SYNTHESIS OF PYRAZOLE-1-CARBON-1,8-NAPHTHYRIDINES AS ANTIMICROBIAL AGENTS

被引：0
|
作者：
RAO, JS
SREENIVASULU, B
MOGILAIAH, K
机构：
[1] KAKATIYA UNIV, DEPT CHEM, WARANGAL 506009, ANDHRA PRADESH, INDIA
[2] UNIV WARANGAL, COLL ARTS & SCI, DEPT CHEM, WARANGAL 506001, ANDHRA PRADESH, INDIA
来源：
INDIAN JOURNAL OF CHEMISTRY SECTION B-ORGANIC CHEMISTRY INCLUDING MEDICINAL CHEMISTRY | 1995年 / 34卷 / 08期
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D O I：
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中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
Condensation of 2-methyl-1,8-naphthyridine-3-carboxolic acid hydrazide (2) with different acetophenones affords the corresponding acetophenone 2-methyl-1,8-naphthyridine-3-carbonylhydrazones (3), which on treatment with POCl3 and DMF furnish the title compound 3-(3-aryl- 4-formylpyrazole-1-carbonyl)- 2-methyl-1,8-naphthyridines (4). Some of the compounds have shown antifungal and antibacterial activities.
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页码：734 / 735
页数：2
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