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- [6] DEVELOPMENT OF A NOVEL SERIES OF STYRYLQUINOLINE COMPOUNDS AS HIGH-AFFINITY LEUKOTRIENE-D4 RECEPTOR ANTAGONISTS - SYNTHETIC AND STRUCTURE ACTIVITY STUDIES LEADING TO THE DISCOVERY OF (+/-)-3-[[[3-[2-(7-CHLORO-2-QUINOLINYL)-(E)-ETHENYL]PHENYL][[3-(DIMETHYLAMINO)-3-OXOPROPYL]THIO]METHYL]THIO]PROPIONIC ACID JOURNAL OF MEDICINAL CHEMISTRY, 1992, 35 (21) : 3832 - 3844
- [9] STEREOSPECIFIC SYNTHESIS, ASSIGNMENT OF ABSOLUTE-CONFIGURATION, AND BIOLOGICAL-ACTIVITY OF THE ENANTIOMERS OF 3-[[[3-[2-(7-CHLOROQUINOLIN-2-YL)-(E)-ETHENYL]PHENYL][[3-(DIMETHYLAMINO)-3-OXOPROPYL]THIO]METHYL]THIO]PROPIONIC ACID, A POTENT AND SPECIFIC LEUKOTRIENE-D4 RECEPTOR ANTAGONIST JOURNAL OF MEDICINAL CHEMISTRY, 1990, 33 (10) : 2841 - 2845