk, Macclesfield SK10 4TG, Cheshire, EnglandMcCarroll, Andrew J.论文数: 0 引用数: 0 h-index: 0机构: Redx Pharma, Alderley Pk, Macclesfield SK10 4TG, Cheshire, England Redx Pharma, Alderley Pk, Macclesfield SK10 4TG, Cheshire, EnglandMcGarry, David论文数: 0 引用数: 0 h-index: 0机构: Redx Pharma, Alderley Pk, Macclesfield SK10 4TG, Cheshire, England Redx Pharma, Alderley Pk, Macclesfield SK10 4TG, Cheshire, EnglandKirkham, James论文数: 0 引用数: 0 h-index: 0机构: Redx Pharma, Alderley Pk, Macclesfield SK10 4TG, Cheshire, England Redx Pharma, Alderley Pk, Macclesfield SK10 4TG, Cheshire, EnglandPichowicz, Mark论文数: 0 引用数: 0 h-index: 0机构: Redx Pharma, Alderley Pk, Macclesfield SK10 4TG, Cheshire, England Redx Pharma, Alderley Pk, Macclesfield SK10 4TG, Cheshire, EnglandWalker, Rolf论文数: 0 引用数: 0 h-index: 0机构: Redx Pharma, Alderley Pk, Macclesfield SK10 4TG, Cheshire, England Redx Pharma, Alderley Pk, Macclesfield SK10 4TG, Cheshire, EnglandWarrilow, Catherine论文数: 0 引用数: 0 h-index: 0机构: Redx Pharma, Alderley Pk, Macclesfield SK10 4TG, Cheshire, England Redx Pharma, Alderley Pk, Macclesfield SK10 4TG, Cheshire, EnglandSalisbury, Anne-Marie论文数: 0 引用数: 0 h-index: 0机构: Redx Pharma, Alderley Pk, Macclesfield SK10 4TG, Cheshire, England Redx Pharma, Alderley Pk, Macclesfield SK10 4TG, Cheshire, EnglandSavage, Victoria J.论文数: 0 引用数: 0 h-index: 0机构: Redx Pharma, Alderley Pk, Macclesfield SK10 4TG, Cheshire, England Redx Pharma, Alderley Pk, Macclesfield SK10 4TG, Cheshire, EnglandMoyo, Emmanuel论文数: 0 引用数: 0 h-index: 0机构: Redx Pharma, Alderley Pk, Macclesfield SK10 4TG, Cheshire, England Redx Pharma, Alderley Pk, Macclesfield SK10 4TG, Cheshire, EnglandForward, Henry论文数: 0 引用数: 0 h-index: 0机构: Redx Pharma, Alderley Pk, Macclesfield SK10 4TG, Cheshire, England Redx Pharma, Alderley Pk, Macclesfield SK10 4TG, Cheshire, EnglandCheung, Jonathan论文数: 0 引用数: 0 h-index: 0机构: Redx Pharma, Alderley Pk, Macclesfield SK10 4TG, Cheshire, England Redx Pharma, Alderley Pk, Macclesfield SK10 4TG, Cheshire, EnglandMetzger, Richard论文数: 0 引用数: 0 h-index: 0机构: Redx Pharma, Alderley Pk, Macclesfield SK10 4TG, Cheshire, England Redx Pharma, Alderley Pk, Macclesfield SK10 4TG, Cheshire, EnglandGault, Zoe论文数: 0 引用数: 0 h-index: 0机构: Redx Pharma, Alderley Pk, Macclesfield SK10 4TG, Cheshire, England Redx Pharma, Alderley Pk, Macclesfield SK10 4TG, Cheshire, EnglandNelson, Gary论文数: 0 引用数: 0 h-index: 0机构: Redx Pharma, Alderley Pk, Macclesfield SK10 4TG, Cheshire, England Redx Pharma, Alderley Pk, Macclesfield SK10 4TG, Cheshire, EnglandHughes, Diarmaid论文数: 0 引用数: 0 h-index: 0机构: Uppsala Univ, Dept Med Biochem & Microbiol, Box 582 Biomed Ctr, Uppsala, Sweden Redx Pharma, Alderley