Prioritization of Eleven-Nineteen-Leukemia (ENL) inhibitors as orally available drug candidates for acute myeloid leukemia

被引:0
|
作者
Liu, Wenshe R.
Guo, Xuejiao
Alta, Sandeep
Xu, Shiqing
机构
关键词
D O I
10.1158/1538-8514.CANCERCHEM24-A013
中图分类号
R73 [肿瘤学];
学科分类号
100214 ;
摘要
A013
引用
收藏
页数:2
相关论文
共 50 条
  • [1] Prioritization of Eleven-Nineteen-Leukemia Inhibitors as Orally Available Drug Candidates for Acute Myeloid Leukemia
    Guo, Xuejiao Shirley
    Atla, Sandeep
    Nyalata, Satyanarayana
    Alugubelli, Yugendar R.
    Chen, Peng-Hsun Chase
    Xu, Shiqing
    Liu, Wenshe Ray
    JOURNAL OF MEDICINAL CHEMISTRY, 2024, 67 (22) : 20100 - 20117
  • [2] The eleven-nineteen-leukemia protein ENL connects nuclear MLL fusion partners with chromatin
    Zeisig, DT
    Bittner, CB
    Zeisig, BB
    García-Cuéllar, MP
    Hess, JL
    Slany, RK
    ONCOGENE, 2005, 24 (35) : 5525 - 5532
  • [3] The eleven-nineteen-leukemia protein ENL connects nuclear MLL fusion partners with chromatin
    Deniz T Zeisig
    Claudia B Bittner
    Bernd B Zeisig
    Maria-Paz García-Cuéllar
    Jay L Hess
    Robert K Slany
    Oncogene, 2005, 24 : 5525 - 5532
  • [4] Structure-Based Approach toward Identification of Inhibitory Fragments for Eleven-Nineteen-Leukemia Protein (ENL)
    Heidenreich, David
    Moustakim, Moses
    Schmidt, Jurema
    Merk, Daniel
    Brennan, Paul E.
    Fedorov, Oleg
    Chaikuad, Apirat
    Knapp, Stefan
    JOURNAL OF MEDICINAL CHEMISTRY, 2018, 61 (23) : 10929 - 10934
  • [5] Effective orally available drug combination of OR2100 and venetoclax in acute myeloid leukemia
    Ureshino, Hiroshi
    Watanabe, Tatsuro
    Kimura, Shinya
    CANCER SCIENCE, 2023, 114 : 44 - 44
  • [6] ENL: structure, function, and roles in hematopoiesis and acute myeloid leukemia
    Jianbiao Zhou
    Yvonne Ng
    Wee-Joo Chng
    Cellular and Molecular Life Sciences, 2018, 75 : 3931 - 3941
  • [7] ENL: structure, function, and roles in hematopoiesis and acute myeloid leukemia
    Zhou, Jianbiao
    Ng, Yvonne
    Chng, Wee-Joo
    CELLULAR AND MOLECULAR LIFE SCIENCES, 2018, 75 (21) : 3931 - 3941
  • [8] Conformational and Thermodynamic Differences Underlying Wild-Type and Mutant Eleven-Nineteen-Leukemia YEATS Domain Specificity for Epigenetic Marks
    Baweja, Lokesh
    Wereszczynski, Jeff
    JOURNAL OF CHEMICAL INFORMATION AND MODELING, 2023, 63 (04) : 1229 - 1238
  • [9] Checkpoint Inhibitors in Acute Myeloid Leukemia
    Damiani, Daniela
    Tiribelli, Mario
    BIOMEDICINES, 2023, 11 (06)
  • [10] HDAC Inhibitors in Acute Myeloid Leukemia
    San Jose-Eneriz, Edurne
    Gimenez-Camino, Naroa
    Agirre, Xabier
    Prosper, Felipe
    CANCERS, 2019, 11 (11)