AN IMPROVED SYNTHESIS OF 4-[3-(TRIFLUOROMETHYL)-3H-DIAZIRIN-3-YL]BENZOIC ACID FOR PHOTOAFFINITY-LABELING

被引：22

作者：

HATANAKA, Y

NAKAYAMA, H

KANAOKA, Y

机构：

[1] HOKKAIDO UNIV,FAC PHARMACEUT SCI,SAPPORO,HOKKAIDO 060,JAPAN

[2] TOYAMA WOMENS COLL,TOYAMA 93001,JAPAN

来源：

HETEROCYCLES | 1993年 / 35卷 / 02期

关键词：

D O I：

10.3987/COM-92-S(T)93

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

An improved synthesis of 4-[3-(trifluoromethyl)-3H-diazirin-3-yl]benzoic acid, a key carbene precursor for photoaffinity labeling, was described. A new diazirine with amino group as a connective part was designed.

引用

页码：997 / 1004

页数：8

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