Pk, Macclesfield SK10 4TG, Cheshire, EnglandCao, Sha论文数: 0 引用数: 0 h-index: 0机构: Uppsala Univ, Dept Med Biochem & Microbiol, Box 582 Biomed Ctr, Uppsala, Sweden Redx Pharma, Alderley Pk, Macclesfield SK10 4TG, Cheshire, EnglandMaclean, John论文数: 0 引用数: 0 h-index: 0机构: Redx Pharma, Alderley Pk, Macclesfield SK10 4TG, Cheshire, England Redx Pharma, Alderley Pk, Macclesfield SK10 4TG, Cheshire, EnglandCharrier, Cedric论文数: 0 引用数: 0 h-index: 0机构: Redx Pharma, Alderley Pk, Macclesfield SK10 4TG, Cheshire, England Redx Pharma, Alderley Pk, Macclesfield SK10 4TG, Cheshire, EnglandCraighead, Mark论文数: 0 引用数: 0 h-index: 0机构: Redx Pharma, Alderley Pk, Macclesfield SK10 4TG, Cheshire, England Redx Pharma, Alderley Pk, Macclesfield SK10 4TG, Cheshire, EnglandBest, Stuart论文数: 0 引用数: 0 h-index: 0机构: Redx Pharma, Alderley Pk, Macclesfield SK10 4TG, Cheshire, England Redx Pharma, Alderley Pk, Macclesfield SK10 4TG, Cheshire, EnglandStokes, Neil R.论文数: 0 引用数: 0 h-index: 0机构: Redx Pharma, Alderley Pk, Macclesfield SK10 4TG, Cheshire, England Redx Pharma, Alderley Pk, Macclesfield SK10 4TG, Cheshire, EnglandRatcliffe, Andrew J.论文数: 0 引用数: 0 h-index: 0机构: Redx Pharma, Alderley Pk, Macclesfield SK10 4TG, Cheshire, England Redx Pharma, Alderley Pk, Macclesfield SK10 4TG, Cheshire, England
- [4] Discovery and structure-activity relationships of a novel oxazolidinone class of bacterial type II topoisomerase inhibitorsBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2022, 65Lyons, Amanda论文数: 0 引用数: 0 h-index: 0机构: Redx Antiinfect Ltd, Alderley Pk, Mereside SK10 4TG, Cheshire, England Redx Antiinfect Ltd, Alderley Pk, Mereside SK10 4TG, Cheshire, EnglandKirkham, James论文数: 0 引用数: 0 h-index: 0机构: Infex Therapeut Ltd, Alderley Pk, Macclesfield SK10 4TG, Cheshire, England Redx Antiinfect Ltd, Alderley Pk, Mereside SK10 4TG, Cheshire, EnglandBlades, Kevin论文数: 0 引用数: 0 h-index: 0机构: Infex Therapeut Ltd, Alderley Pk, Macclesfield SK10 4TG, Cheshire, England Redx Antiinfect Ltd, Alderley Pk, Mereside SK10 4TG, Cheshire, EnglandOrr, David论文数: 0 引用数: 0 h-index: 0机构: Infex Therapeut Ltd, Alderley Pk, Macclesfield SK10 4TG, Cheshire, England Redx Antiinfect Ltd, Alderley Pk, Mereside SK10 4TG, Cheshire, EnglandDauncey, Elizabeth论文数: 0 引用数: 0 h-index: 0机构: Redx Antiinfect Ltd, Alderley Pk, Mereside SK10 4TG, Cheshire, England Redx Antiinfect Ltd, Alderley Pk, Mereside SK10 4TG, Cheshire, EnglandSmith, Oliver论文数: 0 引用数: 0 h-index: 0机构: Infex Therapeut Ltd, Alderley Pk, Macclesfield SK10 4TG, Cheshire, England Redx Antiinfect Ltd, Alderley Pk, Mereside SK10 4TG, Cheshire, EnglandDick, Emma论文数: 0 引用数: 0 h-index: 0机构: Redx Antiinfect Ltd, Alderley Pk, Mereside