共 50 条
- [1] Preclinical characterization of LY3962673, an orally bioavailable, highly potent, and selective KRAS G12D inhibitorMOLECULAR CANCER THERAPEUTICS, 2023, 22 (12)Iyer, Chandrasekar论文数: 0 引用数: 0 h-index: 0Li, Binghui论文数: 0 引用数: 0 h-index: 0Stewart, Trent R.论文数: 0 引用数: 0 h-index: 0Wang, Tao论文数: 0 引用数: 0 h-index: 0Capen, Andrew论文数: 0 引用数: 0 h-index: 0Cavitt, Rachel论文数: 0 引用数: 0 h-index: 0Anderson, Bryan D.论文数: 0 引用数: 0 h-index: 0Bocchinfuso, Wayne论文数: 0 引用数: 0 h-index: 0Zhao, Gaiying论文数: 0 引用数: 0 h-index: 0Rodriguez, Michael J.论文数: 0 引用数: 0 h-index: 0Carballares, Santiago论文数: 0 引用数: 0 h-index: 0Cooke, Andrew论文数: 0 引用数: 0 h-index: 0Bondi, Robert论文数: 0 引用数: 0 h-index: 0Burns, Lee论文数: 0 引用数: 0 h-index: 0Kelamangalath, Lakshmi论文数: 0 引用数: 0 h-index: 0Wallace, Ross论文数: 0 引用数: 0 h-index: 0Kolakowski, Gabrielle论文数: 0 引用数: 0 h-index: 0Henry, James R.论文数: 0 引用数: 0 h-index: 0Si, Chong论文数: 0 引用数: 0 h-index: 0
- [2] MOONRAY-01, a phase 1 study of LY3962673, a potent, orally bioavailable, and selective KRAS G12D inhibitor in KRAS G12D-mutant solid tumorsJOURNAL OF CLINICAL ONCOLOGY, 2025, 43 (4_SUPPL) : TPS845 - TPS845Lakhani, Nehal J.论文数: 0 引用数: 0 h-index: 0机构: START Midwest, Grand Rapids, MI USAMelisi, Davide论文数: 0 引用数: 0 h-index: 0机构: START Midwest, Grand Rapids, MI USASubbiah, Vivek论文数: 0 引用数: 0 h-index: 0机构: START Midwest, Grand Rapids, MI USAAmmakkanavar, Natraj Reddy论文数: 0 引用数: 0 h-index: 0机构: START Midwest, Grand Rapids, MI USAO'Reilly, Eileen M.论文数: 0 引用数: 0 h-index: 0机构: START Midwest, Grand Rapids, MI USACassier, Philippe Alexandre论文数: 0 引用数: 0 h-index: 0机构: START Midwest, Grand Rapids, MI USAWainberg, Zev A.论文数: 0 引用数: 0 h-index: 0机构: START Midwest, Grand Rapids, MI USADuffy, Austin G.论文数: 0 引用数: 0 h-index: 0机构: START Midwest, Grand Rapids, MI USAPatnaik, Amita论文数: 0 引用数: 0 h-index: 0机构: START Midwest, Grand Rapids, MI USAFujiwara, Yutaka论文数: 0 引用数: 0 h-index: 0机构: START Midwest, Grand Rapids, MI USAOberstein, Paul Eliezer论文数: 0 引用数: 0 h-index: 0机构: START Midwest, Grand Rapids, MI USAGarcia-Carbonero, Rocio论文数: 0 引用数: 0 h-index: 0机构: START Midwest, Grand Rapids, MI USAWright, Jennifer论文数: 0 引用数: 0 h-index: 0机构: START Midwest, Grand Rapids, MI USALin, Aimee K.论文数: 0 引用数: 0 h-index: 0机构: START Midwest, Grand Rapids, MI USALi, Jian论文数: 0 引用数: 0 h-index: 0机构: START Midwest, Grand Rapids, MI USAAxelson, Michael D.论文数: 0 引用数: 0 h-index: 0机构: START Midwest, Grand Rapids, MI USAGarrido-Laguna, Ignacio论文数: 0 引用数: 0 h-index: 0机构: START Midwest, Grand Rapids, MI USA
