Tandem AN-AN reactions in the synthesis of tetrahydrothiazolo[4,5-e][1,2,4]triazines

被引：2

作者：

Mochulskaya, Nataliya N. ^{[1
,2
]}

Slepukhin, Pavel A. ^{[1
,2
]}

Charushin, Valery N. ^{[1
,2
]}

Kodess, Mikhail I. ^{[1
,2
]}

机构：

[1] Ural Fed Univ, Dept Chem, Ekaterinburg 620002, Russia

[2] Russian Acad Sci, Ural Branch, I Ya Postovsky Inst Organ Synth, Ekaterinburg 620041, Russia

来源：

MENDELEEV COMMUNICATIONS | 2016年 / 26卷 / 05期

基金：

俄罗斯科学基金会;

关键词：

1,2,4-TRIAZINES; CHEMISTRY;

D O I：

10.1016/j.mencom.2016.09.002

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

Reaction of 3-aryl-1,2,4-triazines with S,N-dinucleophilic N-(het)arylthioureas in acetic anhydride at room temperature affords the cyclization products, tetrahydrothiazolo[4,5-e][1,2,4]triazines in good yields. The structure of the heterocyclic system thus formed was confirmed by X-ray diffraction analysis.

引用

页码：375 / 377

页数：3

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