SK10 4TG, Cheshire, England Redx Antiinfect Ltd, Alderley Pk, Mereside SK10 4TG, Cheshire, EnglandWalker, Rolf论文数: 0 引用数: 0 h-index: 0机构: Redx Antiinfect Ltd, Alderley Pk, Mereside SK10 4TG, Cheshire, England Redx Antiinfect Ltd, Alderley Pk, Mereside SK10 4TG, Cheshire, EnglandMatthews, Teresa论文数: 0 引用数: 0 h-index: 0机构: Redx Antiinfect Ltd, Alderley Pk, Mereside SK10 4TG, Cheshire, England Redx Antiinfect Ltd, Alderley Pk, Mereside SK10 4TG, Cheshire, EnglandBunt, Adam论文数: 0 引用数: 0 h-index: 0机构: Infex Therapeut Ltd, Alderley Pk, Macclesfield SK10 4TG, Cheshire, England Redx Antiinfect Ltd, Alderley Pk, Mereside SK10 4TG, Cheshire, EnglandFinlayson, Jonathan论文数: 0 引用数: 0 h-index: 0机构: Redx Antiinfect Ltd, Alderley Pk, Mereside SK10 4TG, Cheshire, England Redx Antiinfect Ltd, Alderley Pk, Mereside SK10 4TG, Cheshire, EnglandMorrison, Ian论文数: 0 引用数: 0 h-index: 0机构: Redx Antiinfect Ltd, Alderley Pk, Mereside SK10 4TG, Cheshire, England Redx Antiinfect Ltd, Alderley Pk, Mereside SK10 4TG, Cheshire, EnglandSavage, Victoria J.论文数: 0 引用数: 0 h-index: 0机构: Infex Therapeut Ltd, Alderley Pk, Macclesfield SK10 4TG, Cheshire, England Redx Antiinfect Ltd, Alderley Pk, Mereside SK10 4TG, Cheshire, EnglandMoyo, Emmanuel论文数: 0 引用数: 0 h-index: 0机构: Infex Therapeut Ltd, Alderley Pk, Macclesfield SK10 4TG, Cheshire, England Redx Antiinfect Ltd, Alderley Pk, Mereside SK10 4TG, Cheshire, EnglandButler, Hayley S.论文数: 0 引用数: 0 h-index: 0机构: Redx Antiinfect Ltd, Alderley Pk, Mereside SK10 4TG, Cheshire, England Redx Antiinfect Ltd, Alderley Pk, Mereside SK10 4TG, Cheshire, EnglandNewman, Rebecca论文数: 0 引用数: 0 h-index: 0机构: Infex Therapeut Ltd, Alderley Pk, Macclesfield SK10 4TG, Cheshire, England Redx Antiinfect Ltd, Alderley Pk, Mereside SK10 4TG, Cheshire, EnglandOoi, Nicola论文数: 0 引用数: 0 h-index: 0机构: Infex Therapeut Ltd, Alderley Pk, Macclesfield SK10 4TG, Cheshire, England Redx Antiinfect Ltd, Alderley Pk, Mereside SK10 4TG, Cheshire, EnglandSmith, Andrew论文数: 0 引用数: 0 h-index: 0机构: Redx Antiinfect Ltd, Alderley Pk, Mereside SK10 4TG, Cheshire, England Redx Antiinfect Ltd, Alderley Pk, Mereside SK10 4TG, Cheshire, EnglandCharrier, Cedric论文数: 0 引用数: 0 h-index: 0机构: Redx Antiinfect Ltd, Alderley Pk, Mereside SK10 4TG, Cheshire, England Redx Antiinfect Ltd, Alderley Pk, Mereside SK10 4TG, Cheshire, EnglandRatcliffe, Andrew J.论文数: 0 引用数: 0 h-index: 0机构: Redx Antiinfect Ltd, Alderley Pk, Mereside SK10 4TG, Cheshire, England Redx Antiinfect Ltd, Alderley Pk, Mereside SK10 4TG, Cheshire, EnglandStokes, Neil R.