[1] Tech Univ Carolo Wilhelmina Braunschweig, Inst Med & Pharmaceut Chem, Beethovenstr 55, D-38106 Braunschweig, Germany
[2] Bayer AG, Pharmaceut Lab 4, R&D, Bldg S106,231, D-13342 Berlin, Germany
[3] NUVISAN GmbH, Muellerstr 178, D-13353 Berlin, Germany
[4] AbbVie Deutschland GmbH & Co KG, Computat Drug Discovery, Knollstr, D-67061 Ludwigshafen, Germany
[5] Merck Healthcare KGaA, Frankfurter Str 250, D-64293 Darmstadt, Germany
[6] Sanofi R&D, Integrated Drug Discovery Ind Pk Hochst,Bldg G838, D-65926 Frankfurt, Germany
[7] Ludwig Maximilians Univ Munchen, Dept Pharm, Butenandtstr 5-13, D-81377 Munich, Germany
[8] Univ Tubingen, Inst Biomed Engn, Fac Med, Morgenstelle 8, D-72076 Tubingen, Germany
[9] Univ Tubingen, Inst Pharmaceut Sci, Pharmaceut Med Chem Dept, Morgenstelle 8, D-72076 Tubingen, Germany
[10] Univ Leipzig, Inst Drug Discovery, Fac Med, Bruderstr 34, D-04103 Leipzig, Germany