- [3] INCB161734: A novel, potent, and orally bioavailable KRAS G12D selective inhibitor demonstrates antitumor activity in KRAS G12D mutant tumorsCANCER RESEARCH, 2024, 84 (06)Farren, Matthew R.论文数: 0 引用数: 0 h-index: 0Roman, Valerie论文数: 0 引用数: 0 h-index: 0Gallion, Alexandra论文数: 0 引用数: 0 h-index: 0Allali-Hassani, Abdellah论文数: 0 引用数: 0 h-index: 0Sokolsky, Alexander论文数: 0 引用数: 0 h-index: 0Kong, Weixi论文数: 0 引用数: 0 h-index: 0Smith, Amanda论文数: 0 引用数: 0 h-index: 0Wang, Hui论文数: 0 引用数: 0 h-index: 0Correa, Gina论文数: 0 引用数: 0 h-index: 0Deller, Marc论文数: 0 引用数: 0 h-index: 0Epling, Leslie B.论文数: 0 引用数: 0 h-index: 0Procak, Jessica论文数: 0 引用数: 0 h-index: 0Zhang, Guofeng论文数: 0 引用数: 0 h-index: 0Pecko, Katherine论文数: 0 引用数: 0 h-index: 0Kennedy, Keith论文数: 0 引用数: 0 h-index: 0Boer, Jason论文数: 0 引用数: 0 h-index: 0Kurzeja-Lipinski, Kerri论文数: 0 引用数: 0 h-index: 0Covington, Maryanne论文数: 0 引用数: 0 h-index: 0Chen, Kwang-Jong论文数: 0 引用数: 0 h-index: 0Wallower, Renee论文数: 0 引用数: 0 h-index: 0Rocha, Jennifer论文数: 0 引用数: 0 h-index: 0Pan, Rina论文数: 0 引用数: 0 h-index: 0Perry, Anthony论文数: 0 引用数: 0 h-index: 0Yuska, Brad论文数: 0 引用数: 0 h-index: 0Wang, Xiaozhao论文数: 0 引用数: 0 h-index: 0Macarron, Ricardo论文数: 0 引用数: 0 h-index: 0Kim, Sunkyu论文数: 0 引用数: 0 h-index: 0
- [4] Exploring the switch II pocket of KRAS(G12D) with mutant-selective monobody inhibitorsMOLECULAR CANCER RESEARCH, 2023, 21 (05)Hattori, Takamitsu论文数: 0 引用数: 0 h-index: 0机构: NYU Langone Hlth, New York, NY USA NYU Langone Hlth, New York, NY USAAkkapeddi, Padma论文数: 0 引用数: 0 h-index: 0机构: NYU Langone Hlth, New York, NY USA NYU Langone Hlth, New York, NY USAKhan, Imran论文数: 0 引用数: 0 h-index: 0机构: Med Univ South Carolina, Charleston, SC USA NYU Langone Hlth, New York, NY USAKoide, Akiko论文数: 0 引用数: 0 h-index: 0机构: NYU Langone Hlth, New York, NY USA NYU Langone Hlth, New York, NY USAGlasser, Eliezra论文数: 0 引用数: 0 h-index: 0机构: NYU Langone Hlth, New York, NY USA NYU Langone Hlth, New York, NY USAKetavarapu, Gayatri论文数: 0 引用数: 0 h-index: 0机构: NYU Langone Hlth, New York, NY USA NYU Langone Hlth, New York, NY USAWhaby, Michael论文数: 0 引用数: 0 h-index: 0机构: Med Univ South Carolina, Charleston, SC USA NYU Langone Hlth, New York, NY USAZuberi, Mariyam论文数: 0 引用数: 0 h-index: 0机构: Med Univ South Carolina, Charleston, SC USA NYU Langone Hlth, New York, NY USATeng, Kai Wen论文数: 0 引用数: 0 h-index: 0机构: NYU Langone Hlth, New York, NY USA NYU Langone Hlth, New York, NY USALefler, Julia论文数: 0 引用数: 0 h-index: 0机构: Med Univ South Carolina, Charleston, SC USA NYU Langone Hlth, New York, NY USAMaso, Lorenzo论文数: 0 引用数: 0 h-index: 0机构: NYU Langone Hlth, New York, NY USA NYU Langone Hlth, New York, NY USABang, Injin论文数: 0 引用数: 0 h-index: 0机构: NYU Langone Hlth, New York, NY USA NYU Langone Hlth, New York, NY USAOstrowski, Michael C.论文数: 0 引用数: 0 h-index: 0机构: Med Univ South Carolina, Charleston, SC USA NYU Langone Hlth, New York, NY USAO'Bryan, John P.论文数: 0 引用数: 0 h-index: 0机构: Med Univ South Carolina, Charleston, SC USA NYU Langone Hlth, New York, NY USAKoide, Shohei论文数: 0 引用数: 0 h-index: 0机构: NYU Langone Hlth, New York, NY USA NYU Langone Hlth, New York, NY USA