论文数: 0 引用数: 0 h-index: 0机构: Redx Antiinfect Ltd, Alderley Pk, Mereside SK10 4TG, Cheshire, England Redx Antiinfect Ltd, Alderley Pk, Mereside SK10 4TG, Cheshire, EnglandBest, Stuart论文数: 0 引用数: 0 h-index: 0机构: Redx Antiinfect Ltd, Alderley Pk, Mereside SK10 4TG, Cheshire, England Redx Antiinfect Ltd, Alderley Pk, Mereside SK10 4TG, Cheshire, EnglandSalisbury, Anne-Marie论文数: 0 引用数: 0 h-index: 0机构: Redx Antiinfect Ltd, Alderley Pk, Mereside SK10 4TG, Cheshire, England Redx Antiinfect Ltd, Alderley Pk, Mereside SK10 4TG, Cheshire, EnglandCraighead, Mark论文数: 0 引用数: 0 h-index: 0机构: Redx Antiinfect Ltd, Alderley Pk, Mereside SK10 4TG, Cheshire, England Redx Antiinfect Ltd, Alderley Pk, Mereside SK10 4TG, Cheshire, EnglandCooper, Ian R.论文数: 0 引用数: 0 h-index: 0机构: Infex Therapeut Ltd, Alderley Pk, Macclesfield SK10 4TG, Cheshire, England Redx Antiinfect Ltd, Alderley Pk, Mereside SK10 4TG, Cheshire, England
- [5] Antibacterial activity of novel dual bacterial DNA type II topoisomerase inhibitorsPLOS ONE, 2020, 15 (02):D'Atanasio, Noemi论文数: 0 引用数: 0 h-index: 0机构: Angelini SpA, Angelini RR&D Regulatory Res & Dev, Rome, Italy Angelini SpA, Angelini RR&D Regulatory Res & Dev, Rome, Italyde Joannon, Alessandra Capezzone论文数: 0 引用数: 0 h-index: 0机构: Angelini SpA, Angelini RR&D Regulatory Res & Dev, Rome, Italy Angelini SpA, Angelini RR&D Regulatory Res & Dev, Rome, ItalyDi Sante, Laura论文数: 0 引用数: 0 h-index: 0机构: Polytech Univ Marche, Dept Life & Environm Sci, Ancona, Italy Angelini SpA, Angelini RR&D Regulatory Res & Dev, Rome, ItalyMangano, Giorgina论文数: 0 引用数: 0 h-index: 0机构: Angelini SpA, Angelini RR&D Regulatory Res & Dev, Rome, Italy Angelini SpA, Angelini RR&D Regulatory Res & Dev, Rome, ItalyOmbrato, Rosella论文数: 0 引用数: 0 h-index: 0机构: Angelini SpA, Angelini RR&D Regulatory Res & Dev, Rome, Italy Angelini SpA, Angelini RR&D Regulatory Res & Dev, Rome, ItalyVitiello, Marco论文数: 0 引用数: 0 h-index: 0机构: Angelini SpA, Angelini RR&D Regulatory Res & Dev, Rome, Italy Angelini SpA, Angelini RR&D Regulatory Res & Dev, Rome, ItalyBartella, Cristina论文数: 0 引用数: 0 h-index: 0机构: Angelini SpA, Angelini RR&D Regulatory Res & Dev, Rome, Italy Angelini SpA, Angelini RR&D Regulatory Res & Dev, Rome, ItalyMagaro, Gabriele论文数: 0 引用数: 0 h-index: 0机构: Angelini SpA, Angelini RR&D Regulatory Res & Dev, Rome, Italy Angelini SpA, Angelini RR&D Regulatory Res & Dev, Rome, ItalyPrati, Federica论文数: 0 引用数: 0 h-index: 0机构: Angelini SpA, Angelini RR&D Regulatory Res & Dev, Rome, Italy Angelini SpA, Angelini RR&D Regulatory Res & Dev, Rome, ItalyMilanese, Claudio论文数: 0 引用数: 0 h-index: 0机构: Angelini SpA, Angelini RR&D Regulatory Res & Dev, Rome, Italy Angelini SpA, Angelini RR&D Regulatory Res & Dev, Rome, ItalyVignaroli, Carla论文数: 0 引用数: 0 h-index: 0机构: Polytech Univ Marche, Dept Life & Environm Sci, Ancona, Italy Angelini SpA, Angelini RR&D Regulatory Res & Dev, Rome, ItalyDi Giorgio, Francesco Paolo论文数: 0 引用数: 0 h-index: 0机构: Angelini SpA, Angelini RR&D Regulatory Res & Dev, Rome, Italy Angelini SpA, Angelini RR&D Regulatory Res & Dev, Rome, ItalyTongiani, Serena论文数: 0 引用数: 0 h-index: 0机构: Angelini SpA, Angelini RR&D Regulatory Res & Dev, Rome, Italy Angelini SpA, Angelini RR&D Regulatory Res & Dev, Rome, Italy
- [6] Lead optimization of 8-(methylamino)-2-oxo-1,2-dihydroquinolines as bacterial type II topoisomerase inhibitorsBIOORGANIC & MEDICINAL CHEMISTRY, 2020, 28 (22)Ushiyama, Fumihito论文数: 0 引用数: 0 h-index: 0机构: Taisho Pharmaceut Co Ltd, Kita Ku, 1-403 Yoshino Cho, Saitama 3319530, Japan Taisho Pharmaceut Co Ltd, Kita Ku, 1-403 Yoshino Cho, Saitama 3319530, JapanAmada, Hideaki论文数: 0 引用数: 0 h-index: 0机构: Taisho Pharmaceut Co Ltd, Kita Ku, 1-403 Yoshino Cho, Saitama 3319530, Japan Taisho Pharmaceut Co Ltd, Kita Ku, 1-403 Yoshino Cho, Saitama 3319530, JapanMihara, Yasuhiro论文数: 0 引用数: 0 h-index: 0机构: Taisho Pharmaceut Co Ltd, Kita Ku, 1-403 Yoshino Cho, Saitama 3319530, Japan Taisho Pharmaceut Co Ltd, Kita Ku, 1-403 Yoshino Cho, Saitama 3319530, JapanTakeuchi, Tomoki论文数: 0 引用数: 0 h-index: 0机构: Taisho Pharmaceut Co Ltd, Kita Ku, 1-403 Yoshino Cho, Saitama 3319530, Japan Taisho Pharmaceut Co Ltd, Kita Ku, 1-403 Yoshino Cho, Saitama 3319530, JapanTanaka-Yamamoto, Nozomi论文数: 0 引用数: 0 h-index: 0机构: Taisho Pharmaceut Co Ltd, Kita Ku, 1-403 Yoshino Cho, Saitama 3319530, Japan Taisho Pharmaceut Co Ltd, Kita Ku, 1-403 Yoshino Cho, Saitama 3319530, JapanMima, Masashi论文数: 0 引用数: 0 h-index: 0机构: Taisho Pharmaceut Co Ltd, Kita Ku, 1-403 Yoshino Cho, Saitama 3319530, Japan Taisho Pharmaceut Co Ltd, Kita Ku, 1-403 Yoshino Cho, Saitama 3319530, JapanKamitani, Masafumi论文数: 0 引用数: 0 h-index: 0机构: Taisho Pharmaceut Co Ltd, Kita Ku, 1-403 Yoshino Cho, Saitama 3319530, Japan Taisho Pharmaceut Co Ltd, Kita Ku, 1-403 Yoshino Cho, Saitama 3319530, JapanWada, Reiko论文数: 0 引用数: 0 h-index: 0机构: Taisho Pharmaceut Co Ltd, Kita Ku, 1-403 Yoshino Cho, Saitama 3319530, Japan Taisho Pharmaceut Co Ltd, Kita Ku, 1-403 Yoshino Cho, Saitama 3319530, JapanTamura, Yunoshin论文数: 0 引用数: 0 h-index: 0机构: Taisho Pharmaceut Co Ltd, Kita Ku, 1-403 Yoshino Cho, Saitama 3319530, Japan Taisho Pharmaceut Co Ltd, Kita Ku, 1-403 Yoshino Cho, Saitama 3319530, JapanEndo, Mayumi论文数: 0 引用数: 0 h-index: 0机构: Taisho Pharmaceut Co Ltd, Kita Ku, 1-403 Yoshino Cho, Saitama 3319530, Japan Taisho Pharmaceut Co Ltd, Kita Ku, 1-403 Yoshino Cho, Saitama 3319530, JapanMasuko, Aiko论文数: 0 引用数: 0 h-index: 0机构: Taisho Pharmaceut Co Ltd, Kita Ku, 1-403 Yoshino