A cascade indazolone-directed Ir(iii)- and Rh(iii)-catalyzed C(sp2)-H functionalization/[4 + 2] annulation of 1-arylindazolones with sulfoxonium ylides to access chemically divergent 8H-indazolo [1,2-a]cinnolines

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作者
Zheng, Yi-Chuan [1 ]
Shu, Bing [2 ]
Zeng, Yao-Fu [3 ]
Chen, Shao-Yong [1 ]
Song, Jia-Lin [1 ]
Liu, Yan-Zhi [1 ]
Xiao, Lin [1 ]
Liu, Xu-Ge [4 ]
Zhang, Xuanxuan [1 ]
Zhang, Shang-Shi [1 ]
机构
[1] Guangdong Provincial Key Laboratory of Advanced Drug Delivery Systems, Center for Drug Research and Development, Guangdong Pharmaceutical University, Guangzhou,510006, China
[2] School of Pharmacy, Guangdong Pharmaceutical University, Guangzhou,510006, China
[3] School of Pharmaceutical Science, Hunan Provincial Key Laboratory of Tumor Microenvironment Responsive Drug Research, Hengyang Medical School, University of South China, Hunan, Hengyang,421001, China
[4] School of Pharmacy, Henan University, Henan, Kaifeng,475004, China
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页码:5185 / 5190
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