- [5] ASP3082, a First-in-class novel KRAS G12D degrader, exhibits remarkable anti-tumor activity in KRAS G12D mutated cancer modelsEUROPEAN JOURNAL OF CANCER, 2022, 174 : S30 - S30Nagashima, T.论文数: 0 引用数: 0 h-index: 0机构: Astellas Pharma Inc, Targeted Prot Degradat, Tsukuba, Ibaraki, Japan Astellas Pharma Inc, Targeted Prot Degradat, Tsukuba, Ibaraki, JapanInamura, K.论文数: 0 引用数: 0 h-index: 0机构: Astellas Pharma Inc, Targeted Prot Degradat, Tsukuba, Ibaraki, Japan Astellas Pharma Inc, Targeted Prot Degradat, Tsukuba, Ibaraki, JapanNishizono, Y.论文数: 0 引用数: 0 h-index: 0机构: Astellas Pharma Inc, Targeted Prot Degradat, Tsukuba, Ibaraki, Japan Astellas Pharma Inc, Targeted Prot Degradat, Tsukuba, Ibaraki, JapanSuzuki, A.论文数: 0 引用数: 0 h-index: 0机构: Astellas Pharma Inc, Immuno Oncol, Tsukuba, Ibaraki, Japan Astellas Pharma Inc, Targeted Prot Degradat, Tsukuba, Ibaraki, JapanTanaka, H.论文数: 0 引用数: 0 h-index: 0机构: Astellas Pharma Inc, Targeted Prot Degradat, Tsukuba, Ibaraki, Japan Astellas Pharma Inc, Targeted Prot Degradat, Tsukuba, Ibaraki, JapanYoshinari, T.论文数: 0 引用数: 0 h-index: 0机构: Astellas Pharma Inc, Targeted Prot Degradat, Tsukuba, Ibaraki, Japan Astellas Pharma Inc, Targeted Prot Degradat, Tsukuba, Ibaraki, JapanYamanaka, Y.论文数: 0 引用数: 0 h-index: 0机构: Astellas Pharma Inc, Appl Res & Operat, Tsukuba, Ibaraki, Japan Astellas Pharma Inc, Targeted Prot Degradat, Tsukuba, Ibaraki, Japan
- [6] GFH375 (VS-7375): An oral, selective KRAS G12D (ON/ OFF) inhibitor with potent anti-tumor efficacyCANCER RESEARCH, 2024, 84 (06)Yan, Feng论文数: 0 引用数: 0 h-index: 0Jiang, Tao论文数: 0 引用数: 0 h-index: 0Liang, Tao论文数: 0 引用数: 0 h-index: 0Cai, Lijian论文数: 0 引用数: 0 h-index: 0Zhang, Leitao论文数: 0 引用数: 0 h-index: 0Xu, Xiaoming论文数: 0 引用数: 0 h-index: 0Zhao, Yanhui论文数: 0 引用数: 0 h-index: 0Lan, Xiaoling论文数: 0 引用数: 0 h-index: 0Zhang, Xiaohui论文数: 0 引用数: 0 h-index: 0Liu, Meng论文数: 0 引用数: 0 h-index: 0Liu, Qiang论文数: 0 引用数: 0 h-index: 0Gao, Jinting论文数: 0 引用数: 0 h-index: 0Xie, Fubo论文数: 0 引用数: 0 h-index: 0Gao, Xueyan论文数: 0 引用数: 0 h-index: 0Wang, Li论文数: 0 引用数: 0 h-index: 0Zhang, Jingyang论文数: 0 引用数: 0 h-index: 0Ren, Hongcan论文数: 0 引用数: 0 h-index: 0Liu, Dong论文数: 0 引用数: 0 h-index: 0Le, Siyuan论文数: 0 引用数: 0 h-index: 0Tang, Lili论文数: 0 引用数: 0 h-index: 0Coma, Silvia论文数: 0 引用数: 0 h-index: 0Cheng, Yaofeng论文数: 0 引用数: 0 h-index: 0Sanburn, Nathan论文数: 0 引用数: 0 h-index: 0Pachter, Jonathan A.论文数: 0 引用数: 0 h-index: 0Zhou, Fusheng论文数: 0 引用数: 0 h-index: 0Lan, Jiong论文数: 0 引用数: 0 h-index: 0Lu, Qiang论文数: 0 引用数: 0 h-index: 0
- [7] Mutant-selective, covalent inhibitors of K-Ras(G12D)CANCER RESEARCH, 2024, 84 (02)Zheng, Qinheng论文数: 0 引用数: 0 h-index: 0Zhang, Ziyang论文数: 0 引用数: 0 h-index: 0Guiley, Keelan论文数: 0 引用数: 0 h-index: 0Shokat, Kevan论文数: 0 引用数: 0 h-index: 0