Cho, Saitama 3319530, Japan Taisho Pharmaceut Co Ltd, Kita Ku, 1-403 Yoshino Cho, Saitama 3319530, JapanTakata, Iichiro论文数: 0 引用数: 0 h-index: 0机构: Taisho Pharmaceut Co Ltd, Kita Ku, 1-403 Yoshino Cho, Saitama 3319530, Japan Taisho Pharmaceut Co Ltd, Kita Ku, 1-403 Yoshino Cho, Saitama 3319530, JapanHitaka, Kosuke论文数: 0 引用数: 0 h-index: 0机构: Taisho Pharmaceut Co Ltd, Kita Ku, 1-403 Yoshino Cho, Saitama 3319530, Japan Taisho Pharmaceut Co Ltd, Kita Ku, 1-403 Yoshino Cho, Saitama 3319530, JapanSugiyama, Hiroyuki论文数: 0 引用数: 0 h-index: 0机构: Taisho Pharmaceut Co Ltd, Kita Ku, 1-403 Yoshino Cho, Saitama 3319530, Japan Taisho Pharmaceut Co Ltd, Kita Ku, 1-403 Yoshino Cho, Saitama 3319530, JapanOhtake, Norikazu论文数: 0 引用数: 0 h-index: 0机构: Taisho Pharmaceut Co Ltd, Kita Ku, 1-403 Yoshino Cho, Saitama 3319530, Japan Taisho Pharmaceut Co Ltd, Kita Ku, 1-403 Yoshino Cho, Saitama 3319530, Japan
- [7] Structure-based optimization of novel azepane derivatives as PKB inhibitorsJOURNAL OF MEDICINAL CHEMISTRY, 2004, 47 (06) : 1375 - 1390Breitenlechner, CB论文数: 0 引用数: 0 h-index: 0机构: Roch Diagnost GmbH, Pharma Res, D-82372 Penzberg, GermanyWegge, T论文数: 0 引用数: 0 h-index: 0机构: Roch Diagnost GmbH, Pharma Res, D-82372 Penzberg, GermanyBerillon, L论文数: 0 引用数: 0 h-index: 0机构: Roch Diagnost GmbH, Pharma Res, D-82372 Penzberg, GermanyGraul, K论文数: 0 引用数: 0 h-index: 0机构: Roch Diagnost GmbH, Pharma Res, D-82372 Penzberg, GermanyMarzenell, M论文数: 0 引用数: 0 h-index: 0机构: Roch Diagnost GmbH, Pharma Res, D-82372 Penzberg, GermanyFriebe, WG论文数: 0 引用数: 0 h-index: 0机构: Roch Diagnost GmbH, Pharma Res, D-82372 Penzberg, GermanyThomas, U论文数: 0 引用数: 0 h-index: 0机构: Roch Diagnost GmbH, Pharma Res, D-82372 Penzberg, GermanySchumacher, R论文数: 0 引用数: 0 h-index: 0机构: Roch Diagnost GmbH, Pharma Res, D-82372 Penzberg, GermanyHuber, R论文数: 0 引用数: 0 h-index: 0机构: Roch Diagnost GmbH, Pharma Res, D-82372 Penzberg, GermanyEngh, RA论文数: 0 引用数: 0 h-index: 0机构: Roch Diagnost GmbH, Pharma Res, D-82372 Penzberg, GermanyMasjost, B论文数: 0 引用数: 0 h-index: 0机构: Roch Diagnost GmbH, Pharma Res, D-82372 Penzberg, Germany
- [8] Nonpeptide inhibitors of cathepsin G: Optimization of a novel β-ketophosphonic acid lead by structure-based drug designJournal of the American Chemical Society, 2002, 124 (15): : 3810 - 3811Greco, Michael N.论文数: 0 引用数: 0 h-index: 0机构: Johnson and Johnson Pharmaceutical Research and Development, Spring House, PA 19477-0776, United StatesHawkins, Michael J.论文数: 0 引用数: 0 h-index: 0机构: Johnson and Johnson Pharmaceutical Research and Development, Spring House, PA 19477-0776, United StatesPowell, Eugene T.