共 6 条
- [1] A use-dependent blocker of Cav2.2 channel for neuropathic painACTA PHARMACOLOGICA SINICA, 2006, 27 : 6 - 6Kaneko, Shuji论文数: 0 引用数: 0 h-index: 0机构: Kyoto Univ, Dept Mol Pharmacol, Grad Sch Pharmaceut Sci, Kyoto 6068501, Japan Kyoto Univ, Dept Mol Pharmacol, Grad Sch Pharmaceut Sci, Kyoto 6068501, Japan
- [2] Discovery of a state-dependent Cav2.2 blocker for the treatment of chronic painABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2009, 238Hoyt, Scott B.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Dept Basic Chem, Rahway, NJ 07065 USA Merck & Co Inc, Dept Basic Chem, Rahway, NJ 07065 USALondon, Clare论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Dept Basic Chem, Rahway, NJ 07065 USA Merck & Co Inc, Dept Basic Chem, Rahway, NJ 07065 USAWeber, Ann E.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Dept Basic Chem, Rahway, NJ 07065 USA Merck & Co Inc, Dept Basic Chem, Rahway, NJ 07065 USAAbbadie, Catherine论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Dept Pharmacol, Rahway, NJ 07065 USA Merck & Co Inc, Dept Basic Chem, Rahway, NJ 07065 USAArneric, Stephen论文数: 0 引用数: 0 h-index: 0机构: Neuromed Pharmaceut, Vancouver, BC V6T 1Z3, Canada Merck & Co Inc, Dept Basic Chem, Rahway, NJ 07065 USABugianesi, Randal论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Dept Ion Channels, Rahway, NJ 07065 USA Merck & Co Inc, Dept Basic Chem, Rahway, NJ 07065 USAEduljee, Cyrus论文数: 0 引用数: 0 h-index: 0机构: Neuromed Pharmaceut, Vancouver, BC V6T 1Z3, Canada Merck & Co Inc, Dept Basic Chem, Rahway, NJ 07065 USAGreen, Mitchell论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Dept Drug Metab, Rahway, NJ 07065 USA Merck & Co Inc, Dept Basic Chem, Rahway, NJ 07065 USAHerrington, James论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Dept Ion Channels, Rahway, NJ 07065 USA Merck & Co Inc, Dept Basic Chem, Rahway, NJ 07065 USALi, Xiaohua论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Dept Basic Chem, Rahway, NJ 07065 USA Merck & Co Inc, Dept Basic Chem, Rahway, NJ 07065 USALyons, Kathryn A.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Dept Basic Chem, Rahway, NJ 07065 USA Merck & Co Inc, Dept Basic Chem, Rahway, NJ 07065 USAMakarewicz, Amanda论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Dept Basic Chem, Rahway, NJ 07065 USA Merck & Co Inc, Dept Basic Chem, Rahway, NJ 07065 USAMcGowan, Erin论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Dept Pharmacol, Rahway, NJ 07065 USA Merck & Co Inc, Dept Basic Chem, Rahway, NJ 07065 USAMcManus, Owen论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Dept Ion Channels, Rahway, NJ 07065 USA Merck & Co Inc, Dept Basic Chem, Rahway, NJ 07065 USAMistry, Shruti论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Dept Pharmacol, Rahway, NJ 07065 USA Merck & Co Inc, Dept Basic Chem, Rahway, NJ 07065 USAMorris, Judy论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Dept Basic Chem, Rahway, NJ 07065 USA Merck & Co Inc, Dept Basic Chem, Rahway, NJ 07065 USAPutrenko, Igor论文数: 0 引用数: 0 h-index: 0机构: Neuromed Pharmaceut, Vancouver, BC V6T 1Z3, Canada Merck & Co Inc, Dept Basic Chem, Rahway, NJ 07065 USARatliff', Kevin论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Dept Ion Channels, Rahway, NJ 07065 USA Merck & Co Inc, Dept Basic Chem, Rahway, NJ 07065 USASmith, McHardy论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Dept