- [8] Discovery of SHR1127, an orally bioavailable, highly potent and selective KRAS G12D inhibitorCANCER RESEARCH, 2024, 84 (06)Li, Xin论文数: 0 引用数: 0 h-index: 0Shen, Feng论文数: 0 引用数: 0 h-index: 0Zhang, Limin论文数: 0 引用数: 0 h-index: 0Wang, Wei论文数: 0 引用数: 0 h-index: 0Kong, Luyao论文数: 0 引用数: 0 h-index: 0Bao, Yong论文数: 0 引用数: 0 h-index: 0Mao, Yuchang论文数: 0 引用数: 0 h-index: 0Wang, Zaiyong论文数: 0 引用数: 0 h-index: 0Lin, Sophie论文数: 0 引用数: 0 h-index: 0Zhang, Zhe论文数: 0 引用数: 0 h-index: 0Feng, Jun论文数: 0 引用数: 0 h-index: 0Hu, Min论文数: 0 引用数: 0 h-index: 0He, Feng论文数: 0 引用数: 0 h-index: 0
- [9] ALTA3263: an oral, KRAS isoform-selective, dual ON/OFF state, non-covalent inhibitor induces regressions across KRAS G12V, G12D, and G12C cancer modelsEUROPEAN JOURNAL OF CANCER, 2024, 211 : S5 - S6Wang, T.论文数: 0 引用数: 0 h-index: 0机构: Alterome Therapeut Inc, Discovery Biol, San Diego, CA USA Alterome Therapeut Inc, Discovery Biol, San Diego, CA USAIbanez, M.论文数: 0 引用数: 0 h-index: 0机构: Alterome Therapeut Inc, Discovery Biol, San Diego, CA USA Alterome Therapeut Inc, Discovery Biol, San Diego, CA USAYu, K.论文数: 0 引用数: 0 h-index: 0机构: Alterome Therapeut Inc, Discovery Biol, San Diego, CA USA Alterome Therapeut Inc, Discovery Biol, San Diego, CA USAFan, K.论文数: 0 引用数: 0 h-index: 0机构: Alterome Therapeut Inc, Discovery Biol, San Diego, CA USA Alterome Therapeut Inc, Discovery Biol, San Diego, CA USAJuan, J.论文数: 0 引用数: 0 h-index: 0机构: Alterome Therapeut Inc, Discovery Biol, San Diego, CA USA Alterome Therapeut Inc, Discovery Biol, San Diego, CA USAPerez, M.论文数: 0 引用数: 0 h-index: 0机构: Alterome Therapeut Inc, Discovery Biol, San Diego, CA USA Alterome Therapeut Inc, Discovery Biol, San Diego, CA USASmith, T.论文数: 0 引用数: 0 h-index: 0机构: Alterome Therapeut Inc, Discovery Biol, San Diego, CA USA Alterome Therapeut Inc, Discovery Biol, San Diego, CA USAWalsh, B.论文数: 0 引用数: 0 h-index: 0机构: Alterome Therapeut Inc, Discovery Biol, San Diego, CA USA Alterome Therapeut Inc, Discovery Biol, San Diego, CA USAKang, V.论文数: 0 引用数: 0 h-index: 0机构: Alterome Therapeut Inc, Discovery Biol, San Diego, CA USA Alterome Therapeut Inc, Discovery Biol, San Diego, CA USATyhonas, J.论文数: 0 引用数: 0 h-index: 0机构: Alterome Therapeut Inc, Discovery Biol, San Diego, CA USA Alterome Therapeut Inc, Discovery Biol, San Diego, CA USAAlvarez, N.论文数: 0 引用数: 0 h-index: 0机构: Alterome Therapeut Inc, Discovery Biol, San Diego, CA USA Alterome Therapeut Inc, Discovery Biol, San Diego, CA USATran, J.论文数: 0 引用数: 0 h-index: 0机构: Alterome Therapeut Inc, Discovery Biol, San Diego, CA USA Alterome Therapeut Inc, Discovery Biol, San Diego, CA USAMoorefield, K. S.论文数: 0 引用数: 0 h-index: 0机构: Alterome Therapeut Inc, Discovery Biol, San Diego, CA USA Alterome Therapeut Inc, Discovery Biol, San Diego, CA USAPhimister, A.