论文数: 0 引用数: 0 h-index: 0机构: Johnson and Johnson Pharmaceutical Research and Development, Spring House, PA 19477-0776, United StatesAlmond, Jr., Harold R.论文数: 0 引用数: 0 h-index: 0机构: Johnson and Johnson Pharmaceutical Research and Development, Spring House, PA 19477-0776, United StatesCorcoran, Thomas W.论文数: 0 引用数: 0 h-index: 0机构: Johnson and Johnson Pharmaceutical Research and Development, Spring House, PA 19477-0776, United StatesDe, Garavilla, Lawrence论文数: 0 引用数: 0 h-index: 0机构: Johnson and Johnson Pharmaceutical Research and Development, Spring House, PA 19477-0776, United StatesKauffman, Jack A.论文数: 0 引用数: 0 h-index: 0机构: Johnson and Johnson Pharmaceutical Research and Development, Spring House, PA 19477-0776, United StatesRecacha, Rosario论文数: 0 引用数: 0 h-index: 0机构: Johnson and Johnson Pharmaceutical Research and Development, Spring House, PA 19477-0776, United StatesChattopadhyay, Debashish论文数: 0 引用数: 0 h-index: 0机构: Johnson and Johnson Pharmaceutical Research and Development, Spring House, PA 19477-0776, United StatesAndrade-Gordon, Patricia论文数: 0 引用数: 0 h-index: 0机构: Johnson and Johnson Pharmaceutical Research and Development, Spring House, PA 19477-0776, United StatesMaryanoff, Bruce E.论文数: 0 引用数: 0 h-index: 0机构: Johnson and Johnson Pharmaceutical Research and Development, Spring House, PA 19477-0776, United States
- [9] Nonpeptide inhibitors of cathepsin G:: Optimization of a novel β-ketophosphonic acid lead by structure-based drug designJOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2002, 124 (15) : 3810 - 3811Greco, MN论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev, Spring House, PA 19477 USA Johnson & Johnson Pharmaceut Res & Dev, Spring House, PA 19477 USAHawkins, MJ论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev, Spring House, PA 19477 USAPowell, ET论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev, Spring House, PA 19477 USAAlmond, HR论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev, Spring House, PA 19477 USACorcoran, TW论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev, Spring House, PA 19477 USAde Garavilla, L论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev, Spring House, PA 19477 USAKauffman, JA论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev, Spring House, PA 19477 USARecacha, R论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev, Spring House, PA 19477 USAChattopadhyay, D论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev, Spring House, PA 19477 USAAndrade-Gordon, P论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev, Spring House, PA 19477 USAMaryanoff, BE论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev, Spring House, PA 19477 USA
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