Ion Channels, Rahway, NJ 07065 USA Merck & Co Inc, Dept Basic Chem, Rahway, NJ 07065 USASnutch, Terrance论文数: 0 引用数: 0 h-index: 0机构: Neuromed Pharmaceut, Vancouver, BC V6T 1Z3, Canada Merck & Co Inc, Dept Basic Chem, Rahway, NJ 07065 USASun, Shu-Yu论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Dept Pharmacol, Rahway, NJ 07065 USA Merck & Co Inc, Dept Basic Chem, Rahway, NJ 07065 USASwensen, Andrew论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Dept Ion Channels, Rahway, NJ 07065 USA Merck & Co Inc, Dept Basic Chem, Rahway, NJ 07065 USATringham, Elizabeth论文数: 0 引用数: 0 h-index: 0机构: Neuromed Pharmaceut, Vancouver, BC V6T 1Z3, Canada Merck & Co Inc, Dept Basic Chem, Rahway, NJ 07065 USAWarren, Vivien论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Dept Ion Channels, Rahway, NJ 07065 USA Merck & Co Inc, Dept Basic Chem, Rahway, NJ 07065 USAWilliams, Brande论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Dept Ion Channels, Rahway, NJ 07065 USA Merck & Co Inc, Dept Basic Chem, Rahway, NJ 07065 USAKaczorowski, Gregory J.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Dept Ion Channels, Rahway, NJ 07065 USA Merck & Co Inc, Dept Basic Chem, Rahway, NJ 07065 USADuffy, Joseph L.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Dept Basic Chem, Rahway, NJ 07065 USA Merck & Co Inc, Dept Basic Chem, Rahway, NJ 07065 USA
- [3] A potent and selective indole N-type calcium channel (Cav2.2) blocker for the treatment of painBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2011, 21 (02) : 869 - 873Tyagarajan, Sriram论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAChakravarty, Prasun K.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAPark, Min论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAZhou, Bishan论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAHerrington, James B.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USARatliff, Kevin论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USABugianesi, Randall M.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAWilliams, Brande论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAHaedo, Rodolfo J.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USASwensen, Andrew M.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAWarren, Vivien A.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USASmith, McHardy论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAGarcia, Maria论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAKaczorowski, Gregory J.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAMcManus, Owen B.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USALyons, Kathryn A.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USALi, Xiaohua论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAMadeira, Maria论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAKaranam, Bindhu论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAGreen, Mitchell论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAForrest, Michael J.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAAbbadie, Catherine论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAMcGowan, Erin论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAMistry, Shruti论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAJochnowitz, Nina论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USADuffy, Joseph L.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA
- [4] Use-dependent blockade of Cav2.2 voltage-gated calcium channels for neuropathic painBIOCHEMICAL PHARMACOLOGY, 2005, 70 (04) : 489 - 499Winquist, RJ论文数: 0 引用数: 0 h-index: 0机构: Scion Pharmaceut Inc, Dept Pharmacol, Medford, MA 02155 USAPan, JQ论文数: 0 引用数: 0 h-index: 0机构: Scion Pharmaceut Inc, Dept Pharmacol, Medford, MA 02155 USAGribkoff, VK论文数: 0 引用数: 0 h-index: 0机构: Scion Pharmaceut Inc, Dept Pharmacol, Medford, MA 02155 USA
- [5] ZC88, a novel N-type calcium channel blocker from 4-amino-piperidine derivatives state-dependent inhibits Cav2.2 calcium channelsBRAIN RESEARCH, 2015, 1605 : 12 - 21Zhang, Shuzhuo论文数: 0 引用数: 0 h-index: 0机构: Beijing Inst Pharmacol & Toxicol, Beijing 100850, Peoples R China Beijing Inst Pharmacol & Toxicol, Beijing 100850, Peoples R ChinaYang, Lujia论文数: 0 引用数: 0 h-index: 0机构: Chinese Peoples Liberat Army Gen Hosp, Beijing 100853, Peoples R China Beijing Inst Pharmacol & Toxicol, Beijing 100850, Peoples R ChinaZhang, Kang论文数: 0 引用数: 0 h-index: 0机构: Beijing Inst Pharmacol & Toxicol, Beijing 100850, Peoples R China Beijing Inst Pharmacol & Toxicol, Beijing 100850, Peoples R ChinaLiu, Xiaoyan论文数: 0 引用数: 0 h-index: 0机构: Beijing Inst Pharmacol & Toxicol, Beijing 100850, Peoples R China Beijing Inst Pharmacol & Toxicol, Beijing 100850, Peoples R ChinaDai, Weiwei论文数: 0 引用数: 0 h-index: 0机构: Beijing Inst Pharmacol & Toxicol, Beijing 100850, Peoples R China Beijing Inst Pharmacol & Toxicol, Beijing 100850, Peoples R ChinaZhang, Cheng论文数: 0 引用数: 0 h-index: 0机构: Beijing Inst Pharmacol & Toxicol, Beijing 100850, Peoples R China Beijing Inst Pharmacol & Toxicol, Beijing 100850, Peoples R ChinaYong, Zheng论文数: 0 引用数: 0 h-index: 0机构: Beijing Inst Pharmacol & Toxicol, Beijing 100850, Peoples R China Beijing Inst Pharmacol & Toxicol, Beijing 100850, Peoples R ChinaLi, Jin论文数: 0 引用数: 0 h-index: 0机构: Beijing Inst Pharmacol & Toxicol, Beijing 100850, Peoples R China Beijing Inst Pharmacol & Toxicol, Beijing 100850, Peoples R ChinaZheng, Jianquan论文数: 0 引用数: 0 h-index: 0机构: Beijing Inst Pharmacol & Toxicol, Beijing 100850, Peoples R China Beijing Inst Pharmacol & Toxicol, Beijing 100850, Peoples R China
- [6] Anti-allodynic effect of 2-(aminomethyl)adamantane-1-carboxylic acid in a rat model of neuropathic pain: A mechanism dependent on CaV2.2 channel inhibitionBIOORGANIC & MEDICINAL CHEMISTRY, 2014, 22 (06) : 1797 - 1803Zoidis, Grigoris论文数: 0 引用数: 0 h-index: 0机构: Univ Athens, Dept Pharmaceut Chem, Fac Pharm, GR-15771 Athens, Greece Univ Athens, Dept Pharmaceut Chem, Fac Pharm, GR-15771 Athens, GreeceSandoval, Alejandro论文数: 0 引用数: 0 h-index: 0机构: Univ Nacl Autonoma Mexico, UNAM, Sch Med FES Iztacala, Tlalnepantla, Mexico Univ Athens, Dept Pharmaceut Chem, Fac Pharm, GR-15771 Athens, GreeceBaruch Pineda-Farias, Jorge论文数: 0 引用数: 0 h-index: 0机构: Ctr Invest & Estudios Avanzados Cinvesttav, Dept Farmacobiol, Mexico City, DF, Mexico Univ Athens, Dept Pharmaceut Chem, Fac Pharm, GR-15771 Athens, GreeceGranados-Soto, Vinicio论文数: 0 引用数: 0 h-index: 0机构: Ctr Invest & Estudios Avanzados Cinvesttav, Dept Farmacobiol, Mexico City, DF, Mexico Univ Athens, Dept Pharmaceut Chem, Fac Pharm, GR-15771 Athens, GreeceFelix, Ricardo论文数: 0 引用数: 0 h-index: 0机构: CINVESTAV, Dept Cell Biol, Mexico City 14000, DF, Mexico Univ Athens, Dept Pharmaceut Chem, Fac Pharm, GR-15771 Athens, Greece