论文数: 0 引用数: 0 h-index: 0机构: Alterome Therapeut Inc, Discovery Biol, San Diego, CA USA Alterome Therapeut Inc, Discovery Biol, San Diego, CA USAZhu, X.论文数: 0 引用数: 0 h-index: 0机构: Alterome Therapeut Inc, Discovery Biol, San Diego, CA USA Alterome Therapeut Inc, Discovery Biol, San Diego, CA USAChi, A.论文数: 0 引用数: 0 h-index: 0机构: Alterome Therapeut Inc, Discovery Biol, San Diego, CA USA Alterome Therapeut Inc, Discovery Biol, San Diego, CA USABartberger, M. D.论文数: 0 引用数: 0 h-index: 0机构: Alterome Therapeut Inc, Discovery Biol, San Diego, CA USA Alterome Therapeut Inc, Discovery Biol, San Diego, CA USAMurphy, E.论文数: 0 引用数: 0 h-index: 0机构: Alterome Therapeut Inc, Discovery Biol, San Diego, CA USA Alterome Therapeut Inc, Discovery Biol, San Diego, CA USA
- [10] Structure-Based Design and Synthesis of Potent and Selective KRAS G12D InhibitorsACS MEDICINAL CHEMISTRY LETTERS, 2023, 14 (10): : 1351 - 1357Cheng, Hengmiao论文数: 0 引用数: 0 h-index: 0机构: Erasca Inc, San Diego, CA 92121 USA Erasca Inc, San Diego, CA 92121 USALi, Puhui论文数: 0 引用数: 0 h-index: 0机构: Erasca Inc, San Diego, CA 92121 USA Erasca Inc, San Diego, CA 92121 USAChen, Ping论文数: 0 引用数: 0 h-index: 0机构: Erasca Inc, San Diego, CA 92121 USA Erasca Inc, San Diego, CA 92121 USAIrimia, Adriana论文数: 0 引用数: 0 h-index: 0机构: Erasca Inc, San Diego, CA 92121 USA Erasca Inc, San Diego, CA 92121 USABae, Jae Hyun论文数: 0 引用数: 0 h-index: 0机构: Erasca Inc, San Diego, CA 92121 USA Erasca Inc, San Diego, CA 92121 USABrooun, Alexei论文数: 0 引用数: 0 h-index: 0机构: Erasca Inc, San Diego, CA 92121 USA Erasca Inc, San Diego, CA 92121 USAFagan, Patrick论文数: 0 引用数: 0 h-index: 0机构: Erasca Inc, San Diego, CA 92121 USA Erasca Inc, San Diego, CA 92121 USALam, Richard论文数: 0 引用数: 0 h-index: 0机构: Erasca Inc, San Diego, CA 92121 USA Erasca Inc, San Diego, CA 92121 USALin, Bingzhen论文数: 0 引用数: 0 h-index: 0机构: Erasca Inc, San Diego, CA 92121 USA Erasca Inc, San Diego, CA 92121 USAZhang, Jingchuan论文数: 0 引用数: 0 h-index: 0机构: Erasca Inc, San Diego, CA 92121 USA Erasca Inc, San Diego, CA 92121 USAZhan, Xuejun论文数: 0 引用数: 0 h-index: 0机构: Wuxi AppTec Wuhan Co Ltd, Wuhan 430075, Hubei, Peoples R China Erasca Inc, San Diego, CA 92121 USAWu, Xu论文数: 0 引用数: 0 h-index: 0机构: Wuxi AppTec Wuhan Co Ltd, Wuhan 430075, Hubei, Peoples R China Erasca Inc, San Diego, CA 92121 USAXie, Nan论文数: 0 引用数: 0 h-index: 0机构: Wuxi AppTec Shanghai Co Ltd, Shanghai 200131, Peoples R China Erasca Inc, San Diego, CA 92121 USAChiang, Gary论文数: 0 引用数: 0 h-index: 0机构: Erasca Inc, San Diego, CA 92121 USA Erasca Inc, San Diego, CA 92121 USAShoemaker, Robert论文数: 0 引用数: 0 h-index: 0机构: Erasca Inc, San Diego, CA 92121 USA Erasca Inc, San Diego, CA 92121 USAVernier, Jean-Michel论文数: 0 引用数: 0 h-index: 0机构: Erasca Inc, San Diego, CA 92121 USA Erasca Inc, San Diego, CA 92121 USA