Comparison of G-Protein Biased Mu Agonists to Partial and Full Mu Agonists in Measures of Thermal Antinociception, Respiratory Depression, and Drug Self-Administration in Male and Female SpragueDawley Rats

被引：0

作者：

Pham, Loc ^{[1
]}

Pareek, Tanya ^{[1
]}

Shabir, Tooba ^{[1
]}

Gilmore, Jackson ^{[1
]}

Le, Rose ^{[1
]}

Ladner, Alexandra ^{[1
]}

Araunjo, Aaron ^{[1
]}

Blough, Bruce ^{[2
]}

Freeman, Kevin ^{[1
]}

机构：

[1] Univ Mississippi, Med Ctr, Mississippi State, MS USA

[2] RTI Int, Waltham, MA USA

来源：

DRUG AND ALCOHOL DEPENDENCE | 2025年 / 267卷

关键词：

D O I：

10.1016/j.drugalcdep.2024.111699

中图分类号：

R194 [卫生标准、卫生检查、医药管理];

学科分类号：

摘要：

M105

引用

页码：123 / 124

页数：2

共 6 条

[1] Self-administration of G-protein biased mu opioid agonists in nonhuman primates
Paronis, Carol
George, Kristen E.
Bow, Eric W.
Gutman, Eugene S.
Sulima, Agnieszka
Rice, Kenner
Jacobson, Arthur
Bergman, Jack
JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS, 2023, 385
[2] Comparison of the reinforcing, antinociceptive, and respiratory depressant effects of prototypical and G-protein biased mu-opioid receptor agonists in male and female Sprague-Dawley rats
Zamarripa, C. Austin
Pareek, Tanya
Pham, Loc M.
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Vallender, Eric J.
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PSYCHOPHARMACOLOGY, 2024, 241 (12) : 2453 - 2469
[3] Some effects of putative G-protein biased mu-opioid receptor agonists in male rhesus monkeys
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BEHAVIOURAL PHARMACOLOGY, 2021, 32 (05): : 453 - 458
[4] Effect of reduced mu opioid receptor density on the relative efficacy of full and partial agonists for G-protein activation.
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[5] CHARACTERIZING BIASED MU-OPIOID RECEPTOR AGONISTS, PZM21 AND SR17018 IN SELF-ADMINISTRATION, AND WHOLE-PLETHYSMOGRAPHY IN RATS
Pham, Loc
Ladner, Alexandra
Araunjo, Aaron
Blough, Bruce
Freeman, Kevin
DRUG AND ALCOHOL DEPENDENCE, 2024, 260
[6] Effectiveness comparisons of G-protein biased and unbiased mu opioid receptor ligands in warm water tail-withdrawal and drug discrimination in male and female rats
Schwienteck, Kathryn L.
Faunce, Kaycee E.
Rice, Kenner C.
Obeng, Samuel
Zhang, Yan
Blough, Bruce E.
Grim, Travis W.
Negus, S. Stevens
Banks, Matthew L.
NEUROPHARMACOLOGY, 2019, 150 : 200 - 209

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